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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:74/16  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Activation of SIK1 by phanginin A inhibits hepatic gluconeogenesis by increasing PDE4 activity and suppressing the cAMP signaling pathway 期刊论文
MOLECULAR METABOLISM, 2020
作者:  Liu, Siwen;  Huang, Suling;  Wu, Xingde;  Feng, Ying;  Shen, Yu;  Zhao, Qin-shi;  Leng, Ying
Adobe PDF(3899Kb)  |  收藏  |  浏览/下载:104/29  |  提交时间:2021/01/05
Cytotoxic sesquiterpenoids from the leaves of Magnolia grandiflora 期刊论文
PHYTOCHEMISTRY, 2018, 卷号: 155, 页码: 182-190
作者:  Ding, Lin-Fen;  Su, Jia;  Pan, Zheng-Hong;  Zhang, Zhi-Jun;  Li, Xiao-Nian;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
Adobe PDF(1049Kb)  |  收藏  |  浏览/下载:571/144  |  提交时间:2018/11/12
Magnolia Grandiflora (Magnoliaceae)  Sesquiterpenoids  Cytotoxic Activity  Nf-kappa b Transcriptional Activity  
New compound ChlA-F induces autophagy-dependent anti-cancer effect via upregulating Sestrin-2 in human bladder cancer 期刊论文
CANCER LETTERS, 2018, 卷号: 436, 页码: 38-51
作者:  Hua, Xiaohui;  Xua, Jiheng;  Deng, Xu;  Xu, Jiawei;  Li, Jingxia;  Zhu, David Q.;  Zhu, Junlan;  Jin, Honglei;  Tian, Zhongxian;  Huang, Haishan;  Zhao, Qin-shi;  Huang, Chuanshu
收藏  |  浏览/下载:167/0  |  提交时间:2018/11/12
Anchorage-independent growth  Cheliensisine A-fluoride (Ch1A-F)  Macro-autophagy (autophagy)  miR-27a  Sestrin-2  
Vibsanin A sensitizes human acute myeloid leukemia cells to tyrosine kinase inhibitor-induced myeloid differentiation via activation of PKC and upregulation of Lyn 期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2018, 卷号: 502, 期号: 1, 页码: 110-115
作者:  Shen, Xing;  Xing, Shuang;  Zhang, Lu;  Wang, Fangmin;  Ou, Hongling;  Shan, Yajun;  Xiao, He;  Xiang, Guolin;  Wang, Xinru;  Zhao, Qinshi;  Cong, Yuwen;  Yu, Zuyin
收藏  |  浏览/下载:76/0  |  提交时间:2019/03/29
Vibsanin A sensitizes human acute myeloid leukemia cells to tyrosine kinase inhibitor-induced myeloid differentiation via activation of PKC and upregulation of Lyn 期刊论文
ORGANIC LETTERS, 2018, 卷号: 20, 期号: 13, 页码: 4116-4120
作者:  Shen, Xing;  Xing, Shuang;  Zhang, Lu;  Wang, Fangmin;  Ou, Hongling;  Shan, Yajun;  Xiao, He;  Xiang, Guolin;  Wang, Xinru;  Zhao, Qinshi;  Cong, Yuwen;  Yu, Zuyin
收藏  |  浏览/下载:76/0  |  提交时间:2018/12/27
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:372/42  |  提交时间:2017/12/18
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:301/68  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
Sauruchinenols A and B, unprecedented monocyclic diterpenes with new carbon skeleton from the aerial parts of Saururus chinensis 期刊论文
FITOTERAPIA, 2017, 卷号: 116, 页码: 116-120
作者:  Gao, Xiu;  He, Juan;  Wu, Xing-De;  Peng, Li-Yan;  Shao, Li-Dong;  Li, Yan;  Cheng, Xiao;  Zhao, Qin-Shi
Adobe PDF(503Kb)  |  收藏  |  浏览/下载:295/38  |  提交时间:2017/04/18
Saururus Chinensis  Saururaceae  Sauruchinenols A-d  Anti-no Production  
Cheliensisin A (Chel A) induces apoptosis in human bladder cancer cells by promoting PHLPP2 protein degradation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 66689-66699
作者:  Zhang, Ruowen;  Che, Xun;  Zhang, Jingjie;  Li, Yang;  Li, Jingxia;  Deng, Xu;  Zhu, Junlan;  Jin, Honglei;  Zhao, Qinshi;  Huang, Chuanshu
Adobe PDF(9106Kb)  |  收藏  |  浏览/下载:192/44  |  提交时间:2017/01/05
Chel a  Human Bladder Cancer  Apoptosis  Phlpp2  C-jun