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Design, Synthesis, and Structural Optimization of Lycorine-Derived Phenanthridine Derivatives as Wnt/beta-Catenin Signaling Pathway Agonists 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2016, 卷号: 79, 期号: 1, 页码: 180-188
作者:  Chen, Duo-Zhi;  Jing, Chen-Xu;  Cai, Jie-Yun;  Wu, Ji-Bo;  Wang, Sheng;  Yin, Jun -Lin;  Li, Xiao-Nian;  Li, Lin;  Hao, Xiao-Jiang
Adobe PDF(3043Kb)  |  收藏  |  浏览/下载:304/73  |  提交时间:2016/06/27
Synthesis and cytotoxic activity of novel 1-((indol-3-yl)methyl)-1H-imidazolium salts 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 21, 页码: 4926-4930
作者:  Xu, Xiao-Liang;  Wang, Jia;  Yu, Chun-Lei;  Chen, Wen;  Li, Ying-Chao;  Li, Yan;  Zhang, Hong-Bin;  Yang, Xiao-Dong;  Li,Y (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650204,Peoples R China.;  liyanb@mail.kib.ac.cn;  zhanghbyd@gmail.com;  xdyang@ynu.edu.cn
Adobe PDF(670Kb)  |  收藏  |  浏览/下载:375/88  |  提交时间:2014/11/25
Indole  Imidazolium Salts  Structure-activity Relationships  Cell Apoptosis  
Peganumine A, a beta-Carboline Dimer with a New Octacyclic Scaffold from Peganum harmala 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 15, 页码: 4028-4031
作者:  Wang, Kai-Bo;  Di, Ying-Tong;  Bao, Yu;  Yuan, Chun-Mao;  Chen, Gang;  Li, Da-Hong;  Bai, Jiao;  He, Hong-Ping;  Hao, Xiao-Jiang;  Pei, Yue-Hu;  Jing, Yong-Kui;  Li, Zhan-Lin;  Hua, Hui-Ming;  Li, ZL (reprint author), Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, Shenyang 110016, Liaoning, Peoples R China.;  lzl1030@hotmail.com;  huimhua@163.com
Adobe PDF(295Kb)  |  收藏  |  浏览/下载:302/89  |  提交时间:2014/10/11
Light-emitting-diodes  Alkaloid Extract  Potent  L.  Derivatives  Efficiency  Toxicity  Harmine  Cascade  Growth  
Synthesis, structure-activity relationships and biological evaluation of dehydroandrographolide and andrographolide derivatives as novel anti-hepatitis B virus agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 10, 页码: 2353-2359
作者:  Chen, Hao;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Geng, Chang-An;  Zhao, Yong;  Wang, Li-Jun;  Guo, Rui-Hua;  Liang, Wen-Juan;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(3861Kb)  |  收藏  |  浏览/下载:298/72  |  提交时间:2014/06/23
Anti-hbv Activity  DehydroAndrographolide And  Andrographolide Derivatives  Structure-activity Relationships  Octanol-water Partition Coefficients  
Nortriterpenoids from Schisandra chinensis and their absolute configurational assignments by electronic circular dichroism study 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 4, 页码: 859-868
作者:  Shi, Yi-Ming;  Wang, Li-Yan;  Zou, Xi-Sheng;  Li, Xiao-Nian;  Shang, Shan-Zhai;  Gao, Zhong-Hua;  Liang, Cheng-Qin;  Luo, Huai-Rong;  Li, Hong-Lin;  Xiao, Wei-Lie;  Sun, Han-Dong
Adobe PDF(1553Kb)  |  收藏  |  浏览/下载:551/61  |  提交时间:2014/04/09
Schisandra  Schisandra Chinensis  Nortriterpenoid  Electronic Circular Dichroism  Absolute Configuration  
Hybridaphniphyllines A and B, Daphniphyllum alkaloid and iridoid hybrids suggestive of Diels-Alder cycloaddition in Daphniphyllum longeracemosum 期刊论文
PHYTOCHEMISTRY, 2013, 卷号: 95, 页码: 428-435
作者:  Wang, Fei;  Mao, Mei-Fen;  Wei, Guo-Zhu;  Gao, Yuan;  Ren, Fu-Cai;  Liu, Ji-Kai
Adobe PDF(1128Kb)  |  收藏  |  浏览/下载:265/61  |  提交时间:2014/01/13
Daphniphyllum Longeracemosum  Daphniphyllaceae  C-22 Nor-daphniphyllum Alkaloid  Alkaloid And Iridoid Hybrid  Hybridaphniphylline  Diels-alder Cycloaddition  
Synthesis and antitumor activities of novel dibenzo[b,d]furan-imidazole hybrid compounds 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 66, 页码: 423-437
作者:  Liu, Lan-Xiang;  Wang, Xue-Quan;  Yan, Ju-Ming;  Li, Yan;  Sun, Cheng-Jun;  Chen, Wen;  Zhou, Bei;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Adobe PDF(3339Kb)  |  收藏  |  浏览/下载:332/141  |  提交时间:2013/10/16
Hybrid Compound  Imidazole  Dibenzo[b  Antitumor Activities  d]Furan  Structure-activity Relationships  
Synthesis and cytotoxic activities of novel hybrid 2-phenyl-3-alkylbenzofuran and imidazole/triazole compounds 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 卷号: 23, 期号: 15, 页码: 4297-4302
作者:  Chen, Wen;  Deng, Xiao-Yan;  Li, Yan;  Yang, Li-Juan;  Wan, Wei-Chao;  Wang, Xue-Quan;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Adobe PDF(820Kb)  |  收藏  |  浏览/下载:245/45  |  提交时间:2013/10/16
Hybrid Compound  Benzofuran  Imidazole  Triazole  Structure-activity Relationships  
Synthesis, biological evaluation and molecular modeling of substituted 2-aminobenzimidazoles as novel inhibitors of acetylcholinesterase and butyrylcholinesterase 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 14, 页码: 4218-4224
作者:  Zhu, Jinmei;  Wu, Chun-Feng;  Li, Xiaobing;  Wu, Gui-Sheng;  Xie, Shan;  Hu, Qian-Nan;  Deng, Zixin;  Zhu, Michael X.;  Luo, Huai-Rong;  Hong, Xuechuan
Adobe PDF(1174Kb)  |  收藏  |  浏览/下载:529/89  |  提交时间:2013/10/16
Alzheimer's Disease  Acetylcholinesterase  Butyrylcholinesterase  Molecular Modeling  2-aminobenzimidazole  
Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-kappa B Activation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4749-4757
作者:  Zhao, Yu;  Su, Jia;  Goto, Masuo;  Morris-Natschke, Susan L.;  Li, Yan;  Zhao, Qin-Shi;  Yao, Zhu-Jun;  Lee, Kuo-Hsiung
Adobe PDF(531Kb)  |  收藏  |  浏览/下载:302/63  |  提交时间:2013/10/16
Natural-products  Biological-activity  Cancer-therapy  Paclitaxel  Taxol  Resistance  Drugs  Chemotherapy  Parthenolide  Brevifoliol