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Total Synthesis of (-)-Geissoschizol through Ir-Catalyzed Allylic Amidation as the Key Step 期刊论文
ORGANIC LETTERS, 2017, 卷号: 19, 期号: 23, 页码: 6460-6462
作者:  Zheng, Yu;  Wei, Kun;  Yang, Yu-Rong
浏览  |  Adobe PDF(870Kb)  |  收藏  |  浏览/下载:165/55  |  提交时间:2018/05/08
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:385/42  |  提交时间:2017/12/18
Manginoids A-G: Seven Monoterpene-Shikimate-Conjugated Meroterpenoids with a Spiro Ring System from Guignardia mangiferae 期刊论文
ORGANIC LETTERS, 2017, 卷号: 19, 期号: 21, 页码: 5956-5959
作者:  Chen, Keliang;  Zhang, Xuwen;  Sun, Weiguang;  Liu, Junjun;  Yang, Jing;  Chen, Chunmei;  Liu, Xiulan;  Gao, Limin;  Wang, Jianping;  Li, Hua;  Luo, Zengwei;  Xue, Yongbo;  Zhu, Hucheng;  Zhang, Yonghui
浏览  |  Adobe PDF(1771Kb)  |  收藏  |  浏览/下载:327/34  |  提交时间:2017/12/18
Borapetoside E 对高脂饮食诱导小鼠糖脂代谢的影响及其机制研究 学位论文
: 中国科学院大学, 2017
作者:  许宇辉
Adobe PDF(4170Kb)  |  收藏  |  浏览/下载:137/5  |  提交时间:2019/06/14
老药新用:奥柳氮钠的降尿酸作用及分子机制研究 学位论文
: 中国科学院大学, 2017
作者:  牛艳芬
Adobe PDF(4338Kb)  |  收藏  |  浏览/下载:113/6  |  提交时间:2019/06/14
钯催化非活泼碳氢键胺化反应构建氮杂环骨架的方法学研究 学位论文
: 中国科学院大学, 2017
作者:  赵杰
Adobe PDF(10881Kb)  |  收藏  |  浏览/下载:157/2  |  提交时间:2019/06/14
Old drug, new indication: Olsalazine sodium reduced serum uric acid levels in mice via inhibiting xanthine oxidoreductase activity 期刊论文
JOURNAL OF PHARMACOLOGICAL SCIENCES, 2017, 卷号: 135, 期号: 3, 页码: 114-120
作者:  Niu, Yanfen;  Li, Hongjian;  Gao, Lihui;  Lin, Hua;  Kung, Hsiangfu;  Lin, Marie Chia-mi;  Leung, Kwong-Sak;  Wong, Man-Hon;  Xiong, Wenyong;  Li, Ling
收藏  |  浏览/下载:99/0  |  提交时间:2018/05/08
Olsalazine Sodium  Hyperuricemia  Xanthine Oxidase  Uric Acid  
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70, 页码: 186-190
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun;  Chen, Ya-Juan;  Xie, Hui-Ding
浏览  |  Adobe PDF(371Kb)  |  收藏  |  浏览/下载:148/24  |  提交时间:2017/12/11
B-raf Kinase Inhibitors  Virtual Screening  Pharmacophore  Molecular Docking  3d Qsar  Binding Free Energy Calculation  
Potential role of CYP1B1 in the development and treatment of metabolic diseases 期刊论文
PHARMACOLOGY & THERAPEUTICS, 2017, 卷号: 178, 页码: 18-30
作者:  Li, Fei;  Zhu, Weifeng;  Gonzalez, Frank J.
浏览  |  Adobe PDF(2083Kb)  |  收藏  |  浏览/下载:183/60  |  提交时间:2017/11/20
Cyp1b1  Metabolic Diseases  Metabolic Pathways  Metabolomics  
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:316/73  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar