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Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:  Chen, Duo-zhi;  Yang, Bi-juan;  He, Xiao-li;  Fan, Shi-rui;  Cai, Jie-yun;  Jing, Chen-xu;  Zhang, Heng;  Zhang, Yu;  Li, Lin;  Hao, Xiao-jiang
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Wnt/beta-catenin signalling pathway agonist  Phenanthridine derivatives  Structural optimization  Structure-activity relationships (SARs)  
Acetyl-macrocalin B suppresses tumor growth in esophageal squamous cell carcinoma and exhibits synergistic anti-cancer effects with the Chk1/2 inhibitor AZD7762 期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2019, 卷号: 365, 页码: 71-83
作者:  Wang, Jing-Nan;  Che, Yun;  Yuan, Zu-Yang;  Lu, Zhi-Liang;  Li, Yuan;  Zhang, Zhi-Rong;  Li, Ning;  Li, Ren-Da;  Wan, Jun;  Sun, Han-Dong;  Sun, Nan;  Puno, Pema-Tenzin;  He, Jie
浏览  |  Adobe PDF(3457Kb)  |  收藏  |  浏览/下载:320/72  |  提交时间:2019/03/18
Acetyl-macrocalin B  Reactive oxygen species  p38 MAPK  Chk1/Chk2  Esophageal squamous cell carcinoma  
Synthesis, structure activity relationship and in vitro anti-influenza virus activity of novel polyphenol-pentacyclic triterpene conjugates 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 560-568
作者:  Li, Haiwei;  Li, Man;  Xu, Renyang;  Wang, Shouxin;  Zhang, Yongmin;  Zhang, Lihe;  Zhou, Demin;  Xiao, Sulong
浏览  |  Adobe PDF(1830Kb)  |  收藏  |  浏览/下载:227/30  |  提交时间:2019/03/25
Influenza virus  Pentacyclic triterpene  Polyphenol  Entry inhibitor  Hemagglutinin  
Naphthomycin-derived macrolactams with two new carbon skeletons from endophytic Streptomyces 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 2, 页码: 177-182
作者:  Zhang, Zhouxin;  Cao, Pei;  Shang, Ning-Ning;  Yang, Jing;  Wang, Li;  Yan, Yijun;  Huang, Sheng-Xiong
浏览  |  Adobe PDF(990Kb)  |  收藏  |  浏览/下载:219/41  |  提交时间:2019/03/18
Maoeriocalysins A-D, four novel ent-kaurane diterpenoids from Isodon eriocalyx and their structure determination utilizing quantum chemical calculation in conjunction with quantitative interproton distance analysis 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 1, 页码: 45-53
作者:  Yang, Qian;  Hu, Kun;  Yan, Bing-Chao;  Liu, Miao;  Li, Xiao-Nian;  Sun, Han-Dong;  Puno, Pema-Tenzin
Adobe PDF(1823Kb)  |  收藏  |  浏览/下载:241/34  |  提交时间:2019/03/18
Tricholopardins A and B, Anti-inflammatory Terpenoids from the Fruiting Bodies of Tricholoma pardinum 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2019, 卷号: 82, 期号: 1, 页码: 45-50
作者:  Feng, Tao;  Gan, Xiao-Qing;  Zhao, Yun-Li;  Zhang, Shuai-Bing;  Chen, He-Ping;  He, Juan;  Zheng, Yong-Sheng;  Sun, Huan;  Huang, Rong;  Li, Zheng-Hui;  Liu, Ji-Kai
Adobe PDF(1583Kb)  |  收藏  |  浏览/下载:249/69  |  提交时间:2019/03/18
Renoprotective meroterpenoids from the fungus Ganoderma cochlear 期刊论文
FITOTERAPIA, 2019, 卷号: 132, 页码: 88-93
作者:  Wang, Xin-Long;  Wu, Ze-Hong;  Di, Lei;  Zhou, Feng-Jiao;  Yan, Yong-Ming;  Cheng, Yong-Xian
Adobe PDF(827Kb)  |  收藏  |  浏览/下载:196/54  |  提交时间:2019/03/18
Ganoderma cochlear  Meroterpenoids  ECD calculations  Renal fibrosis  
Synthesis of Fucosylated Chondroitin Sulfate Nonasaccharide as a Novel Anticoagulant Targeting Intrinsic Factor Xase Complex 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2018, 卷号: 57, 期号: 39, 页码: 12880-12885
作者:  Zhang, Xiao;  Liu, Huiying;  Lin, Lisha;  Yao, Wang;  Zhao, Jinhua;  Wu, Mingyi;  Li, Zhongjun
Adobe PDF(1568Kb)  |  收藏  |  浏览/下载:227/60  |  提交时间:2018/10/22
Anticoagulants  Drug Discovery  Fucosylated Chondroitin Sulfate  Glycosaminoglycans  Oligosaccharides  
Enantioselective Radical Cyclization of Tryptamines by Visible Light-Excited Nitroxides 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 83, 期号: 18, 页码: 10948-10958
作者:  Liang, Kangjiang;  Tong, Xiaogang;  Li, Tao;  Shi, Bingfei;  Wang, Haiyang;  Yan, Pengcheng;  Xia, Chengfeng
收藏  |  浏览/下载:95/0  |  提交时间:2018/11/06
Heterocyclic Compounds from the Mushroom Albatrellus confluens and Their Inhibitions against Lipopolysaccharides-Induced B Lymphocyte Cell Proliferation 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 83, 期号: 17, 页码: 10158-10165
作者:  Zhang, Shuaibing;  Huang, Ying;  He, Shijun;  Chen, Heping;  Wu, Bin;  Li, Shanyong;  Zhao, Zhenzhu;  Li, Zhenghui;  Wang, Xian;  Zuo, Jianping;  Feng, Tao;  Liu, Jikai
收藏  |  浏览/下载:132/0  |  提交时间:2018/10/22