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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:58/15  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Huperserratines A and B, Two Macrocyclic Lycopodium Alkaloids with an Unusual Skeleton from Huperzia serrata 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020
作者:  Wu, Xing-De;  Li, Xiao-Nian;  Peng, Li-Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1810Kb)  |  收藏  |  浏览/下载:123/63  |  提交时间:2021/01/05
Activation of SIK1 by phanginin A inhibits hepatic gluconeogenesis by increasing PDE4 activity and suppressing the cAMP signaling pathway 期刊论文
MOLECULAR METABOLISM, 2020
作者:  Liu, Siwen;  Huang, Suling;  Wu, Xingde;  Feng, Ying;  Shen, Yu;  Zhao, Qin-shi;  Leng, Ying
浏览  |  Adobe PDF(3899Kb)  |  收藏  |  浏览/下载:92/25  |  提交时间:2021/01/05
Magnograndins J-M, elemane sesquiterpenoids from the leaves of Magnolia grandiflora and their inhibitory effects on nitric oxide production 期刊论文
PHYTOCHEMISTRY LETTERS, 2019, 卷号: 31, 页码: 121-124
作者:  Ding, Lin-Fen;  Liu, Jiang-Xin;  Xie, Zhang-Qiao;  Wang, De-Shen;  Nie, Wei;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(649Kb)  |  收藏  |  浏览/下载:142/26  |  提交时间:2019/07/29
Magnolia grandiflora  Elemane sesquiterpenoid  Nitric oxide (NO)  
Three new Lycopodium alkaloids from Lycopodium japonicum 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2019, 卷号: 21, 期号: 1, 页码: 17-24
作者:  Zhu, Yu;  Dong, Liao-Bin;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  Qi, Yan-Yan;  Liu, Yu-Chen;  Peng, Li-Yan;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1103Kb)  |  收藏  |  浏览/下载:208/54  |  提交时间:2019/05/24
Lycopodiaceae  Lycopodium japonicum  Lycopodium alkaloids  T-type calcium channel  
Cytotoxic sesquiterpenoids from the leaves of Magnolia grandiflora 期刊论文
PHYTOCHEMISTRY, 2018, 卷号: 155, 页码: 182-190
作者:  Ding, Lin-Fen;  Su, Jia;  Pan, Zheng-Hong;  Zhang, Zhi-Jun;  Li, Xiao-Nian;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
Adobe PDF(1049Kb)  |  收藏  |  浏览/下载:548/139  |  提交时间:2018/11/12
Magnolia Grandiflora (Magnoliaceae)  Sesquiterpenoids  Cytotoxic Activity  Nf-kappa b Transcriptional Activity  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:361/40  |  提交时间:2017/12/18
Five new Lycopodium alkaloids from the aerial parts of Phlegmariurus henryi 期刊论文
FITOTERAPIA, 2016, 卷号: 115, 期号: 1, 页码: 148-154
作者:  Liu, Yu-Chen;  Su, Jia;  Wu, Xing-De;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  He, Juan;  Li, Xiao-Nian;  Peng, Li-Yan;  Cheng, Xiao;  Zhao, Qin-Shi
浏览  |  Adobe PDF(964Kb)  |  收藏  |  浏览/下载:215/49  |  提交时间:2017/02/14
Phlegmariurus Henryi  Lycopodium Alkaloids  Anti-ache Activity  Cytotoxicity  
Cheliensisin A (Chel A) induces apoptosis in human bladder cancer cells by promoting PHLPP2 protein degradation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 66689-66699
作者:  Zhang, Ruowen;  Che, Xun;  Zhang, Jingjie;  Li, Yang;  Li, Jingxia;  Deng, Xu;  Zhu, Junlan;  Jin, Honglei;  Zhao, Qinshi;  Huang, Chuanshu
Adobe PDF(9106Kb)  |  收藏  |  浏览/下载:184/42  |  提交时间:2017/01/05
Chel a  Human Bladder Cancer  Apoptosis  Phlpp2  C-jun  
Bioactive sesquiterpenoids from the flowers of Inula japonica 期刊论文
PHYTOCHEMISTRY, 2016, 卷号: 129, 页码: 68-76
作者:  Wu, Xing-De;  Ding, Lin-Fen;  Tu, Wen-Chao;  Yang, Hui;  Su, Jia;  Peng, Li-Yan;  Li, Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1070Kb)  |  收藏  |  浏览/下载:241/59  |  提交时间:2016/11/04
Inula Japonica  Asteraceae  Sesquiterpenoids  Inujaponins A-i  Cytotoxicity  Nitric Oxide (No)