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Polybenzyls from Gastrodia elata, their agonistic effects on melatonin receptors and structure-activity relationships 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3299-3306
作者:  Chen, Si-Yue;  Geng, Chang-An;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Yang, Xiao-Tong;  Su, Li-Hua;  He, Xiao-Feng;  Li, Tian-Ze;  Deng, Zhen-Tao;  Gao, Zhen;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(1837Kb)  |  收藏  |  浏览/下载:205/37  |  提交时间:2019/09/10
Gastrodia elata  Polybenzyls  Melatonin receptors  Structure-activity relationships  Docking study  
Synthesis and antitumor activity of novel steroidal imidazolium salt derivatives 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 168, 页码: 232-252
作者:  Deng, Guogang;  Zhou, Bei;  Wang, Jing;  Chen, Zhuo;  Gong, Liang;  Gong, Yaxiao;  Wu, Dongmei;  Li, Yan;  Zhang, Hongbin;  Yang, Xiaodong
浏览  |  Adobe PDF(1727Kb)  |  收藏  |  浏览/下载:259/39  |  提交时间:2019/07/29
Diosgenin  Cholesterol  Dehydroepiandrosterone  Imidazolium salt  Antitumor activities  Structure-activity relationships  
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:312/72  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
New Phragmalin-Type Limonoid Orthoesters from the Bark of Chukrasia tabularis var. velutina 期刊论文
HELVETICA CHIMICA ACTA, 2015, 卷号: 98, 期号: 10, 页码: 1403-1410
作者:  Liu,Wen-Xing;  Chen,Duo-Zhi;  Ding,Jia-Yin;  Hao,Xiao-Jiang;  Li,Shun-Lin
浏览  |  Adobe PDF(460Kb)  |  收藏  |  浏览/下载:298/77  |  提交时间:2016/01/19
Limonoids  Orthoesters  X-ray Diffraction  Brine Shrimp Lethality  Chukrasia Tabularis  
Design, Synthesis and Cytotoxic Activity of Novel Hybrid Compounds between Aza-brazilin and Imidazolium 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2015, 卷号: 35, 期号: 6, 页码: 1276-1285
作者:  Wang Xuequan;  Li Yan;  Yang Xiaodong;  Zhang Hongbin
浏览  |  Adobe PDF(566Kb)  |  收藏  |  浏览/下载:187/50  |  提交时间:2016/01/19
Aza-brazilin  Imidazole  Hybrid Compound  Cytotoxic Activity  
氮杂Brazilin-咪唑盐杂合物的设计、合成及细胞毒活性研究 期刊论文
有机化学, 2015, 期号: 6, 页码: 1276-1285
作者:  汪学全;  李艳;  羊晓东;  张洪彬
浏览  |  Adobe PDF(1137Kb)  |  收藏  |  浏览/下载:165/42  |  提交时间:2016/06/27
氮杂brazilin  咪唑  杂合物  细胞毒活性  
Novel Tricyclic Indeno[5,6-b] furan-imidazole Hybrid Compounds: Design, Synthesis and Antitumor Activity 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2013, 卷号: 10, 期号: 7, 页码: 561-571
作者:  Chen, Wen;  Yang, Li-Juan;  Li, Yan;  Wang, Xue-Quan;  Wang, Shao-Jie;  Wan, Wei-Chao;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Unknown(243Kb)  |  收藏  |  浏览/下载:240/3  |  提交时间:2013/10/16
Hybrid Compound  Imidazole  Synthesis  Indeno[5  Cytotoxic Activity  6-b]Furan  Structure-activity Relationships  
Chlojaponilactones B - E, Four New Lindenane Sesquiterpenoid Lactones from Chloranthus japonicus 期刊论文
HELVETICA CHIMICA ACTA, 2013, 卷号: 96, 期号: 7, 页码: 1386-1391
作者:  Yan, Huan;  Li, Xu-Hong;  Zheng, Xue-Fang;  Sun, Chang-Li;  Liu, Hai-Yang
Adobe PDF(192Kb)  |  收藏  |  浏览/下载:336/122  |  提交时间:2014/01/13
Chloranthus Japonicus  Lindenanes  Chlojaponilactones B-e  Sesquiterpenoids  Lactones  
Protein-based alignment in 3D-QSAR of FBPase inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 卷号: 46, 期号: 3, 页码: 885-892
作者:  Yi, Ping;  Di, Ying-Tong;  Liu, Wei;  Hao, Xiao-Jiang;  Ming, Yong;  Huang, Du-Shu;  Yang, Jin;  Yi, Zhong-Zhou;  Li, Zi-Jing;  Yang, Rui-Dong;  Zhang, Ju-Cheng
Adobe PDF(777Kb)  |  收藏  |  浏览/下载:399/164  |  提交时间:2012/04/10
3d-qsar  Gold  Comfa  Fbpase  
Four New 9,19-Cyclolanostane Derivatives from the Rhizomes of Cimicifuga yunnanensis HSIAO 期刊论文
HELVETICA CHIMICA ACTA, 2009, 卷号: 92, 期号: 1, 页码: 112-120
作者:  Nian, Yin;  Chen, Jian-Chao;  Lu, Lu;  Zhang, Xian-Ming;  Zhou, Lin;  Qiu, Ming-Hua
Adobe PDF(207Kb)  |  收藏  |  浏览/下载:257/101  |  提交时间:2011/12/19
Crude Drug Shoma  Simplex Wormsk  Triterpene Glycosides  Aerial Parts  Cyclolanostanol Glycosides  Underground Parts  Foetida l  Constituents  Racemosa  Xylosides