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Catalyzed Synthesis of 3-hydroxy-indol-2-one Derivatives as a Novel Phosphodiesterases 10 Inhibitor 期刊论文
BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2020, 卷号: 126, 页码: 33-34
作者:  Wu, Ya;  Li, Hao;  Yan, Jiao;  Cai, Qing;  Huang, Shengxiong;  Tang, Ying;  Ji, Yue;  Hao, Xiaojiang;  Chen, Gang
收藏  |  浏览/下载:193/0  |  提交时间:2020/03/24
Synthesis and PDE-10 Inhibition of 3-substituted Phenylimino-indolin-2-ones 期刊论文
BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2020, 卷号: 126, 页码: 34-34
作者:  Wu, Ya;  Lin, Zhiwei;  Bai, Yun;  Zhang, Yu;  Cai, Qing;  Mu, Shuzhen;  Han, Weiwei;  Hao, Xiaojiang;  Chen, Gang
收藏  |  浏览/下载:156/0  |  提交时间:2020/03/24
Aromatization of natural products by a specialized detoxification enzyme 期刊论文
NATURE CHEMICAL BIOLOGY, 2020, 卷号: 16, 期号: 3, 页码: 11
作者:  Huang, Jin-Quan;  Fang, Xin;  Tian, Xiu;  Chen, Ping;  Lin, Jia-Ling;  Guo, Xiao-Xiang;  Li, Jian-Xu;  Fan, Zhen;  Song, Wei-Meng;  Chen, Fang-Yan;  Ahati, Ruzha;  Wang, Ling-Jian;  Zhao, Qing;  Martin, Cathie;  Chen, Xiao-Ya
收藏  |  浏览/下载:111/0  |  提交时间:2020/03/18
Plant Specialized Metabolism Regulated by Jasmonate Signaling 期刊论文
PLANT AND CELL PHYSIOLOGY, 2019, 卷号: 60, 期号: 12, 页码: 2638-2647
作者:  Chen, Xueying;  Wang, Dan-Dan;  Fang, Xin;  Chen, Xiao-Ya;  Mao, Ying-Bo
浏览  |  Adobe PDF(1086Kb)  |  收藏  |  浏览/下载:151/30  |  提交时间:2020/03/18
Jasmonate  Metabolites  Plant defense  
Design, synthesis, and cytotoxic activities of novel hybrids of parthenolide and thiazolidinedione via click chemistry 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2019, 页码: 9
作者:  Qiu, Jie;  Yuan, Chun-Mao;  Wen, Min;  Li, Ya-Nan;  Chen, Juan;  Jian, Jun-You;  Huang, Lie-Jun;  Gu, Wei;  Li, Yan-Mei;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(1093Kb)  |  收藏  |  浏览/下载:188/45  |  提交时间:2019/07/29
Parthenolide-thiazolidinedione hybrids  click chemistry  cytotoxic activities  
Autocatalytic synthesis of 3-ethyl-3-hydroxy-indole-2-ones and their neuroprotection and antitumor activities' evaluation 期刊论文
COMPTES RENDUS CHIMIE, 2018, 卷号: 21, 期号: 5, 页码: 471-474
作者:  Chen, Gang;  Lin, Jiao;  Zhang, Jie;  Wu, Ya;  Gu, Xuefan;  Hao, Xiaojiang;  Zhang, Yu
收藏  |  浏览/下载:95/0  |  提交时间:2019/03/29
Isatin  3-Ethyl-3-hydroxy-indole-2-one  Antitumor  Neuroprotection  
Synthesis and anti-proliferative activity of allogibberic acid derivatives containing 1,2,3-triazole pharmacophore 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 14, 页码: 2543-2549
作者:  Wu, Ming-Jiang;  Wu, Dong-Mei;  Chen, Jing-Bo;  Zhao, Jing-Feng;  Gong, Liang;  Gong, Ya-Xiao;  Li, Yan;  Yang, Xiao-Dong;  Zhang, Hongbin
收藏  |  浏览/下载:127/0  |  提交时间:2019/03/29
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70, 页码: 186-190
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun;  Chen, Ya-Juan;  Xie, Hui-Ding
浏览  |  Adobe PDF(371Kb)  |  收藏  |  浏览/下载:116/21  |  提交时间:2017/12/11
B-raf Kinase Inhibitors  Virtual Screening  Pharmacophore  Molecular Docking  3d Qsar  Binding Free Energy Calculation  
Melokhanines A-J, Bioactive Monoterpenoid Indole Alkaloids with Diverse Skeletons from Melodinus khasianus 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2016, 卷号: 79, 期号: 9, 页码: 2158-2166
作者:  Cheng, Gui-Guang;  Li, Dan;  Hou, Bo;  Li, Xiao-Nian;  Liu, Lu;  Chen, Ying-Ying;  Lunga, Paul-Keilah;  Khan, Afsar;  Liu, Ya-Ping;  Zuo, Zhi-Li;  Luo, Xiao-Dong
浏览  |  Adobe PDF(1399Kb)  |  收藏  |  浏览/下载:246/60  |  提交时间:2017/01/05
New Cytotoxic Tigliane Diterpenoids from Croton caudatus 期刊论文
PLANTA MEDICA, 2016, 卷号: 82, 期号: 8, 页码: 729-733
作者:  Chen, Ying-Ying;  Yang, Kun-Xian;  Yang, Xing-Wei;  Khan, Afsar;  Liu, Lu;  Wang, Bei;  Zhao, Yun-Li;  Liu, Ya-Ping;  Li, Yan;  Luo, Xiao-Dong
浏览  |  Adobe PDF(2219Kb)  |  收藏  |  浏览/下载:253/67  |  提交时间:2016/08/22
Croton Caudatus  Euphorbiaceae  Tigliane Diterpenoid  Cytotoxic Activity