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Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:  Chen, Duo-zhi;  Yang, Bi-juan;  He, Xiao-li;  Fan, Shi-rui;  Cai, Jie-yun;  Jing, Chen-xu;  Zhang, Heng;  Zhang, Yu;  Li, Lin;  Hao, Xiao-jiang
Adobe PDF(3047Kb)  |  收藏  |  浏览/下载:312/37  |  提交时间:2019/03/18
Wnt/beta-catenin signalling pathway agonist  Phenanthridine derivatives  Structural optimization  Structure-activity relationships (SARs)  
Munronin O, a potential activator for plant resistance 期刊论文
PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY, 2018, 卷号: 146, 页码: 13-18
作者:  Yan, Ying;  Tang, Lei;  Hu, Jiaqi;  Wang, Jianta;  Adelakun, Tiwalade Adegoke;  Yang, Dongqiong;  Di, Yingtong;  Zhang, Yu;  Hao, Xiaojiang
Adobe PDF(1146Kb)  |  收藏  |  浏览/下载:593/156  |  提交时间:2018/06/11
Limonoids  Munronia Henryi Harms  Tobacco Mosaic Virus  Antiviral Activity  Plant Resistance  
Phytotoxic Terpenoids from Ligularia cymbulifera Roots 期刊论文
FRONTIERS IN PLANT SCIENCE, 2017, 卷号: 7, 页码: Article 2033
作者:  Chen, Jia;  Zheng, Guowei;  Zhang, Yu;  Aisa, Haji A.;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(2504Kb)  |  收藏  |  浏览/下载:186/34  |  提交时间:2017/11/20
Ligularia Cymbulifera  Ligulacymirin a  Ligulacymirin b  Eremophilane Sesquiterpenes  Phytotoxic Activity  
16-nor Limonoids from Harrisonia perforata as promising selective 11 beta-HSD1 inhibitors 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6, 页码: 1
作者:  Xiao-HuiYan;  Yi, Ping;  Cao, Pei;  Yang, Shi-Ying;  Fang, Xin;  Zhang, Yu;  Wu, Bin;  Leng, Ying;  Di, Ying-Tong;  Lv, Yang;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(1151Kb)  |  收藏  |  浏览/下载:343/54  |  提交时间:2017/01/05
Bavachinin, as a novel natural pan-PPAR agonist, exhibits unique synergistic effects with synthetic PPAR-gamma and PPAR-alpha agonists on carbohydrate and lipid metabolism in db/db and diet-induced obese mice 期刊论文
DIABETOLOGIA, 2016, 卷号: 59, 期号: 6, 页码: 1276-1286
作者:  Feng, Li;  Luo, Huan;  Xu, Zhijian;  Yang, Zhuo;  Du, Guoxin;  Zhang, Yu;  Yu, Lijing;  Hu, Kaifeng;  Zhu, Weiliang;  Tong, Qingchun;  Chen, Kaixian;  Guo, Fujiang;  Huang, Cheng;  Li, Yiming
浏览  |  Adobe PDF(841Kb)  |  收藏  |  浏览/下载:236/96  |  提交时间:2016/08/22
Alternative Binding Site  Bavachinin  Canonical Ligand-binding Pocket  Carbohydrate Metabolism  Lipid Metabolism  Pan-ppar Agonist  Synergistic Effects  
Synthesis, Neuro-protection and Anti-cancer Activities of Simple Isatin Mannich and Schiff Bases 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2016, 卷号: 13, 期号: 5, 页码: 395-400
作者:  Chen, Gang;  Ning, Yang;  Zhao, Wei;  Zhang, Yanqiu;  Zhang, Yu;  Hao, Xiaojiang;  Wang, Ye;  Mu, Shuzhen
浏览  |  Adobe PDF(1361Kb)  |  收藏  |  浏览/下载:230/70  |  提交时间:2016/08/22
Isatin  Mannich Base  Schiff Base  Synthesis  Neuro-protection  Anti-tumor  
Lycorine-derived phenanthridine downregulators of host Hsc70 as potential hepatitis C virus inhibitors 期刊论文
FUTURE MEDICINAL CHEMISTRY, 2015, 卷号: 7, 期号: 5, 页码: 561-570
作者:  Chen, Duozhi;  Cai, Jieyun;  Yin, Junlin;  Jiang, Jiandong;  Jing, Chenxu;  Zhu, Yanping;  Cheng, Junjun;  Di, Yingtong;  Zhang, Yu;  Cao, Mingming;  Li, Shunlin;  Peng, Zonggen;  Hao, Xiaojiang;  Hao,XJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Yunnan,Peoples R China.;  haoxj@mail.kib.ac.cn
浏览  |  Adobe PDF(1560Kb)  |  收藏  |  浏览/下载:291/54  |  提交时间:2015/07/20
Synthesis, Cytoprotective and Anti-tumor Activities of Isatin Schiff Bases 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2015, 卷号: 12, 期号: 10, 页码: 802-805
作者:  Chen, Gang;  Meng, Mei;  Zhang, Yu;  Hao, Xiaojiang;  Wang, Ye;  Mu, Shuzhen
浏览  |  Adobe PDF(1108Kb)  |  收藏  |  浏览/下载:138/38  |  提交时间:2016/01/19
Isatin  Synthesis  Schiff Base  Structure  Cytoprotective  Anti-tumor  
Phragmalin Limonoids from the Stem Barks of Chukrasia tabularis var. velutina 期刊论文
PLANTA MEDICA, 2014, 卷号: 80, 期号: 15, 页码: 1304-1309
作者:  Yin, Jun-Lin;  Fang, Xin;  Liu, En-De;  Yuan, Chun-Mao;  Li, Shi-Fei;  Zhang, Yu;  He, Hong-Ping;  Li, Shun-Lin;  Di, Ying-Tong;  Hao, Xiao-Jiang;  Hao,XJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,132 Lanhei Rd,Kunming 650201,Peoples R China.;  diyt@mail.kib.ac.cn;  haoxj@mail.kib.ac.cn
Adobe PDF(128Kb)  |  收藏  |  浏览/下载:276/79  |  提交时间:2014/11/25
Chukrasia Tabularis  Meliaceae  Phragmalin  Limonoid  Chukvelutilide i  Artemia Sinica  
New steroids and sesquiterpene from Turraea pubescens 期刊论文
FITOTERAPIA, 2013, 卷号: 90, 页码: 119-125
作者:  Yuan, Chun-Mao;  Tang, Gui-Hua;  Wang, Xiao-Ying;  Zhang, Yu;  Cao, Ming-Ming;  Li, Xiao-Hui;  Li, Yan;  Li, Shun-Lin;  Di, Ying-Tong;  He, Hong-Ping;  Hao, Xiao-Jiang;  Hua, Hui-Ming
Adobe PDF(899Kb)  |  收藏  |  浏览/下载:494/262  |  提交时间:2014/01/13
Turraea Pubescens  Meliaceae  Steroids  Sesquiterpene  Anti-inflammatory