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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
作者:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
Adobe PDF(1403Kb)  |  收藏  |  浏览/下载:295/1  |  提交时间:2017/07/24
Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
Canescones A-E: aromatic polyketide dimers with PTP1B inhibitory activity from Penicillium canescens 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 18, 页码: 3274-3281
作者:  Zang, Yi;  Gong, Yi-Hua;  Li, Xu-Wen;  Li, Xiao-Nian;  Liu, Jun-Jun;  Chen, Chun-Mei;  Zhou, Yuan;  Gu, Liang-Hu;  Luo, Zeng-Wei;  Wang, Jian-Ping;  Sun, Wei-Guang;  Zhu, Hu-Cheng;  Zhang, Yong-Hui
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Synergistic use of NMR computation and quantitative interproton distance analysis in the structural determination of neokadcoccitane A, a rearranged triterpenoid featuring an aromatic ring D from Kadsura coccinea 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 10, 页码: 1619-1626
作者:  Xu, Hou-Chao;  Hu, Kun;  Shi, Xiao-Huo;  Tang, Jian-Wei;  Li, Xiao-Nian;  Sun, Han-Dong;  Puno, Pema-Tenzin
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Ganolearic Acid A, a Hexanorlanostane Triterpenoid with a 3/5/6/5-Fused Tetracyclic Skeleton from Ganoderma cochlear 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 83, 期号: 21, 页码: 13178-13183
作者:  Peng, Xing-Rong;  Huang, Yan-Jie;  Lu, Shuang-Yang;  Yang, Jing;  Qiu, Ming-Hua
浏览  |  Adobe PDF(319Kb)  |  收藏  |  浏览/下载:538/160  |  提交时间:2018/12/18
Virtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2017, 卷号: 70, 页码: 186-190
作者:  Zhang, Wen;  Qiu, Kai-Xiong;  Yu, Fang;  Xie, Xiao-Guang;  Zhang, Shu-Qun;  Chen, Ya-Juan;  Xie, Hui-Ding
浏览  |  Adobe PDF(371Kb)  |  收藏  |  浏览/下载:150/26  |  提交时间:2017/12/11
B-raf Kinase Inhibitors  Virtual Screening  Pharmacophore  Molecular Docking  3d Qsar  Binding Free Energy Calculation  
Structure and Function of the PriC DNA Replication Restart Protein 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2016, 卷号: 291, 期号: 35, 页码: 18384-18396
作者:  Wessel, Sarah R.;  Cornilescu, Claudia C.;  Cornilescu, Gabriel;  Metz, Alice;  Leroux, Maxime;  Hu, Kaifeng;  Sandler, Steven J.;  Markley, John L.;  Keck, James L.
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Dna Helicase  Dna Replication  Dna-protein Interaction  Nuclear Magnetic Resonance (Nmr)  Protein-protein Interaction  Dna Replication Restart  Dnab Helicase  Pric  Single-stranded Dna-binding Protein  
Enantiomeric Lignans and Neolignans from Phyllanthus glaucus: Enantioseparation and Their Absolute Configurations 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:  Wu, Zhaodi;  Lai, Yongji;  Zhou, Lei;  Wu, Ye;  Zhu, Hucheng;  Hu, Zhengxi;  Yang, Jing;  Zhang, Jinwen;  Wang, Jianping;  Luo, Zengwei;  Xue, Yongbo;  Zhang, Yonghui
浏览  |  Adobe PDF(1383Kb)  |  收藏  |  浏览/下载:184/52  |  提交时间:2016/08/22
New Anti-angiogenic Leading Structure Discovered in the Fruit of Cimicifuga yunnanensis 期刊论文
SCIENTIFIC REPORTS, 2015, 卷号: 5, 页码: 9026
作者:  Nian, Yin;  Yang, Jing;  Liu, Tong-Yang;  Luo, Ying;  Zhang, Ji-Hong;  Qiu, Ming-Hua;  Qiu,MH (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  zhjihong2000@126.com;  mhchiu@mail.kib.ac.cn
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Hyperattenins A-I, bioactive polyprenylated acylphloroglucinols from Hypericum attenuatum Choisy 期刊论文
RSC ADVANCES, 2015, 卷号: 5, 期号: 7, 页码: 5277-5287
作者:  Li,Dongyan;  Xue,Yongbo;  Zhu,Hucheng;  Li,Yan;  Sun,Bin;  Liu,Junjun;  Yao,Guangmin;  Zhang,Jinwen;  Du,Guang;  Zhang,Yonghui;  Zhang,YH (reprint author),Huazhong Univ Sci & Technol,Sch Pharm,Tongji Med Coll,Hubei Key Lab Nat Med Chem & Resource Evaluat,Wuhan 430030,Peoples R China.
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Scapiformolactones A-I: Germacrane sesquiterpenoids with an unusual Delta(3)-15,6-lactone moiety from Salvia scapiformis 期刊论文
PHYTOCHEMISTRY, 2013, 卷号: 96, 页码: 378-388
作者:  Lai, Yongji;  Xue, Yongbo;  Zhang, Mengke;  Zhang, Jinwen;  Tang, Wei;  Liu, Junjun;  Lei, Liang;  Yan, Juming;  Luo, Zengwei;  Zuo, Jianping;  Li, Yan;  Yao, Guangmin;  Zhang, Yonghui
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Salvia Scapiformis  Lamiaceae  Germacrane Sesquiterpene  Conformation  Chemical Transformation  Quantum Mechanical Calculation  Cytotoxicity Immunomodulatory Activity