KIB OpenIR

浏览/检索结果: 共189条,第1-10条 帮助

已选(0)清除 条数/页:   排序方式:
Pharmacology and anti-addiction effects of the novel kappa opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin A 期刊论文
出版物, 3111, 期号: 0, 页码: 1-53
作者:  B Simonson;  A S Morani;  A W M Ewald;  L Walker;  N Kumar;  D Simpson;  J H Miller;  T E Prisinzano;  B M Kivell
Adobe PDF(1394Kb)  |  收藏  |  浏览/下载:297/1  |  提交时间:2017/07/24
FXR activation prevents liver injury induced by Tripterygium wilfordii preparations 期刊论文
XENOBIOTICA, 2021, 卷号: 51, 期号: 6, 页码: 716-727
作者:  Peng,Wan;  Dai,Man-Yun;  Bao,Li-Juan;  Zhu,Wei-Feng;  Li,Fei
浏览  |  Adobe PDF(2010Kb)  |  收藏  |  浏览/下载:106/15  |  提交时间:2022/04/02
Tripterygium wilfordii  liver injury  farnesoid X receptor  bile acid metabolism  metabolomics  
A Cryptic Plant Terpene Cyclase Producing Unconventional 18-and 14-Membered Macrocyclic C-25 and C-20 Terpenoids with Immunosuppressive Activity 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 卷号: 60, 期号: 48, 页码: 25468-25476
作者:  Chen,Yue-Gui;  Li,De-Sen;  Ling,Yi;  Liu,Yan-Chun;  Zuo,Zhi-Li;  Gan,Li-She;  Luo,Shi-Hong;  Hua,Juan;  Chen,Ding-Yuan;  Xu,Fan;  Li,Man;  Guo,Kai;  Liu,Yan;  Gershenzon,Jonathan;  Li,Sheng-Hong
浏览  |  Adobe PDF(2177Kb)  |  收藏  |  浏览/下载:118/58  |  提交时间:2022/04/02
enzyme engineering  immunosuppressive activity  Leucosceptrum canum  macrocyclic terpenoids  sesterterpene synthase  GERANYLFARNESYL DIPHOSPHATE SYNTHASE  GLANDULAR TRICHOMES  LEUCOSCEPTRUM-CANUM  SCALE INSECT  SESTERTERPENOIDS  CONVERSION  EVOLUTION  PRECURSOR  HARBOR  
CtBP1/2 differentially regulate genomic stability and DNA repair pathway in high-grade serous ovarian cancer cell 期刊论文
ONCOGENESIS, 2021, 卷号: 10, 期号: 7, 页码: 49
作者:  He,YingYing;  He,Zhicheng;  Lin,Jian;  Chen,Cheng;  Chen,Yuanzhi;  Liu,Shubai
浏览  |  Adobe PDF(3008Kb)  |  收藏  |  浏览/下载:79/13  |  提交时间:2022/04/02
BINDING-PROTEIN CTBP  TRANSCRIPTIONAL COREPRESSOR  NEGATIVE MODULATION  PROMOTES APOPTOSIS  GENE-EXPRESSION  DAMAGE RESPONSE  PK  OVEREXPRESSION  PHOSPHOPROTEIN  TRANSFORMATION  
Discovery of novel inhibitors against main protease (Mpro) of SARS-CoV-2 via virtual screening and biochemical evaluation 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 104767
作者:  Guo,Sheng;  Xie,Hang;  Lei,Yu;  Liu,Bin;  Zhang,Li;  Xu,Yechun;  Zuo,Zhili
浏览  |  Adobe PDF(3181Kb)  |  收藏  |  浏览/下载:88/29  |  提交时间:2022/04/02
SARS-CoV-2  Main protease  Virtual screening  Biochemical evaluation  
Discovery of pseudolaric acid A as a new Hsp90 inhibitor uncovers its potential anticancer mechanism 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 112, 页码: 104963
作者:  Liu,Jiangxin;  Wu,Xing-De;  Li,Wenyan;  Yuan,Zaifeng;  Yang,Kun;  Zhao,Qin-Shi
浏览  |  Adobe PDF(3665Kb)  |  收藏  |  浏览/下载:69/9  |  提交时间:2022/04/02
Pseudolaric acid A  Hsp90 inhibitor  Apoptosis  NMR  Structure-activity relationship  Photoaffinity-based probe  Protein-ligand interaction  MOLECULAR CHAPERONE  PROTEIN  TARGET  CANCER  KINASE  NMR  IDENTIFICATION  SELECTIVITY  BINDING  DESIGN  
月季连续开花调控候选基因WD40-60功能探究 学位论文
, 2020
作者:  孙弋博
Adobe PDF(6926Kb)  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/11/02
颗粒野生稻与同源四倍体水稻的基因组变异与进化 学位论文
, 2020
作者:  施聪
Adobe PDF(13080Kb)  |  收藏  |  浏览/下载:29/0  |  提交时间:2023/11/02
新颖USP7抑制剂Parthenolide的发现及抗结直肠肿瘤研究 学位论文
, 2020
作者:  李雪
Adobe PDF(11623Kb)  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/11/02
Isowalsuranolide(HXJ-2351)诱导溶酶体生成及细胞凋亡的分子机制研究 学位论文
, 2020
作者:  陈远志
Adobe PDF(4328Kb)  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/11/02