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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:92/20  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Activation of SIK1 by phanginin A inhibits hepatic gluconeogenesis by increasing PDE4 activity and suppressing the cAMP signaling pathway 期刊论文
MOLECULAR METABOLISM, 2020
作者:  Liu, Siwen;  Huang, Suling;  Wu, Xingde;  Feng, Ying;  Shen, Yu;  Zhao, Qin-shi;  Leng, Ying
浏览  |  Adobe PDF(3899Kb)  |  收藏  |  浏览/下载:122/34  |  提交时间:2021/01/05
Phlegmadine A: A Lycopodium Alkaloid with a Unique Cyclobutane Ring from Phlegmariurus phlegmaria 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 期号: 17, 页码: 11301-11305
作者:  Zhang, Zhi-Jun;  Wang, Chen;  Wu, Xing-De;  Huang, Yan;  Zhou, Wen-Xia;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1540Kb)  |  收藏  |  浏览/下载:210/21  |  提交时间:2019/11/07
Diterpenoids and sesquiterpenoids from the stem bark of Metasequoia glyptostroboides 期刊论文
PHYTOCHEMISTRY, 2019, 卷号: 161, 页码: 86-96
作者:  Tu, Wen-Chao;  Qi, Yan-Yan;  Ding, Lin-Fen;  Yang, Hui;  Liu, Jiang-Xin;  Peng, Li-Yan;  Song, Liu-Dong;  Gong, Xun;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1045Kb)  |  收藏  |  浏览/下载:234/73  |  提交时间:2019/07/29
Metasequoia glyptostroboides Hu & WC Cheng  Cupressaceae  Sesquiterpenoids  Diterpenoids  Cytotoxicity  
Vibsane-Type Diterpenoids from Viburnum odoratissimum and Their Cytotoxic and HSP90 Inhibitory Activities 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 5, 页码: 1800049
作者:  Zhu, Qin-Feng;  Qi, Yan-Yan;  Zhang, Zhi-Jun;  Fan, Min;  Bi, Ran;  Su, Jia;  Wu, Xing-De;  Shao, Li-Dong;  Zhao, Qin-Shi
收藏  |  浏览/下载:347/0  |  提交时间:2018/07/16
Vibsane-type Diterpenoids  Viburnum Odoratissimum  Cytotoxicity  Hsp90 Inhibitor  
Two New Anti-Proliferative C-18-Norditerpenes from the Roots of Podocarpus macrophyllus 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 4, 页码: e1800043
作者:  Qi, Yan-Yan;  Su, Jia;  Zhang, Zhi-Jun;  Li, Lai-Wei;  Fan, Min;  Zhu, Yu;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1080Kb)  |  收藏  |  浏览/下载:497/114  |  提交时间:2018/07/02
Podocarpus Macrophyllus  Norditerpenoid  Anti-proliferative Activity  Activity-guided Fractionation  Structure Revision  
Hypofolins A - L, ent-Labdane Diterpenoids from the Roots of Hypoestes phyllostachya "Pink Splash' 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 6, 页码: e1800124
作者:  Cheng, Bin;  Ding, Lin-Fen;  Yan, Tong;  Xie, Zhang-Qiao;  Zhang, Zhi-jun;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:154/78  |  提交时间:2019/03/29
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:385/42  |  提交时间:2017/12/18
New neo-clerodane diterpenoids with neurotrophic activity from the aerial parts of Salvia tiliifolia 期刊论文
FITOTERAPIA, 2017, 卷号: 123, 页码: 44-50
作者:  Fan, Min;  Bao, Ying;  Zhang, Zhi-Jun;  Zhang, Hong-Bin;  Zhao, Qin-Shi
浏览  |  Adobe PDF(515Kb)  |  收藏  |  浏览/下载:164/63  |  提交时间:2018/05/08
Salvia Tiliifolia  Neo-clerodane Diterpenoids  Neurotrophic Activities  Cytotoxicity  
Total Synthesis of (+/-)-Cermizine B 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 82, 期号: 20, 页码: 11110-11116
作者:  Shi, Xin;  Deng, Zhen-Tao;  Zhu, Yu;  Bao, Ying;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:193/47  |  提交时间:2017/12/18