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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:96/21  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Huperserratines A and B, Two Macrocyclic Lycopodium Alkaloids with an Unusual Skeleton from Huperzia serrata 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020
作者:  Wu, Xing-De;  Li, Xiao-Nian;  Peng, Li-Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1810Kb)  |  收藏  |  浏览/下载:172/68  |  提交时间:2021/01/05
Phlegmadine A: A Lycopodium Alkaloid with a Unique Cyclobutane Ring from Phlegmariurus phlegmaria 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 期号: 17, 页码: 11301-11305
作者:  Zhang, Zhi-Jun;  Wang, Chen;  Wu, Xing-De;  Huang, Yan;  Zhou, Wen-Xia;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1540Kb)  |  收藏  |  浏览/下载:216/21  |  提交时间:2019/11/07
Diterpenoids and sesquiterpenoids from the stem bark of Metasequoia glyptostroboides 期刊论文
PHYTOCHEMISTRY, 2019, 卷号: 161, 页码: 86-96
作者:  Tu, Wen-Chao;  Qi, Yan-Yan;  Ding, Lin-Fen;  Yang, Hui;  Liu, Jiang-Xin;  Peng, Li-Yan;  Song, Liu-Dong;  Gong, Xun;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1045Kb)  |  收藏  |  浏览/下载:234/73  |  提交时间:2019/07/29
Metasequoia glyptostroboides Hu & WC Cheng  Cupressaceae  Sesquiterpenoids  Diterpenoids  Cytotoxicity  
A practical total synthesis of (+/-)-cermizine D and a formal synthesis of (+/-)-cermizine C 期刊论文
JOURNAL OF CHEMICAL RESEARCH, 2018, 期号: 5, 页码: 274-279
作者:  Shi, Xin;  Bao, Ying;  Deng, Zhen-Tao;  Zhu, Yu;  Shao, Li-Dong;  Zhang, Hong-Bin;  Zhao, Qin-Shi
收藏  |  浏览/下载:242/0  |  提交时间:2018/07/30
Cermizine c  Cermizine d  Total Synthesis  Michael Addition  Reductive Amination  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:390/43  |  提交时间:2017/12/18
Total Synthesis of (+/-)-Cermizine B 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 82, 期号: 20, 页码: 11110-11116
作者:  Shi, Xin;  Deng, Zhen-Tao;  Zhu, Yu;  Bao, Ying;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:194/47  |  提交时间:2017/12/18
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:316/73  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
A biomimetic semisynthesis enables structural elucidation of selaginellin U: a tautomeric cyclic alkynylphenol from Selaginella tamariscina 期刊论文
ROYAL SOCIETY OPEN SCIENCE, 2017, 卷号: 4, 期号: 7, 页码: 170352
作者:  Zhu, Qin-Feng;  Bao, Ying;  Zhang, Zhi-Jun;  Su, Jia;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(698Kb)  |  收藏  |  浏览/下载:169/23  |  提交时间:2017/10/23
Biomimetic Semisynthesis  Structural Elucidation  Selaginellins  Alkynylphenol  Selaginella Tamariscina  
Five new Lycopodium alkaloids from the aerial parts of Phlegmariurus henryi 期刊论文
FITOTERAPIA, 2016, 卷号: 115, 期号: 1, 页码: 148-154
作者:  Liu, Yu-Chen;  Su, Jia;  Wu, Xing-De;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  He, Juan;  Li, Xiao-Nian;  Peng, Li-Yan;  Cheng, Xiao;  Zhao, Qin-Shi
浏览  |  Adobe PDF(964Kb)  |  收藏  |  浏览/下载:251/57  |  提交时间:2017/02/14
Phlegmariurus Henryi  Lycopodium Alkaloids  Anti-ache Activity  Cytotoxicity