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The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:288/1  |  提交时间:2017/07/24
The dipyrone metabolite 4-MAA induces hypothermia and inhibits PGE2-dependent and -independent fever while 4-AA only blocks PGE2-dependent fever1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-44
作者:  David do C. Malvar;  Fernando A. Aguiar;  Artur de L. L. Vaz;  Débora C. R. Assis;  Miriam C. C. de Melo;  Valquíria A. P. Jabor;  Evanguedes Kalapothakis;  Sérgio H. Ferreira;  Giuliano C. Clososki;  Glória E. P. de Souza
Adobe PDF(2243Kb)  |  收藏  |  浏览/下载:304/1  |  提交时间:2017/07/24
Dipyrone  Dipyrone Metabolites  Fever  Hypothermia  Lps  Tityus Serrulatus Venom  
The TRPC channel blocker SKF 96365 Inhibits Glioblastoma Cell Growth by Enhancing Reverse Mode of the Na+/Ca2+ Exchanger and Increasing Intracellular Ca2+ 期刊论文
出版物, 3111, 期号: 0, 页码: 1-45
作者:  M Song;  D Chen;  S P Yu
Adobe PDF(1390Kb)  |  收藏  |  浏览/下载:178/1  |  提交时间:2017/07/24
Skf 96365  Trpc Channel  Glioblastoma  Calcium  na+/ca2+ Exchanger  Cell Cycle  Cell Death  
Effects of CO-RM2 on LPS-induced vascular cell adhesion molecule-1 expression and leukocyte adhesion in human rheumatoid synovial fibroblasts 期刊论文
出版物, 3111, 期号: 0, 页码: 1-44
作者:  Pei-Ling Chi;  Yu-Chen Chuang;  Yu-Wen Chen;  Chih-Chung Lin;  Li-Der Hsiao;  Chuen-Mao Yang
Adobe PDF(1319Kb)  |  收藏  |  浏览/下载:183/1  |  提交时间:2017/07/24
Carbon Monoxide  Lipopolysaccharide  Vcam-1  Leukocyte Adhesion  
Artematrovirenolides A-D and Artematrolides S-Z, Sesquiterpenoid Dimers with Cytotoxicity against Three Hepatoma Cell Lines from Artemisia atrovirens 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2022, 卷号: 40, 期号: 1, 页码: 104-114
作者:  Su,Li-Hua;  Li,Tian-Ze;  Ma,Yun-Bao;  Geng,Chang-An;  Huang,Xiao-Yan;  Zhang,Xin;  Gao,Zhen;  Chen,Ji-Jun
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Artemisia atrovirens  Sesquiterpenoid dimers  Structure elucidation  X-ray diffraction  Antihepatoma activity  GUAIANOLIDE  ARGYI  
Discovery of novel coffee diterpenoids with inhibitions on Ca(v)3.1 low voltage-gated Ca2+ channel 期刊论文
FOOD CHEMISTRY, 2022, 卷号: 376, 页码: 131923
作者:  Hu,Guilin;  Dong,Ding;  Du,Shuzong;  Peng,Xingrong;  Wu,Mingkun;  Shi,Qiangqiang;  Hu,Kun;  Hong,Defu;  Wang,Xiaoyuan;  Zhou,Lin;  Nian,Yin;  Qiu,Minghua
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Coffea arabica L  Roasted coffee  Coffee diterpenoid  Cafestol  Kahweol  T-type Ca2+ channels  Ca(v)3.1 low voltage-gated Ca2+ channel  Ca(v)3.1 inhibitors  CALCIUM-CHANNELS  CAFESTOL  KAHWEOL  PHYSIOLOGY  ESTERS  NOMENCLATURE  PHARMACOLOGY  APOPTOSIS  FURANS  
Wheelchair basketball improves the treatment of urinary tract infection in people with motor disabilities: a clinical trial 期刊论文
REVISTA DA ASSOCIACAO MEDICA BRASILEIRA, 2022, 卷号: 68, 期号: 5, 页码: 559-567
作者:  Cavalcante, Ramirie N.;  Santos, Adeliana C. S.;  Rodrigues, Rosilene Andrade Silva;  Napoleao, Amanda Colichio Bini;  Balogun, Sikiru O.;  de Andrade, Benedito R. M.;  Fett, Carlos A.;  Zavala, Arturo A. Z.;  Arunachalam, Karuppusamy;  de Oliveira, Ruberlei G.
浏览  |  Adobe PDF(376Kb)  |  收藏  |  浏览/下载:7/1  |  提交时间:2024/04/30
C-reactive protein  Klebsiella pneumoniae  Interleukin-6  Escherichia coli  Sports medicine  Quality of life  RENAL-FUNCTION  EXERCISE  MARKERS  
Detailed Structural Analysis of the Immunoregulatory Polysaccharides from the Mycobacterium Bovis BCG 期刊论文
MOLECULES, 2022, 卷号: 27, 期号: 17, 页码: 5691
作者:  Luo, Lan;  Song, Xuemei;  Chang, Xiao;  Huang, Sheng;  Zhou, Yunxi;  Yang, Shengmei;  Zhu, Yan;  Zhang, Lanyan;  Wu, Yongsheng;  Zhang, Junyin;  Zhou, Zhipeng;  Wu, Mingyi
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active ingredients  polysaccharide purification  glucan  mannan  immunomodulator  BACILLUS-CALMETTE-GUERIN  (BCG)-INDUCED MACROPHAGE CYTOTOXICITY  IMMUNOMODULATORY ACTIVITY  MALDI-TOF  INTERLEUKIN-10  ACTIVATION  IMMUNITY  GLUCANS  SULFATE  MANNAN  
HRESIMS-guided isolation of aspidosperma-scandine type bisindole alkaloids from Melodinus cochinchinensis and their anti-inflammatory and cytotoxic activities 期刊论文
PHYTOCHEMISTRY, 2021, 卷号: 184, 页码: 112673
作者:  Li,Fang-Ru;  Liu,Lu;  Liu,Ya-Ping;  Wang,Jin-Tang;  Yang,Mei-Lian;  Khan,Afsar;  Qin,Xu-Jie;  Wang,Yu-Dan;  Cheng,Gui-Guang
收藏  |  浏览/下载:71/0  |  提交时间:2022/04/02
Melodinus cochinchinensis (Lour.) Merr. (Apocynaceae)  melokhanines  Bisindole alkaloids  Anti-inflammatory  Cytotoxicity  MONOTERPENOID INDOLE ALKALOIDS  CHEMISTRY  FRUITS  
New guaiane-type sesquiterpenoid dimers from Artemisia atrovirens and their antihepatoma activity 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 6, 页码: 1648-1666
作者:  Su,Lihua;  Zhang,Xintian;  Ma,Yunbao;  Geng,Changan;  Huang,Xiaoyan;  Hu,Jing;  Li,Tianze;  Tang,Shuang;  Shen,Cheng;  Gao,Zhen;  Zhang,Xuemei;  Chen,Ji-Jun
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Guaianolide dimers  Artematrolides AeR  Artemisia atrovirens  Cytotoxicity  Cell cycle  Apoptosis  FARNESYL-PROTEIN TRANSFERASE  CELL-CYCLE ARREST  HEPATOCELLULAR-CARCINOMA  GUAIANOLIDES  LACTONES  INHIBITORS  ARTEMINOLIDE  APOPTOSIS  ARGYI  HELA