KIB OpenIR

浏览/检索结果: 共271条,第1-10条 帮助

已选(0)清除 条数/页:   排序方式:
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:305/1  |  提交时间:2017/07/24
YC-1 inhibits proliferation of breast cancer cells by downregulating EZH2 expression via activation of c-Cbl and ERK 期刊论文
出版物, 3111, 期号: 0, 页码: 1-46
作者:  Ling-Chu Chang;  Hui-Yi Lin;  Meng-Tung Tsai;  Ruey-Hwang Chou;  Fang-Yu Lee;  Che-Ming Teng;  Min-Tsang Hsieh;  Hsin-Yi Hung;  Li-Jiau Huang;  Yung-Luen Yu;  Sheng-Chu Kuo
Adobe PDF(1357Kb)  |  收藏  |  浏览/下载:323/1  |  提交时间:2017/07/24
Yc-1  Triple-negative Breast Cancer  Erk  Ezh2  C-cbl  
Oligosaccharide Blocks PAR1 (Proteinase-Activated Receptor 1)-PAR4-Mediated Platelet Activation by Binding to Thrombin Exosite II and Impairs Thrombosis 期刊论文
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY, 2023, 卷号: 43, 期号: 2, 页码: 253-266
作者:  Li,Sujuan;  Wang,Weili;  Lin,Lisha;  Yang,Lian;  Cai,Ying;  Yang,Xingzhi;  Zhang,Taocui;  Xiao,Chuang;  Yan,Hui;  Gao,Na;  Zhao,Jinhua
浏览  |  Adobe PDF(2610Kb)  |  收藏  |  浏览/下载:27/4  |  提交时间:2024/05/09
oligosaccharide  platelet activation  receptor  protease-activated  thrombin thrombosis  ANTIPLATELET THERAPIES  ALLOSTERIC LINKAGE  TISSUE FACTOR  PROTEASE  VORAPAXAR  MECHANISM  REVEALS  SITE  
重楼属中富含偏诺甾体皂苷的植物资源挖掘及其研究 学位论文
: 中国科学院大学, 2022
作者:  余玲玲
Adobe PDF(11095Kb)  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/05/14
重楼属 (Paris L.),黑药花科,偏诺皂苷,球药隔重楼,LC-MS/MS,诱导血小板聚集活性  Paris L., Melanthiaceae, Pennogenin saponins, Paris fargesii, LC-MS/MS, Inducing platelet aggregation activity  
FG 寡糖对血小板蛋白酶激活受体的阻断作用及机制研究 学位论文
: 中国科学院大学, 2022
作者:  李素娟
Adobe PDF(5079Kb)  |  收藏  |  浏览/下载:171/0  |  提交时间:2024/05/14
血小板活化,蛋白酶激活受体,凝血酶外位点 II,血栓,岩藻糖化糖胺 聚糖  Platelet activation, Protease-activated receptor, Thrombin exosite II, Thrombosis, Fucosylated glycosaminoglycan  
岩藻糖化糖胺聚糖 系统给药的毒性作用及其相关的血小板激活作用与机制 学位论文
: 中国科学院大学, 2022
作者:  林丽莎
Adobe PDF(5816Kb)  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/05/14
岩藻糖化糖胺聚糖,毒性机制,血小板聚集,构效关系,血小板受体  Fucosylated glycosaminoglycan, Toxic effect, Platelet aggregation, Structure-activity relationship, Platelet receptor  
抗血小板活性松香烷二萜的合成、结构优化及机制研究 学位论文
: 中国科学院大学, 2022
作者:  夏凡
Adobe PDF(4437Kb)  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/05/14
康定鼠尾草,松香烷二萜,抗血小板活性,合成和结构优化研究  Salvia prattii, Abietane diterpenoid, Antiplatelet aggregation activity, Synthesis and structure optimization  
Discovery of novel coffee diterpenoids with inhibitions on Ca(v)3.1 low voltage-gated Ca2+ channel 期刊论文
FOOD CHEMISTRY, 2022, 卷号: 376, 页码: 131923
作者:  Hu,Guilin;  Dong,Ding;  Du,Shuzong;  Peng,Xingrong;  Wu,Mingkun;  Shi,Qiangqiang;  Hu,Kun;  Hong,Defu;  Wang,Xiaoyuan;  Zhou,Lin;  Nian,Yin;  Qiu,Minghua
浏览  |  Adobe PDF(4722Kb)  |  收藏  |  浏览/下载:168/42  |  提交时间:2022/04/02
Coffea arabica L  Roasted coffee  Coffee diterpenoid  Cafestol  Kahweol  T-type Ca2+ channels  Ca(v)3.1 low voltage-gated Ca2+ channel  Ca(v)3.1 inhibitors  CALCIUM-CHANNELS  CAFESTOL  KAHWEOL  PHYSIOLOGY  ESTERS  NOMENCLATURE  PHARMACOLOGY  APOPTOSIS  FURANS  
Kadsura longipedunculata Finet & Gagnepain (Schisandraceae): An Overview of Botany, Traditional Uses, Phytochemistry and Pharmacological Activities 期刊论文
FORESTS, 2022, 卷号: 13, 期号: 8, 页码: 1281
作者:  Idrees, Muhammad;  Zhang, Zhiyong;  Yaseen, Aftab;  Jiao, Yongqing;  Zheng, Xu
浏览  |  Adobe PDF(1340Kb)  |  收藏  |  浏览/下载:10/2  |  提交时间:2024/04/30
Kadsura longipedunculata  phytochemistry  pharmacology  medicinal plant  LOWERS SERUM-CHOLESTEROL  ESSENTIAL OILS  DIBENZOCYCLOOCTADIENE LIGNANS  TRITERPENE DILACTONES  CHEMICAL-CONSTITUENTS  STRUCTURE ELUCIDATION  GENUS KADSURA  HETEROCLITA  STEMS  5-ALPHA-CHOLEST-8(14)-EN-3-BETA-OL-15-ONE  
丫蕊花中水溶性皂苷的制备及其活性评价 学位论文
, 2021
作者:  张仕娟
Adobe PDF(5526Kb)  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/03/20