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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:376/42  |  提交时间:2017/12/18
Click Glycosylation for the Synthesis of 1,2,3-Triazole-Linked Picropodophyllotoxin Glycoconjugates and Their Anticancer Activity 期刊论文
CHEMISTRYSELECT, 2017, 卷号: 2, 期号: 18, 页码: 5038-5044
作者:  Zi, Cheng-Ting;  Yang, Liu;  Gao, Wei;  Li, Yan;  Zhou, Jun;  Ding, Zhong-Tao;  Hu, Jiang-Miao;  Jiang, Zi-Hua
Adobe PDF(3775Kb)  |  收藏  |  浏览/下载:225/45  |  提交时间:2017/10/23
Anticancer Activity  Cu(i)-catalyzed Click Reaction  Glycoconjugates  Picropodophyllotoxin  Podophyllotoxin  
Synthesis and Cytotoxic Activity of Novel Hybrid Compounds between Indolo[b]tetrahydrofuran and Imidazolium Salts 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 6, 页码: 1506-1515
作者:  Liu Zhengfen;  Zhang Chaobo;  Duan Shengzu;  Liu Yang;  Chen Wen;  Li Yan;  Zhang Hongbin;  Yang Xiaodong
Adobe PDF(1186Kb)  |  收藏  |  浏览/下载:222/42  |  提交时间:2017/10/23
Indolo[b]Tetrahydrofuran  Imidazolium Salts  Hybrid Compound  Cytotoxic Activity  
Lanostane-type triterpenoids from Kadsura coccinea 期刊论文
TETRAHEDRON, 2017, 卷号: 73, 期号: 20, 页码: 2931-2937
作者:  Hu, Zheng-Xi;  Li, Xiao-Nian;  Shi, Yi-Ming;  Wang, Wei-Guang;  Du, Xue;  Li, Yan;  Zhang, Yong-Hui;  Pu, Jian-Xin;  Sun, Han-Dong
Adobe PDF(860Kb)  |  收藏  |  浏览/下载:772/236  |  提交时间:2017/07/10
Kadsura Coccinea  Lanostane-type Triterpenoids  Cytotoxicity  
USP7 inhibitor P5091 inhibits Wnt signaling and colorectal tumor growth 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2017, 卷号: 131, 期号: 1, 页码: 29-39
作者:  An, Tao;  Gong, Yaxiao;  Li, Xue;  Kong, Lingmei;  Ma, Pengcheng;  Gong, Liang;  Zhu, Huifang;  Yu, Chunlei;  Liu, Jianmei;  Zhou, Hongyu;  Mao, Bingyu;  Li, Yan
Adobe PDF(3138Kb)  |  收藏  |  浏览/下载:787/145  |  提交时间:2017/04/06
Usp7 Inhibitor  Wnt Signaling  Colorectal Cancer  
Synthesis and cytotoxic activity of novel tetrahydrobenzodifuran-imidazolium salt derivatives 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 8, 页码: 1808-1814
作者:  Zhang, Chao-Bo;  Liu, Yang;  Liu, Zheng-Fen;  Duan, Sheng-Zu;  Li, Min-Yan;  Chen, Wen;  Li, Yan;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Adobe PDF(1192Kb)  |  收藏  |  浏览/下载:625/105  |  提交时间:2017/06/30
Tetrahydrobenzodifurans  Imidazolium Salts  Cytotoxic Activity  Cell Cycle  Apoptosis  
Discovery of new dual binding TNKS inhibitors of Wnt signaling inhibition by pharmacophore modeling, molecular docking and bioassay 期刊论文
MOLECULAR BIOSYSTEMS, 2017, 卷号: 13, 期号: 2, 页码: 363-370
作者:  Pu, Yinglan;  Zhang, Shuqun;  Chang, Zhe;  Zhang, Yunqin;  Wang, Dong;  Zhang, Li;  Li, Yan;  Zuo, Zhili
Adobe PDF(972Kb)  |  收藏  |  浏览/下载:685/118  |  提交时间:2017/05/19
Star-PAP, a poly(A) polymerase, functions as a tumor suppressor in an orthotopic human breast cancer model 期刊论文
CELL DEATH & DISEASE, 2017, 卷号: 8, 期号: 1, 页码: e2582
作者:  Yu, C.;  Gong, Y.;  Zhou, H.;  Wang, M.;  Kong, L.;  Liu, J.;  An, T.;  Zhu, H.;  Li, Y.
Adobe PDF(3022Kb)  |  收藏  |  浏览/下载:193/39  |  提交时间:2017/04/19
Ent-Abietanoids Isolated from Isodon serra 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 2, 页码: 309
作者:  Wan, Jun;  Jiang, Hua-Yi;  Tang, Jian-Wei;  Li, Xing-Ren;  Du, Xue;  Li, Yan;  Sun, Han-Dong;  Pu, Jian-Xin
Adobe PDF(821Kb)  |  收藏  |  浏览/下载:661/114  |  提交时间:2017/05/19
Isodon Serra  Ent-abietane Diterpenoids  Anti-inflammation  Cytotoxicity  
microRNA-375 inhibits colorectal cancer cells proliferation by downregulating JAK2/STAT3 and MAP3K8/ERK signaling pathways 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 10, 页码: 16633-16641
作者:  Wei, Ran;  Yang, Qin;  Han, Bing;  Li, Yan;  Yao, Kun;  Yang, Xiuyu;  Chen, Zexi;  Yang, Shanshan;  Zhou, Jiaqi;  Li, Meizhang;  Yu, Haijing;  Yu, Min;  Cui, Qinghua
Adobe PDF(12068Kb)  |  收藏  |  浏览/下载:420/36  |  提交时间:2017/04/19
Microrna-375  Colorectal Cancer  Jak2/stat3 Pathway  Map3k8/erk Pathway  Atg7