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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:63/15  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Neo-clerodane diterpenoids from aerial parts of Salvia hispanica L. and their cardioprotective effects 期刊论文
PHYTOCHEMISTRY, 2019, 卷号: 166, 页码: 11
作者:  Fan, Min;  Luo, Dan;  Peng, Li-Yan;  Li, Xiao-Nian;  Wu, Xing-De;  Ji, Xu;  Zhao, Qin-Shi
Adobe PDF(1457Kb)  |  收藏  |  浏览/下载:196/54  |  提交时间:2019/10/28
Salvia hispanica L. (Lamiaceae)  Chia  Neo-clerodane diterpenoids  Hispanins A-J  Single crystal X-ray diffraction analysis  Cardioprotective effects  
Total Synthesis of (+/-)-Cermizine B 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 82, 期号: 20, 页码: 11110-11116
作者:  Shi, Xin;  Deng, Zhen-Tao;  Zhu, Yu;  Bao, Ying;  Shao, Li-Dong;  Zhao, Qin-Shi
Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:173/44  |  提交时间:2017/12/18
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:293/67  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
Five new Lycopodium alkaloids from the aerial parts of Phlegmariurus henryi 期刊论文
FITOTERAPIA, 2016, 卷号: 115, 期号: 1, 页码: 148-154
作者:  Liu, Yu-Chen;  Su, Jia;  Wu, Xing-De;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  He, Juan;  Li, Xiao-Nian;  Peng, Li-Yan;  Cheng, Xiao;  Zhao, Qin-Shi
Adobe PDF(964Kb)  |  收藏  |  浏览/下载:219/50  |  提交时间:2017/02/14
Phlegmariurus Henryi  Lycopodium Alkaloids  Anti-ache Activity  Cytotoxicity  
Cheliensisin A (Chel A) induces apoptosis in human bladder cancer cells by promoting PHLPP2 protein degradation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 66689-66699
作者:  Zhang, Ruowen;  Che, Xun;  Zhang, Jingjie;  Li, Yang;  Li, Jingxia;  Deng, Xu;  Zhu, Junlan;  Jin, Honglei;  Zhao, Qinshi;  Huang, Chuanshu
Adobe PDF(9106Kb)  |  收藏  |  浏览/下载:190/44  |  提交时间:2017/01/05
Chel a  Human Bladder Cancer  Apoptosis  Phlpp2  C-jun  
neo-Clerodanes from the aerial parts of Salvia leucantha 期刊论文
TETRAHEDRON, 2016, 卷号: 72, 期号: 35, 页码: 5507-5514
作者:  Jiang, Yong-Jun;  Su, Jia;  Shi, Xin;  Wu, Xing-De;  Chen, Xuan-Qin;  He, Juan;  Shao, Li-Dong;  Li, Xiao-Nian;  Peng, Li-Yan;  Li, Rong-Tao;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1147Kb)  |  收藏  |  浏览/下载:224/46  |  提交时间:2016/11/04
Neo-clerodanes  Salvia Leucantha  Cytotoxicity  Heat Shock Protein 90 Inhibitor  Acetyl Cholinesterase Inhibitory Activity  
Synthesis of a Small-Molecule Library with Skeletal Diversity from Hemslecin A via the Reaction-Discovery Strategy 期刊论文
ORGANIC LETTERS, 2016, 卷号: 18, 期号: 16, 页码: 3948-3951
作者:  Ren, Jian;  Shi, Xin;  Li, Xiao-Nian;  Li, Lai-Wei;  Su, Jia;  Shao, Li-Dong;  Zhao, Qin-Shi
Adobe PDF(390Kb)  |  收藏  |  浏览/下载:166/53  |  提交时间:2016/11/04
Hupehenols A-E, Selective 11 beta-Hydroxysteroid Dehydrogenase Type 1 (11 beta-HSD1) Inhibitors from Viburnum hupehense 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2015, 卷号: 78, 期号: 2, 页码: 330-334
作者:  Chen, Xuan-Qin;  Shao, Li-Dong;  Pal, Mahesh;  Shen, Yu;  Cheng, Xiao;  Xu, Gang;  Peng, Li-Yan;  Wang, Kou;  Pan, Zheng-Hong;  Li, Ming-Ming;  Leng, Ying;  He, Juan;  Zhao, Qin-Shi;  He,J (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650204,Yunnan,Peoples R China.;  hejuan@mail.kib.ac.cn;  qinshizhao@mail.kib.ac.cn
Adobe PDF(811Kb)  |  收藏  |  浏览/下载:289/83  |  提交时间:2015/06/29
Construction of Tetracyclic 3-Spirooxindole through Cross-Dehydrogenation of Pyridinium: Applications in Facile Synthesis of (+/-)-Corynoxine and (+/-)-Corynoxine B 期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2014, 卷号: 136, 期号: 52, 页码: 17962-17965
作者:  Xu, Jun;  Shao, Li-Dong;  Li, Dashan;  Deng, Xu;  Liu, Yu-Chen;  Zhao, Qin-Shi;  Xia, Chengfeng
Adobe PDF(696Kb)  |  收藏  |  浏览/下载:486/83  |  提交时间:2015/06/17