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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
作者:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
Adobe PDF(1403Kb)  |  收藏  |  浏览/下载:451/1  |  提交时间:2017/07/24
Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
ABT-263 enhances sorafenib-induced apoptosis associated with Akt activity and the expression of Bax and p21 (CIP1/WAF1) in human cancer cells1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-35
作者:  Jingru Li;  Yicheng Chen;  Jiali Wan;  Xin Liu;  Chunrong Yu;  Wenhua Li
Adobe PDF(1198Kb)  |  收藏  |  浏览/下载:365/1  |  提交时间:2017/07/24
Abt-263  Sorafenib  Combination Therapy  Cancer  
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:488/1  |  提交时间:2017/07/24
Pharmacological characterizationof tachykinin tetrabranched derivatives 期刊论文
出版物, 3111, 期号: 0, 页码: 1-36
作者:  Chiara Ruzza;  Anna Rizzi;  Davide Malfacini;  Maria Camilla Cerlesi;  Federica Ferrari;  Erika Marzola;  Caterina Ambrosio;  Cristina Gro;  Salvadori Severo;  Tommaso Costa;  Girolamo Calo;  Remo Guerrini
Adobe PDF(1277Kb)  |  收藏  |  浏览/下载:302/1  |  提交时间:2017/07/24
Tachykinins  Substance p  Pwt2-sp  Nk1 Receptor  Calcium Mobilization  Bioluminescence Resonance Energy Transfer  Guinea Pig Ileum  Rat Urinary Bladder  Nociceptive Behaviour Induced By Spinal Substance p  Mice  
Antidepressant and anxiolytic profiles of newly synthesized arginine vasopressin 期刊论文
出版物, 3111, 期号: 0, 页码: 1-62
作者:  M Iijima;  T Yoshimizu;  T Shimazaki;  K Tokugawa;  K Fukumoto;  S Kurosu;  T Kuwada;  Y Sekiguchi;  S Chaki
Adobe PDF(776Kb)  |  收藏  |  浏览/下载:245/2  |  提交时间:2017/07/24
Arginine Vasopressin  V1b Receptor Antagonist  Depression  Anxiety  Hpa Axis  
Artematrolide A inhibited cervical cancer cell proliferation via ROS/ERK/mTOR pathway and metabolic shift 期刊论文
PHYTOMEDICINE, 2021, 卷号: 91, 页码: 153707
作者:  Zhang,Xin-Tian;  Hu,Jing;  Su,Li-Hua;  Geng,Chang-An;  Chen,Ji-Jun
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Artemisia atrovirens  Cervical cancer  ERK pathway  Cell metabolism  ALKALINE-PHOSPHATASE  SIGNALING PATHWAY  DIFFERENTIATION  APOPTOSIS  ERK  MECHANISMS  
Rubinoboletus ballouii polysaccharides exhibited immunostimulatory activities through toll-like receptor-4 via NF-kappa B pathway 期刊论文
PHYTOTHERAPY RESEARCH, 2021, 卷号: 35, 期号: 4, 页码: 2108-2118
作者:  Li,Long-Fei;  Yue,Grace G-L;  Chan,Ben C-L;  Zeng,Qiang;  Han,Quan-Bin;  Leung,Ping-Chung;  Fung,Kwok-Pui;  Liu,Ji-Kai;  Lau,Clara B-S
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immunostimulatory effects  immunosuppression  myelosuppression  polysaccharide  Rubinoboletus ballouii  toll‐  like receptor‐  4  GANODERMA-LUCIDUM  DENDRITIC CELLS  IN-VITRO  ANTITUMOR  MUSHROOMS  
A natural acylphloroglucinol triggered antiproliferative possessions in HEL cells by impeding STAT3 signaling and attenuating angiogenesis in transgenic zebrafish model 期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2021, 卷号: 141, 页码: 111877
作者:  Hu,Mi;  Varier,Krishnapriya M.;  Li,Zhicao;  Qin,Xujie;  Rao,Qing;  Song,Jingrui;  Hu,Anling;  Hang,Yubing;  Yuan,Chunmao;  Gajendran,Babu;  Shu,Liping;  Wen,Min;  Li,Yanmei;  Liu,Haiyang
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Acylphloroglucinol  HEL cells  Intrinsic apoptotic pathway  Anti-angiogenesis  STAT3  Flk-1  CALLISTEMON-CITRINUS  TUMOR ANGIOGENESIS  DNA  DERIVATIVES  ANTICANCER  APOPTOSIS  ACTIVATION  INHIBITORS  TARGETS  LEAVES  
Identified Three Interferon Induced Proteins as Novel Biomarkers of Human Ischemic Cardiomyopathy 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 卷号: 22, 期号: 23, 页码: 13116
作者:  Chen,Cheng;  Tian,Jiao;  He,Zhicheng;  Xiong,Wenyong;  He,Yingying;  Liu,Shubai
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ischemic cardiomyopathy  heart failure  WGCNA  interferon stimulated genes  IFIT2  3  MYOCARDIAL-INFARCTION  NETWORK ANALYSIS  GENE  
FPR2-based anti-inflammatory and anti-lipogenesis activities of novel meroterpenoid dimers from Ganoderma 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 105338
作者:  Peng,Xing-Rong;  Wang,Qian;  Wang,Hui-Rong;  Hu,Kun;  Xiong,Wen-Yong;  Qiu,Ming-Hua
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Ganoderma applanatum  Meroterpenoid dimers  Molecular docking  Anti-lipogenesis  FPR2-based inflammation  INDUCED INSULIN-RESISTANCE  ADIPOCYTE DIFFERENTIATION  OBESITY  INFLAMMATION  DEFICIENCY  MACROPHAGES  ACTIVATION  EXPRESSION  LIGAND  MICE