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First total synthesis of rhuscholide A, glabralide B and denudalide 期刊论文
TETRAHEDRON LETTERS, 2019, 卷号: 60, 期号: 38, 页码: 4
作者:  Li, Tian-Ze;  Geng, Chang-An;  Chen, Ji-Jun
浏览  |  Adobe PDF(709Kb)  |  收藏  |  浏览/下载:244/45  |  提交时间:2019/11/07
Total synthesis  Rhuscholide A  Glabralide B  Denudalide  
Polybenzyls from Gastrodia elata, their agonistic effects on melatonin receptors and structure-activity relationships 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3299-3306
作者:  Chen, Si-Yue;  Geng, Chang-An;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Yang, Xiao-Tong;  Su, Li-Hua;  He, Xiao-Feng;  Li, Tian-Ze;  Deng, Zhen-Tao;  Gao, Zhen;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(1837Kb)  |  收藏  |  浏览/下载:192/35  |  提交时间:2019/09/10
Gastrodia elata  Polybenzyls  Melatonin receptors  Structure-activity relationships  Docking study  
Anti-hepatitis B virus effects of the traditional Chinese herb Arteinisia capillaris and its active enynes 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2018, 卷号: 224, 页码: 283-289
作者:  Geng, Chang-An;  Yang, Tong-Hua;  Huang, Xiao-Yan;  Yang, Jing;  Ma, Yun-Bao;  Li, Tian-Ze;  Zhang, Xue-Mei;  Chen, Ji-Jun
收藏  |  浏览/下载:257/0  |  提交时间:2018/09/27
Artemisia capillaris  Enynes  Anti-HBV activity  Structure-activity relationships  
Synthesis and biological evaluation of magnolol derivatives as melatonergic receptor agonists with potential use in depression 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 期号: 0, 页码: 381-393
作者:  Yang, Tong-Hua;  Ma, Yun-Bao;  Geng, Chang-An;  Yan, De-Xiu;  Huang, Xiao-Yan;  Li, Tian-Ze;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(2088Kb)  |  收藏  |  浏览/下载:221/71  |  提交时间:2018/10/04
Depression  Magnolol Derivatives  Mt1/2 Receptors  Metabolites  Monoamine Neurotransmitter  
(+/-)-Uncarilins A and B, Dimeric Isoechinulin-Type Alkaloids from Uncaria rhynchophylla 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2017, 卷号: 80, 期号: 4, 页码: 959-964
作者:  Geng, Chang-An;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Hou, Bo;  Li, Tian-Ze;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(1424Kb)  |  收藏  |  浏览/下载:349/87  |  提交时间:2017/08/29
Bioactivity-guided synthesis of gramine derivatives as new MT1 and 5-HT1A receptors agonists 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2017, 卷号: 19, 期号: 6, 页码: 610-622
作者:  Yin, Xiu-Juan;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Geng, Chang-An;  Li, Tian-Ze;  Chen, Xing-Long;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(2718Kb)  |  收藏  |  浏览/下载:333/60  |  提交时间:2017/07/10
Gramine  Melatonin Receptor  5-hydroxy-tryptamine Receptor  Agonistic Activity  Structure-activity Relationships  
LC-MS guided isolation of ent-kaurane diterpenoids from Nouelia insignis 期刊论文
FITOTERAPIA, 2016, 卷号: 111, 页码: 42-48
作者:  Sun, Chang-Li;  Geng, Chang-An;  Chen, Xing-Long;  Yang, Tong-Hua;  Yin, Xiu-Juan;  Huang, Xiao-Yan;  Peng, Hua;  Chen, Ji-Jun
Adobe PDF(830Kb)  |  收藏  |  浏览/下载:232/72  |  提交时间:2016/08/22
Nouelia Insignis  Lc-ms  Diterpenoids  Nitric Oxide Production Inhibitory Activity  
Bioactivity-guided synthesis of tropine derivatives as new agonists for melatonin receptors 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 51, 页码: 45059-45063
作者:  Yin, Xiu-Juan;  Geng, Chang-An;  Huang, Xiao-Yan;  Chen, Hao;  Ma, Yun-Bao;  Chen, Xing-Long;  Sun, Chang-Li;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(1380Kb)  |  收藏  |  浏览/下载:264/66  |  提交时间:2016/08/22
Design, Synthesis and Biological Evaluation of Caudatin Analogs as Potent Hepatitis B Virus Inhibitors 期刊论文
MEDICINAL CHEMISTRY, 2015, 卷号: 11, 期号: 2, 页码: 165-179
作者:  Wang, Li-Jun;  Chen, Hao;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Geng, Chang-An;  Zhang, Xue-Mei;  Chen, Ji-Jun;  Chen,JJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.
Adobe PDF(375Kb)  |  收藏  |  浏览/下载:203/70  |  提交时间:2015/06/29
Anti-hbv Activity  Caudatin Analogs  Hepatitis b e Antigen (Hbeag)  Hepatitis b Surface Antigen (Hbsag)  Hbv Dna Replication  Structure-activity Relationships(Sars)  Synthesis  
Polyacetylenes and anti-hepatitis B virus active constituents from Artemisia capillaris 期刊论文
FITOTERAPIA, 2014, 卷号: 95, 页码: 187-193
作者:  Zhao, Yong;  Geng, Chang-An;  Sun, Chang-Li;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Cao, Tuan-Wu;  He, Kang;  Wang, Hao;  Zhang, Xue-Mei;  Chen, Ji-Jun;  Chen,JJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  chenjj@mail.kib.ac.cn
Adobe PDF(441Kb)  |  收藏  |  浏览/下载:318/77  |  提交时间:2014/07/28
Polyacetylenes  Anti-hbv Activity  Artemisia Capillaris