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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations Eph antagonist and angiogenesis 期刊论文
出版物, 3111, 期号: 0, 页码: 1-32
作者:  I Hassan-Mohamed;  C Giorgio;  M Incerti;  S Russo;  D Pala;  E B Pasquale;  P Vicini;  E Barocelli;  S Rivara;  M Mor;  A Lodola;  M Tognolini
Adobe PDF(1403Kb)  |  收藏  |  浏览/下载:458/1  |  提交时间:2017/07/24
Eph Kinase  Ephrin  Small Molecules  Angiogenesis  Bile Acid  Lithocholic Acid  
ABT-263 enhances sorafenib-induced apoptosis associated with Akt activity and the expression of Bax and p21 (CIP1/WAF1) in human cancer cells1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-35
作者:  Jingru Li;  Yicheng Chen;  Jiali Wan;  Xin Liu;  Chunrong Yu;  Wenhua Li
Adobe PDF(1198Kb)  |  收藏  |  浏览/下载:371/1  |  提交时间:2017/07/24
Abt-263  Sorafenib  Combination Therapy  Cancer  
Design and synthesis of guaianolide-germacranolide heterodimers as novel anticancer agents against hepatocellular carcinoma 期刊论文
DRUG DEVELOPMENT RESEARCH, 2023
作者:  Yan,Jia-Xin;  Li,Qi-Hao;  Li,Tian-Ze;  Huang,Zhi-Yan;  Ma,Yun-Bao;  Chen,Ji-Jun
浏览  |  Adobe PDF(7663Kb)  |  收藏  |  浏览/下载:175/35  |  提交时间:2024/07/10
antihepatoma effects  guaianolide-germacranolide heterodimers  PDGFRA  DERIVATIVES  
Artemdubinoids A-N: novel sesquiterpenoids with antihepatoma cytotoxicity from Artemisia dubia 期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 12, 页码: 902-915
作者:  Gao,Zhen;  Li,Tianze;  Ma,Yunbao;  Huang,Xiaoyan;  Geng,Changan;  Zhang,Xuemei;  Chen,Jijun
浏览  |  Adobe PDF(872Kb)  |  收藏  |  浏览/下载:175/31  |  提交时间:2024/07/22
Artemdubinoids A-N  Artemisia dubia  Sesquiterpenoids  Antihepatoma activity  
Design, synthesis, and biological evaluation of artemyrianolide H derivatives as potential antihepatoma agents 期刊论文
BIOORGANIC CHEMISTRY, 2023, 卷号: 137, 页码: 106617
作者:  Li,Tian-Ze;  Yang,Xiao-Tong;  Ma,Wen-Jing;  Ma,Yun-Bao;  Li,Feng-Jiao;  Wang,Yong-Cui;  Chen,Ji-Jun
浏览  |  Adobe PDF(9670Kb)  |  收藏  |  浏览/下载:194/47  |  提交时间:2024/07/22
Artemyrianolide H  Germacranolide derivatives  Antihepatoma activity  Apoptosis  DIMERS  
Artemiprinolides A-M, thirteen undescribed sesquiterpenoid dimers from Artemisia princeps and their antihepatoma activity 期刊论文
PHYTOCHEMISTRY, 2023, 卷号: 211, 页码: 113714
作者:  Su,Li-Hua;  Ma,Wen-Jing;  Ma,Yun-Bao;  Li,Tian-Ze;  Geng,Chang-An;  Dong,Wei;  He,Xiao-Feng;  Chen,Ji-Jun
浏览  |  Adobe PDF(7208Kb)  |  收藏  |  浏览/下载:191/52  |  提交时间:2024/07/22
Artemisia princeps Pamp  Sesquiterpenoid dimers  Artemiprinolides A-M  Antihepatoma activity  Apoptosis  FARNESYL-PROTEIN TRANSFERASE  ETHANOL EXTRACT  PAMPANINI  INHIBITORS  JACEOSIDIN  
多花蒿中流份 B 和 E 的抗肝癌活性成分研究 学位论文
: 中国科学院大学, 2022
作者:  张鑫
Adobe PDF(3975Kb)  |  收藏  |  浏览/下载:41/0  |  提交时间:2024/05/14
多花蒿,多花蒿素 A~L,吉玛烷型倍半萜,抗肝癌细胞毒活性  Artemisia myriantha, artemyrianosins A~L, germacrane sesquiterpenoids, antihepatoma activity  
茵陈蒿和牛尾蒿的抗肝纤维化与抗肝癌活性成分研究 学位论文
: 中国科学院大学, 2022
作者:  高振
Adobe PDF(11670Kb)  |  收藏  |  浏览/下载:183/0  |  提交时间:2024/05/14
茵陈蒿,牛尾蒿,茵陈香豆酸,倍半萜二聚体,倍半萜,抗肝纤维化活性,抗肝癌活性,细胞周期,凋亡  Artemisia capillaris, Artemisia dubia, Coumaric acids, Sesquiterpenoids, Sesquiterpenoid dimers, Antihepatic fibrosis effects, Antihepatoma activity, Cell cycle, Apoptosis  
愈创木烷倍半萜 ludartin 衍生物合成与抗 肝癌活性研究 学位论文
: 中国科学院大学, 2022
作者:  孙金金
Adobe PDF(7657Kb)  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/05/14
Ludartin 衍生物合成  Synthesis of ludartin derivatives, Antihepatoma activity, HepG2 cells, Huh7 cells  抗肝癌活性  HepG2 细胞  Huh7 细胞  
Artematrovirenolides A-D and Artematrolides S-Z, Sesquiterpenoid Dimers with Cytotoxicity against Three Hepatoma Cell Lines from Artemisia atrovirens 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2022, 卷号: 40, 期号: 1, 页码: 104-114
作者:  Su,Li-Hua;  Li,Tian-Ze;  Ma,Yun-Bao;  Geng,Chang-An;  Huang,Xiao-Yan;  Zhang,Xin;  Gao,Zhen;  Chen,Ji-Jun
浏览  |  Adobe PDF(2103Kb)  |  收藏  |  浏览/下载:348/86  |  提交时间:2022/04/02
Artemisia atrovirens  Sesquiterpenoid dimers  Structure elucidation  X-ray diffraction  Antihepatoma activity  GUAIANOLIDE  ARGYI