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Structural and mechanistic basis of penicillin-bindingprotein inhibition by lactivicins 期刊论文
NATURE CHEMICAL BIOLOGY, 3111, 期号: 0, 页码: 1—5
作者:  Pauline Macheboeuf;  Delphine S Fischer;  Tom Brown Jr;  Astrid Zervosen;  Andre´Luxen;  Bernard Joris;  Andrea Dessen;  Christopher J Schofield
Adobe PDF(425Kb)  |  收藏  |  浏览/下载:93/1  |  提交时间:2017/07/21
Biosynthetically Inspired Divergent Syntheses of Merocytochalasans 期刊论文
CHEM, 2021, 卷号: 7, 期号: 1, 页码: 212-223
作者:  Long,Xianwen;  Wu,Hai;  Ding,Yiming;  Qu,Chunlei;  Deng,Jun
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RING-SYSTEM  REARRANGEMENTS  DIMER  
The untapped potential of plant sesterterpenoids: chemistry, biological activities and biosynthesis 期刊论文
NATURAL PRODUCT REPORTS, 2021, 卷号: 38, 期号: 12, 页码: 2293-2314
作者:  Guo,Kai;  Liu,Yan;  Li,Sheng-Hong
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LEUCOSCEPTRUM-CANUM  GLANDULAR TRICHOMES  FERN CONSTITUENTS  AERIAL PARTS  ABSOLUTE STEREOCHEMISTRY  SALVIA  CYCLIZATION  SYNTHASES  NORSESTERTERPENES  CONFIGURATION  
Three new diterpenoids fromEuphorbia peplus 期刊论文
NATURAL PRODUCT RESEARCH, 2021, 卷号: 35, 期号: 21, 页码: 3901-3907
作者:  Chen,Yan-Ni;  Lu,Qing-Yun;  Li,Dong-Mei;  Li,Ying-Yao;  Pu,Xue-Xue;  Li,Bo-Ting;  Tang,Xiao-Han;  Tang,Hong-Yu;  Liu,Shuai;  Yang,Lei;  Zhang,Yu;  Di,Ying-Tong;  Fang,Xin;  Hao,Xiao-Jiang
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Euphorbiaceae  Euphorbia peplus  ent-abietane diterpenoids  paralianone diterpenoids  EUPHORBIA-PEPLUS  STEMS  
Diarylheptanoid-flavanone Hybrids as Multiple-target Antidiabetic Agents from Alpinia katsumadai 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 11, 页码: 3051-3063
作者:  He,Xiao-Feng;  Chen,Ji-Jun;  Li,Tian-Ze;  Hu,Jing;  Huang,Xiao-Yan;  Zhang,Xue-Mei;  Guo,Yuan-Qiang;  Geng,Chang-An
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Alpinia katsumadai  Katsumadainols B-1-B-15  Natural products  Structure elucidation  Biological activity  TYROSINE-PHOSPHATASE 1B  GLYCOGEN-PHOSPHORYLASE  ALPHA-GLUCOSIDASE  ABSOLUTE-CONFIGURATION  STRUCTURE ELUCIDATION  DUAL INHIBITION  SEEDS  CONSTITUENT  DERIVATIVES  CHALCONE  
Monoterpene Indole Alkaloids with Ca(v)3.1 T-Type Calcium Channel Inhibitory Activity from Catharanthus roseus 期刊论文
MOLECULES, 2021, 卷号: 26, 期号: 21, 页码: 6516
作者:  Deng,Zhen-Tao;  Li,Wen-Yan;  Wang,Lei;  Zhou,Zhi-Ping;  Wu,Xing-De;  Ding,Zhong-Tao;  Zhao,Qin-Shi
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Catharanthus roseus  monoterpene indole alkaloid  catharanosine A  Ca(v)3  1 low voltage-gated calcium channel (LVGCC)  VINCA ALKALOIDS  CELL-PROLIFERATION  N-OXIDE  SARPAGINE  BIOSYNTHESIS  VINORELBINE  VINBLASTINE  MECHANISM  ROOTS  BASES  
Chemical profiling and antidiabetic potency of Paeonia delavayi: Comparison between different parts and constituents 期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 198, 页码: 113998
作者:  Huang,Qian;  Chen,Ji-Jun;  Pan,Yang;  He,Xiao-Feng;  Wang,Yuan;  Zhang,Xue-Mei;  Geng,Chang-An
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Paeonia delavayi  Chemical comparison  LCMS analyses  Antidiabetic effects  PTP1B/TCPTP selective inhibitors  LIQUID-CHROMATOGRAPHY  MULTIPLE CONSTITUENTS  RAPID IDENTIFICATION  GLYCOSIDES  ROOT  DERIVATIVES  TARGETS  CAPSULE  L.  
Diarylheptanoid-chalcone hybrids with PTP1B and alpha-glucosidase dual inhibition from Alpinia katsumadai 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 104683
作者:  He,Xiao-Feng;  Chen,Ji-Jun;  Li,Tian-Ze;  Hu,Jing;  Zhang,Xue-Mei;  Geng,Chang-An
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Alpinia katsumadai  Katsumadainols A(1)-A(16)  PTP1B/TCPTP selective inhibitors  alpha-glucosidase inhibitors  Antidiabetic effects  THEORETICAL CALCULATION  ABSOLUTE-CONFIGURATION  SEEDS  BLEPHAROCALYXINS  ADDUCT  MOIETY  
Targeting ubiquitin conjugating enzyme UbcH5b by a triterpenoid PC3-15 from Schisandra plants sensitizes triple-negative breast cancer cells to lapatinib 期刊论文
CANCER LETTERS, 2021, 卷号: 504, 页码: 125-136
作者:  Huang,Maobo;  Zhou,Yuanfei;  Duan,Dongzhu;  Yang,Chuanyu;  Zhou,Zhongmei;  Li,Fubing;  Kong,Yanjie;  Hsieh,Yi-Ching;  Zhang,Ruihan;  Ding,Wenping;  Xiao,Weilie;  Puno,PemaTenzin;  Chen,Ceshi
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HECTD3  UbcH5b  Ubiquitination  Autophagy  Schisandraceae triterpenoid  
Polymethylated acylphloroglucinols from Rhodomyrtus tomentosa exert acetylcholinesterase inhibitory effects 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 107, 页码: 104519
作者:  Qin,Xu-Jie;  Liu,Hui;  Li,Pan-Pan;  Ni,Wei;  He,Li;  Khan,Afsar;  Hao,Xiao-Jiang;  Liu,Hai-Yang
Adobe PDF(2105Kb)  |  收藏  |  浏览/下载:100/44  |  提交时间:2022/04/02
Rhodomyrtus tomentosa  Polymethylated acyphloroglucinols  AChE inhibitory effect  Molecular docking  PHLOROGLUCINOL MEROTERPENOIDS  LEAVES  DERIVATIVES  TWIGS  BETA