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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:63/15  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Diterpenoids and sesquiterpenoids from the stem bark of Metasequoia glyptostroboides 期刊论文
PHYTOCHEMISTRY, 2019, 卷号: 161, 页码: 86-96
作者:  Tu, Wen-Chao;  Qi, Yan-Yan;  Ding, Lin-Fen;  Yang, Hui;  Liu, Jiang-Xin;  Peng, Li-Yan;  Song, Liu-Dong;  Gong, Xun;  Wu, Xing-De;  Zhao, Qin-Shi
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Metasequoia glyptostroboides Hu & WC Cheng  Cupressaceae  Sesquiterpenoids  Diterpenoids  Cytotoxicity  
Cytotoxic sesquiterpenoids from the leaves of Magnolia grandiflora 期刊论文
PHYTOCHEMISTRY, 2018, 卷号: 155, 页码: 182-190
作者:  Ding, Lin-Fen;  Su, Jia;  Pan, Zheng-Hong;  Zhang, Zhi-Jun;  Li, Xiao-Nian;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
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Magnolia Grandiflora (Magnoliaceae)  Sesquiterpenoids  Cytotoxic Activity  Nf-kappa b Transcriptional Activity  
Two New Anti-Proliferative C-18-Norditerpenes from the Roots of Podocarpus macrophyllus 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 4, 页码: e1800043
作者:  Qi, Yan-Yan;  Su, Jia;  Zhang, Zhi-Jun;  Li, Lai-Wei;  Fan, Min;  Zhu, Yu;  Wu, Xing-De;  Zhao, Qin-Shi
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Podocarpus Macrophyllus  Norditerpenoid  Anti-proliferative Activity  Activity-guided Fractionation  Structure Revision  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
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Cheliensisin A (Chel A) induces apoptosis in human bladder cancer cells by promoting PHLPP2 protein degradation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 66689-66699
作者:  Zhang, Ruowen;  Che, Xun;  Zhang, Jingjie;  Li, Yang;  Li, Jingxia;  Deng, Xu;  Zhu, Junlan;  Jin, Honglei;  Zhao, Qinshi;  Huang, Chuanshu
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Chel a  Human Bladder Cancer  Apoptosis  Phlpp2  C-jun  
Synthesis of a Small-Molecule Library with Skeletal Diversity from Hemslecin A via the Reaction-Discovery Strategy 期刊论文
ORGANIC LETTERS, 2016, 卷号: 18, 期号: 16, 页码: 3948-3951
作者:  Ren, Jian;  Shi, Xin;  Li, Xiao-Nian;  Li, Lai-Wei;  Su, Jia;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(390Kb)  |  收藏  |  浏览/下载:165/53  |  提交时间:2016/11/04
Vinmajorines C-E, Monoterpenoid Indole Alkaloids from Vinca major 期刊论文
HELVETICA CHIMICA ACTA, 2016, 卷号: 99, 期号: 2, 页码: 157-160
作者:  Zhang, Zhi-Jun;  Du, Ru-Nan;  He, Juan;  Wu, Xing-De;  Li, Yan;  Li, Rong-Tao;  Zhao, Qin-Shi
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Vinca Major  Monoterpenoid Indole Alkaloid  Vinmajorines C-e  Cytotoxic Activity  
Nor-lupane triterpenoid and guaiane sesquiterpenoids from Schefflera venulosa 期刊论文
FITOTERAPIA, 2015, 卷号: 103, 页码: 294-298
作者:  Peng, Li-Yan;  Xu, Gang;  He, Juan;  Wu, Xing-De;  Dong, Liao-Bin;  Gao, Xiu;  Cheng, Xiao;  Su, Jia;  Li, Yan;  Dong, Wen-Ming;  Zhao, Qin-Shi
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Schefflera Venulosa  Nor-lupane Triterpenoid  Sesquiterpenoids  3-oxo-29 Alpha-hydroxy-17 Beta  Schvenols A-b  20-epoxy-28-norlupane  
Crucial Role of c-Jun Phosphorylation at Ser63/73 Mediated by PHLPP Protein Degradation in the Cheliensisin A Inhibition of Cell Transformation 期刊论文
CANCER PREVENTION RESEARCH, 2014, 卷号: 7, 期号: 12, 页码: 1270-1281
作者:  Zhu, Junlan;  Zhang, Jingjie;  Huang, Haishan;  Li, Jingxia;  Yu, Yonghui;  Jin, Honglei;  Li, Yang;  Deng, Xu;  Gao, Jimin;  Zhao, Qinshi;  Huang, Chuanshu;  Huang,CS (reprint author),NYU,Sch Med,Nelson Inst Environm Med,57 Old Forge Rd,Tuxedo Pk,NY 10987 USA.
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Naturally Occurring Substances  Magnetic-resonance Spectroscopy  Stem-bark  Melodinus-henryi  Conformational-analysis  (+)-scholarisine  Mechanism  Leaves  Seeds  Camptothecin  Indole Alkaloids  Cytotoxicity  Absolute Configuration  Vinca Major