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中国科学院昆明植物研究所知识管理系统
Knowledge Management System of Kunming Institute of Botany,CAS
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植物化学与西部植物... [11]
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李艳 [11]
胡江苗 [3]
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Design, Synthesis, and Biological Evaluation of Novel Biotinylated Podophyllotoxin Derivatives as Potential Antitumor Agents
期刊论文
FRONTIERS IN CHEMISTRY, 2019, 卷号: 7, 页码: 14
作者:
Zi, Cheng-Ting
;
Gao, Yin-Sheng
;
Yang, Liu
;
Feng, Shu-Yun
;
Huang, Yue
;
Sun, Li
;
Jin, Yi
;
Xu, Feng-Qing
;
Dong, Fa-Wu
;
Li, Yan
;
Ding, Zhong-Tao
;
Zhou, Jun
;
Jiang, Zi-Hua
;
Yuan, Sheng-Tao
;
Hu, Jiang-Miao
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Adobe PDF(1387Kb)
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浏览/下载:274/63
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提交时间:2019/07/29
podophyllotoxin derivatives
biotin
anticancer activity
synthesis
apoptosis
Synthesis and antitumor activity of biotinylated camptothecin derivatives as potent cytotoxic agents
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 2, 页码: 234-237
作者:
Zi, Cheng-Ting
;
Yang, Liu
;
Xu, Feng-Qing
;
Dong, Fa-Wu
;
Ma, Rui-Jing
;
Li, Yan
;
Zhou, Jun
;
Ding, Zhong-Tao
;
Jiang, Zi-Hua
;
Hu, Jiang-Miao
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浏览/下载:457/199
  |  
提交时间:2019/03/18
Biodnylated Camptothecin Derivatives
Anticancer Activity
Synthesis
Click Chemistry
Structure-activity Relationships (Sars)
One-Step Semisynthesis of a Segetane Diterpenoid from a Jatrophane Precursor via a Diels-Alder Reaction
期刊论文
ORGANIC LETTERS, 2016, 卷号: 18, 期号: 3, 页码: 496-499
作者:
Wan, Luo-Sheng
;
Shao, Li-Dong
;
Fu, Liangbing
;
Xu, Jun
;
Zhu, Guo-Lei
;
Peng, Xing-Rong
;
Li, Xiao-Nian
;
Li, Yan
;
Qiu, Ming-Hua
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Adobe PDF(584Kb)
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浏览/下载:223/63
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提交时间:2016/06/27
New Labdane diterpenes from Hedychium yunnanense with cytotoxicity and inhibitory effects on nitric oxide production
期刊论文
NATURAL PRODUCT RESEARCH, 2016, 卷号: 30, 期号: 23, 页码: 2669-2674
作者:
Li, Yu-Peng
;
Zhao, Si-Meng
;
Xu, Jun-Ju
;
Zeng, Guang-Zhi
;
Li, Yan
;
Tan, Ning-Hua
;
Yang, Ye
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Adobe PDF(900Kb)
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浏览/下载:242/51
  |  
提交时间:2017/01/05
Zingiberaceae
Hedychium Yunnanense
Labdane Diterpenes
Inhibition Of No Production
Cytotoxicity
Mangiferin and its aglycone, norathyriol, improve glucose metabolism by activation of AMP-activated protein kinase
期刊论文
PHARMACEUTICAL BIOLOGY, 2014, 卷号: 52, 期号: 1, 页码: 68-73
作者:
Wang, Fang
;
Yan, Juming
;
Niu, Yanfen
;
Li, Yan
;
Lin, Hua
;
Liu, Xu
;
Liu, Jikai
;
Li, Ling
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Adobe PDF(383Kb)
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浏览/下载:295/64
  |  
提交时间:2014/04/09
Active Metabolite
Ampk
Insulin Resistance
L6 Muscle Cells
Norathyriol
Cytotoxicity of naturally occurring rhamnofolane diterpenes from Jatropha curcas
期刊论文
PHYTOCHEMISTRY, 2013, 卷号: 96, 页码: 265-272
作者:
Liu, Jie-Qing
;
Yang, Yuan-Feng
;
Li, Xu-Yang
;
Liu, En-Qian
;
Li, Zhong-Rong
;
Zhou, Lin
;
Li, Yan
;
Qiu, Ming-Hua
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  |  
Adobe PDF(915Kb)
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浏览/下载:303/103
  |  
提交时间:2015/05/14
Jatropha Curcas
Euphorbiaceae
Rhamnofolane Diterpenoids
Cytotoxicity
Synthesis and Anticancer Activity of Glucosylated Podophyllotoxin Derivatives Linked via 4 beta-Triazole Rings
期刊论文
MOLECULES, 2013, 卷号: 18, 期号: 11, 页码: 13992-14012
作者:
Zi, Cheng-Ting
;
Xu, Feng-Qing
;
Li, Gen-Tao
;
Li, Yan
;
Ding, Zhong-Tao
;
Zhou, Jun
;
Jiang, Zi-Hua
;
Hu, Jiang-Miao
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Adobe PDF(404Kb)
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浏览/下载:194/52
  |  
提交时间:2015/05/13
Podophyllotoxin
4 Beta-triazole Ring
Click Chemistry
Anticancer Activity
Three unusual sesquineolignans from Alpinia conchigera
期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2013, 卷号: 15, 期号: 8, 页码: 833-839
作者:
Xu, Jun-Ju
;
Zhao, Hong-Mei
;
Shen, Yong
;
Chen, Jian-Hua
;
Li, Yan
;
Tan, Ning-Hua
;
Yang, Sheng-Chao
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Adobe PDF(118Kb)
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浏览/下载:213/51
  |  
提交时间:2013/10/16
Zingiberaceae
Alpinia Conchigera
Sesquineolignans
Conchignans A-c
Apoptosis induction and G2/M arrest of 2-methyl-1,3,6-trihydroxy-9,10-anthraquinone from Rubia yunnanensis in human cervical cancer HeLa cells
期刊论文
PHARMAZIE, 2013, 卷号: 68, 期号: 4, 页码: 293-299
作者:
Zeng, Guang-Zhi
;
Fan, Jun-Ting
;
Xu, Jun-Ju
;
Li, Yan
;
Tan, Ning-Hua
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Adobe PDF(6299Kb)
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浏览/下载:276/46
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提交时间:2015/05/14
One Of The Major compOnents Isolated From The Traditional
2-methyl-1
Chinese Medicine Rubia Yunnanensis
3
Exhibited Inhibitory Activity On The proliferatiOn Of Several
6-trihydroxy-9
HumAn CAncer Cell Lines. The Results From An Annexin V-fitc (fluoresein-5-isothiocyAnate) Apoptosis Assay
10-anthraquinone (Mta)
And Dna Content Analysis Showed That Mta Exerted Cytotoxicity Via Apoptosis Induction And G2/m Cell Cycle
Arrest In Human Cervical carcInoma Hela Cells. Further
Mta Was Found To Induce apopTosis Of Hela Cells
Through The MITochondria-mediated Pathway. It Caused The Translocation Of Bax To The mITochondria And
Release Of Cytochrome c Into The Cytosol
Which Caused The Cleavage Of Caspase And Poly(Adp-ribose)
Polymerase And Finally Triggered The Apoptosis. furThermore
The P53/p21/cdc2-cyclin B1 Signaling Was
Found Related To The G2/m Arrest Caused By Mta. The Over-expression Of P21 And Down-expression Of
Cyclin B1 Caused By Mta Inactivated The cdc2-Cyclin B1 Complex Of G2/m Checkpoint And Finally Caused
The G2/m Arrest In Hela Cells. ThIs Study Demonstrated That Mta Is a Potential Anti-cancer Component Of
R. Yunnanensis
a Folk Anti-cancer Herb Used In Yunnan
China.
Gelsemium alkaloids, immunosuppressive agents from Gelsemium elegans
期刊论文
FITOTERAPIA, 2012, 卷号: 83, 期号: 6, 页码: 1120-1124
作者:
Xu, You-Kai
;
Liao, Shang-Gao
;
Na, Zhi
;
Hu, Hua-Bin
;
Li, Yan
;
Luo, Huai-Rong
Adobe PDF(604Kb)
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浏览/下载:300/91
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提交时间:2012/11/30
Gelsemium Elegant
21-(2-oxopropyl)-koumine
11-methoxygelselegine
Immunosuppressive Activity