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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:127/29  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Activation of SIK1 by phanginin A inhibits hepatic gluconeogenesis by increasing PDE4 activity and suppressing the cAMP signaling pathway 期刊论文
MOLECULAR METABOLISM, 2020
作者:  Liu, Siwen;  Huang, Suling;  Wu, Xingde;  Feng, Ying;  Shen, Yu;  Zhao, Qin-shi;  Leng, Ying
浏览  |  Adobe PDF(3899Kb)  |  收藏  |  浏览/下载:148/43  |  提交时间:2021/01/05
Three new Lycopodium alkaloids from Lycopodium japonicum 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2019, 卷号: 21, 期号: 1, 页码: 17-24
作者:  Zhu, Yu;  Dong, Liao-Bin;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  Qi, Yan-Yan;  Liu, Yu-Chen;  Peng, Li-Yan;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1103Kb)  |  收藏  |  浏览/下载:289/68  |  提交时间:2019/05/24
Lycopodiaceae  Lycopodium japonicum  Lycopodium alkaloids  T-type calcium channel  
Cytotoxic sesquiterpenoids from the leaves of Magnolia grandiflora 期刊论文
PHYTOCHEMISTRY, 2018, 卷号: 155, 页码: 182-190
作者:  Ding, Lin-Fen;  Su, Jia;  Pan, Zheng-Hong;  Zhang, Zhi-Jun;  Li, Xiao-Nian;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1049Kb)  |  收藏  |  浏览/下载:607/152  |  提交时间:2018/11/12
Magnolia Grandiflora (Magnoliaceae)  Sesquiterpenoids  Cytotoxic Activity  Nf-kappa b Transcriptional Activity  
Ly1 cogladines A-H, fawcettimine-type Lycopodium alkaloids from Lycopodium complanatum var. glaucum Ching 期刊论文
TETRAHEDRON, 2018, 卷号: 74, 期号: 14, 页码: 1692-1697
作者:  Zhang, Zhi-Jun;  Qi, Yan-Yan;  Wu, Xing-De;  Su, Jia;  Zhao, Qin-Shi
收藏  |  浏览/下载:380/0  |  提交时间:2018/05/08
Lycopodium Complanatum Var. Glaucum  Ching  Lycopodium Alkaloids  Lycogladines A-h  Anti-ache Activity  Anti-bace1 Activity  
Salvihispin A and its glycoside, two neo-clerodane diterpenoids with neurotrophic activities from Salvia hispanica L. 期刊论文
TETRAHEDRON LETTERS, 2018, 卷号: 59, 期号: 2, 页码: 143-146
作者:  Fan, Min;  Zhu, Yu;  Zhang, Zhi-Jun;  Du, Ru-Nan;  Zhu, Qin-Feng;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(742Kb)  |  收藏  |  浏览/下载:481/113  |  提交时间:2018/05/08
Neo-clerodane Diterpenoids  Salvia Hispanica  Neurotrophic Activities  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:411/46  |  提交时间:2017/12/18
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:350/88  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
A biomimetic semisynthesis enables structural elucidation of selaginellin U: a tautomeric cyclic alkynylphenol from Selaginella tamariscina 期刊论文
ROYAL SOCIETY OPEN SCIENCE, 2017, 卷号: 4, 期号: 7, 页码: 170352
作者:  Zhu, Qin-Feng;  Bao, Ying;  Zhang, Zhi-Jun;  Su, Jia;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(698Kb)  |  收藏  |  浏览/下载:186/31  |  提交时间:2017/10/23
Biomimetic Semisynthesis  Structural Elucidation  Selaginellins  Alkynylphenol  Selaginella Tamariscina  
Cheliensisin A (Chel A) induces apoptosis in human bladder cancer cells by promoting PHLPP2 protein degradation 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 66689-66699
作者:  Zhang, Ruowen;  Che, Xun;  Zhang, Jingjie;  Li, Yang;  Li, Jingxia;  Deng, Xu;  Zhu, Junlan;  Jin, Honglei;  Zhao, Qinshi;  Huang, Chuanshu
浏览  |  Adobe PDF(9106Kb)  |  收藏  |  浏览/下载:231/50  |  提交时间:2017/01/05
Chel a  Human Bladder Cancer  Apoptosis  Phlpp2  C-jun