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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:369/41  |  提交时间:2017/12/18
Click Glycosylation for the Synthesis of 1,2,3-Triazole-Linked Picropodophyllotoxin Glycoconjugates and Their Anticancer Activity 期刊论文
CHEMISTRYSELECT, 2017, 卷号: 2, 期号: 18, 页码: 5038-5044
作者:  Zi, Cheng-Ting;  Yang, Liu;  Gao, Wei;  Li, Yan;  Zhou, Jun;  Ding, Zhong-Tao;  Hu, Jiang-Miao;  Jiang, Zi-Hua
浏览  |  Adobe PDF(3775Kb)  |  收藏  |  浏览/下载:214/44  |  提交时间:2017/10/23
Anticancer Activity  Cu(i)-catalyzed Click Reaction  Glycoconjugates  Picropodophyllotoxin  Podophyllotoxin  
Natural and Semisynthetic Tigliane Diterpenoids with New Carbon Skeletons from Euphorbia dracunculoides as a Wnt Signaling Pathway Inhibitor 期刊论文
ORGANIC LETTERS, 2017, 卷号: 19, 期号: 14, 页码: 3911-3914
作者:  Wang, Li;  Yang, Jing;  Kong, Ling-Mei;  Deng, Jun;  Xiong, Zijun;  Huang, Jianping;  Luo, Jianping;  Yan, Yijun;  Hu, Yikao;  Li, Xiao-Nian;  Li, Yan;  Zhao, Yong;  Huang, Sheng-Xiong
浏览  |  Adobe PDF(1338Kb)  |  收藏  |  浏览/下载:262/75  |  提交时间:2017/10/23
Protein-kinase-c  Phorbol Esters  Biological Evaluation  Biosynthesis  (+)-phorbol  Analogs  Cancer  Seeds  
Synthesis and Cytotoxic Activity of Novel Hybrid Compounds between Indolo[b]tetrahydrofuran and Imidazolium Salts 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 6, 页码: 1506-1515
作者:  Liu Zhengfen;  Zhang Chaobo;  Duan Shengzu;  Liu Yang;  Chen Wen;  Li Yan;  Zhang Hongbin;  Yang Xiaodong
浏览  |  Adobe PDF(1186Kb)  |  收藏  |  浏览/下载:196/40  |  提交时间:2017/10/23
Indolo[b]Tetrahydrofuran  Imidazolium Salts  Hybrid Compound  Cytotoxic Activity  
Lanostane-type triterpenoids from Kadsura coccinea 期刊论文
TETRAHEDRON, 2017, 卷号: 73, 期号: 20, 页码: 2931-2937
作者:  Hu, Zheng-Xi;  Li, Xiao-Nian;  Shi, Yi-Ming;  Wang, Wei-Guang;  Du, Xue;  Li, Yan;  Zhang, Yong-Hui;  Pu, Jian-Xin;  Sun, Han-Dong
浏览  |  Adobe PDF(860Kb)  |  收藏  |  浏览/下载:767/235  |  提交时间:2017/07/10
Kadsura Coccinea  Lanostane-type Triterpenoids  Cytotoxicity  
USP7 inhibitor P5091 inhibits Wnt signaling and colorectal tumor growth 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2017, 卷号: 131, 期号: 1, 页码: 29-39
作者:  An, Tao;  Gong, Yaxiao;  Li, Xue;  Kong, Lingmei;  Ma, Pengcheng;  Gong, Liang;  Zhu, Huifang;  Yu, Chunlei;  Liu, Jianmei;  Zhou, Hongyu;  Mao, Bingyu;  Li, Yan
浏览  |  Adobe PDF(3138Kb)  |  收藏  |  浏览/下载:779/143  |  提交时间:2017/04/06
Usp7 Inhibitor  Wnt Signaling  Colorectal Cancer  
Discovery of new dual binding TNKS inhibitors of Wnt signaling inhibition by pharmacophore modeling, molecular docking and bioassay 期刊论文
MOLECULAR BIOSYSTEMS, 2017, 卷号: 13, 期号: 2, 页码: 363-370
作者:  Pu, Yinglan;  Zhang, Shuqun;  Chang, Zhe;  Zhang, Yunqin;  Wang, Dong;  Zhang, Li;  Li, Yan;  Zuo, Zhili
浏览  |  Adobe PDF(972Kb)  |  收藏  |  浏览/下载:677/116  |  提交时间:2017/05/19
Star-PAP, a poly(A) polymerase, functions as a tumor suppressor in an orthotopic human breast cancer model 期刊论文
CELL DEATH & DISEASE, 2017, 卷号: 8, 期号: 1, 页码: e2582
作者:  Yu, C.;  Gong, Y.;  Zhou, H.;  Wang, M.;  Kong, L.;  Liu, J.;  An, T.;  Zhu, H.;  Li, Y.
浏览  |  Adobe PDF(3022Kb)  |  收藏  |  浏览/下载:191/39  |  提交时间:2017/04/19
Ent-Abietanoids Isolated from Isodon serra 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 2, 页码: 309
作者:  Wan, Jun;  Jiang, Hua-Yi;  Tang, Jian-Wei;  Li, Xing-Ren;  Du, Xue;  Li, Yan;  Sun, Han-Dong;  Pu, Jian-Xin
浏览  |  Adobe PDF(821Kb)  |  收藏  |  浏览/下载:652/113  |  提交时间:2017/05/19
Isodon Serra  Ent-abietane Diterpenoids  Anti-inflammation  Cytotoxicity  
ent-Kaurene diterpenoids from Isodon phyllostachys 期刊论文
TETRAHEDRON LETTERS, 2017, 卷号: 58, 期号: 4, 页码: 349-351
作者:  Yang, Jin;  Wang, Wei-Guang;  Wu, Hai-Yan;  Liu, Miao;  Jiang, Hua-Yi;  Du, Xue;  Li, Yan;  Pu, Jian-Xin;  Sun, Han-Dong
浏览  |  Adobe PDF(532Kb)  |  收藏  |  浏览/下载:425/55  |  提交时间:2017/04/17
Isodon Phyllostachys  Diterpenoid  Ent-kaurene