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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
作者:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
Adobe PDF(1403Kb)  |  收藏  |  浏览/下载:268/1  |  提交时间:2017/07/24
Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
Structural and mechanistic basis of penicillin-bindingprotein inhibition by lactivicins 期刊论文
NATURE CHEMICAL BIOLOGY, 3111, 期号: 0, 页码: 1—5
作者:  Pauline Macheboeuf;  Delphine S Fischer;  Tom Brown Jr;  Astrid Zervosen;  Andre´Luxen;  Bernard Joris;  Andrea Dessen;  Christopher J Schofield
Adobe PDF(425Kb)  |  收藏  |  浏览/下载:89/1  |  提交时间:2017/07/21
Increased Catalytic Efficiency following Gene Fusion of Bifunctional MethionineSulfoxide Reductase Enzymes from Shewanella oneidensis 期刊论文
Biochemistry, 3111, 页码: 1—9
作者:  C.B. Li;  D.M. Zhang;  S. Ge;  D.Y. Hong
Adobe PDF(436Kb)  |  收藏  |  浏览/下载:128/1  |  提交时间:2017/07/19
YC-1 inhibits proliferation of breast cancer cells by downregulating EZH2 expression via activation of c-Cbl and ERK 期刊论文
出版物, 3111, 期号: 0, 页码: 1-46
作者:  Ling-Chu Chang;  Hui-Yi Lin;  Meng-Tung Tsai;  Ruey-Hwang Chou;  Fang-Yu Lee;  Che-Ming Teng;  Min-Tsang Hsieh;  Hsin-Yi Hung;  Li-Jiau Huang;  Yung-Luen Yu;  Sheng-Chu Kuo
Adobe PDF(1357Kb)  |  收藏  |  浏览/下载:304/1  |  提交时间:2017/07/24
Yc-1  Triple-negative Breast Cancer  Erk  Ezh2  C-cbl  
Mono-/Bis-Alkenoic Acid Derivatives From an Endophytic Fungus Scopulariopsis candelabrum and Their Antifungal Activity 期刊论文
FRONTIERS IN CHEMISTRY, 2022
作者:  Tang, Jun;  Huang, Xueshuang;  Cao, Ming-Hang;  Wang, Zhiyan;  Yu, Zhiyin;  Yan, Yijun;  Huang, Jian-Ping;  Wang, Li;  Huang, Sheng-Xiong
浏览  |  Adobe PDF(1321Kb)  |  收藏  |  浏览/下载:157/57  |  提交时间:2023/09/08
seco-Prezizanne Sesquiterpenes and Prenylated C6-C3 Compounds from the Fruits of Illicium lanceolatum A. C. Smith 期刊论文
CHEMISTRY & BIODIVERSITY, 2022, 卷号: 19, 期号: 1, 页码: e202100868
作者:  Nie,Wei;  Ding,Lin-Fen;  Tie-Lei;  Zhou,Hao-Feng;  Bao,Yi;  Song,Liu-Dong;  Pan,Zheng-Hong;  Wu,Xing-De;  Zhao,Qin-Shi
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Illicium lanceolatum A  C  Smith  seco-prezizanne sesquiterpene  prenylated C6-C3 compound  neuroprotective activity  NEUROTROPHIC ACTIVITY  C-6-C-3 COMPOUNDS  STEM BARK  ROOTS  SKELETON  
Isolation and identification of belamcandaoids A-N from Belamcanda chinensis seeds and their inhibition on extracellular matrix in TGF-beta 1 induced kidney proximal tubular cells 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 114, 页码: 105067
作者:  Song,Ying-Ying;  Jiang,Jian-Bing;  Yan,Yong-Ming;  Cheng,Yong-Xian
浏览  |  Adobe PDF(4755Kb)  |  收藏  |  浏览/下载:90/30  |  提交时间:2022/04/02
Belamcanda chinensis  Triterpenoids  TGF-beta 1  Kidney proximal tubular cells  TGF-BETA  TRITERPENOIDS  CONSTITUENTS  
Structure Revision of Four Classes of Prenylated Aromatic Natural Products Based on a Rule for Diagnostic C-13 NMR Chemical Shifts 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 16, 页码: 10982-10990
作者:  Ren,Fu-Cai;  Wang,Li-Xia;  Lv,Yong-Feng;  Hu,Jiang-Miao;  Zhou,Jun
浏览  |  Adobe PDF(1507Kb)  |  收藏  |  浏览/下载:82/29  |  提交时间:2022/04/02
ISOPRENYLATED FLAVONOIDS  CONSTITUENTS  DERIVATIVES  ANALOGS  
Nine Unique Iridoids and Iridoid Glycosides From Patrinia scabiosaefolia 期刊论文
FRONTIERS IN CHEMISTRY, 2021, 卷号: 9, 页码: 657028
作者:  Liu,Zhenhua;  Niu,Yun;  Zhou,Li;  Meng,Lijun;  Chen,Sitan;  Wang,Mengke;  Hu,Jiangmiao;  Kang,Wenyi
浏览  |  Adobe PDF(2310Kb)  |  收藏  |  浏览/下载:96/40  |  提交时间:2022/04/02
Patrinia scabiosaefolia  iridoid  iridoid glycoside  bis-iridoid glycoside  cytotoxic activity  
Hypermonones A-I, New Polyprenylated Acylphloroglucinols from Hypericum monogynum with Multidrug Resistance Reversal Activity 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 9, 页码: 2422-2432
作者:  Zeng,Yan-Rong;  Li,Ya-Nan;  Yang,Jue;  Yi,Ping;  Huang,Lei;  Huang,Lie-Jun;  Gu,Wei;  Hu,Zhan-Xing;  Li,Yan-Mei;  Yuan,Chun-Mao;  Hao,Xiao-Jiang
浏览  |  Adobe PDF(2840Kb)  |  收藏  |  浏览/下载:71/21  |  提交时间:2022/04/02
Hypericum monogynum  Phytochemistry  Structure elucidation  Biological activity  Multidrug resistance reversal activity  P-GLYCOPROTEIN  MODULATORS  CANCER