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Design, Synthesis, and Evaluation of the COX-2 Inhibitory Activities of New 1,3-Dihydro-2H-indolin-2-one Derivatives 期刊论文
MOLECULES, 2023, 卷号: 28, 期号: 12, 页码: 4668
作者:  Pan,Taohua;  He,Maofei;  Deng,Lulu;  Li,Jiang;  Fan,Yanhua;  Hao,Xiaojiang;  Mu,Shuzhen
浏览  |  Adobe PDF(3057Kb)  |  收藏  |  浏览/下载:10/3  |  提交时间:2024/05/09
oxindoles  alpha,beta-unsaturated ketone  anti-inflammatory  COX-2 inhibitory activity  ANTIINFLAMMATORY ACTIVITY  NATURAL-PRODUCTS  OXINDOLE-DERIVATIVES  NITRIC-OXIDE  POTENT  CYCLOOXYGENASE-2  DISCOVERY  PAIN  LIABILITY  
Perforatactones D and E, two new C-20 quassinoids with potential activity to induce lysosomal biogenesis from the twigs of Harrisonia perforata (Blanco) Merr. 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2021, 卷号: 19, 期号: 44, 页码: 9637-9640
作者:  Liu,Shuai;  Zhang,Cui-Shan;  Ran,Xiao-Qian;  Tang,Xiao-Han;  Guo,Ya-Rong;  Yan,Ying;  Yao,Yong-Gang;  Hao,Xiao-Jiang;  Luo,Rong-Can;  Di,Ying-Tong
浏览  |  Adobe PDF(997Kb)  |  收藏  |  浏览/下载:96/31  |  提交时间:2022/04/02
PROMISING BIOLOGICAL-ACTIVITY  LIMONOIDS  CHROMONES  FRUITS  DRUG  
16-nor Limonoids from Harrisonia perforata as promising selective 11 beta-HSD1 inhibitors 期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6, 页码: 1
作者:  Xiao-HuiYan;  Yi, Ping;  Cao, Pei;  Yang, Shi-Ying;  Fang, Xin;  Zhang, Yu;  Wu, Bin;  Leng, Ying;  Di, Ying-Tong;  Lv, Yang;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(1151Kb)  |  收藏  |  浏览/下载:343/54  |  提交时间:2017/01/05
Design, Synthesis and Structure-Activity Relationship Optimization of Lycorine Derivatives for HCV Inhibition 期刊论文
SCIENTIFIC REPORTS, 2015, 卷号: 5
作者:  Chen,Duozhi;  Cai,Jieyun;  Cheng,Junjun;  Jing,Chenxu;  Yin,Junlin;  Jiang,Jiandong;  Peng,Zonggen;  Hao,Xiaojiang
浏览  |  Adobe PDF(833Kb)  |  收藏  |  浏览/下载:210/77  |  提交时间:2016/01/19
New acyclic diterpenoids from the fruits of Aphanamixis grandifolia and structure revision of nemoralisin B 期刊论文
PHYTOCHEMISTRY LETTERS, 2014, 卷号: 8, 页码: 81-85
作者:  Zhang, Hai-Yuan;  Yuan, Chun-Mao;  Cao, Ming-Ming;  Li, Xiao-Hui;  Li, Shun-Lin;  Zhang, Yu;  Hao, Xiao-Jiang;  He, Hong-Ping
Adobe PDF(350Kb)  |  收藏  |  浏览/下载:283/62  |  提交时间:2014/06/23
Aphanamixis Grandifolia  Meliaceae  Acyclic Diterpenoids  Structure Revision  
Spiramine derivatives induce apoptosis of Bax(-/-)/Bak(-/-) cell and cancer cells 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 8, 页码: 1884-1888
作者:  Yan, Chen;  Huang, Li;  Liu, Hong-Chun;  Chen, Duo-Zhi;  Liu, Hai-Yang;  Li, Xiao-Hui;  Zhang, Yu;  Geng, Mei-Yu;  Chen, Quan;  Hao, Xiao-Jiang
Adobe PDF(1562Kb)  |  收藏  |  浏览/下载:297/45  |  提交时间:2014/06/23
Spiramine Derivative  Bax(-/-)/bak(-/-) Cells  Alpha  Apoptosis  Beta-unsaturated Ketone  Cytotoxicity  
Asymmetric Synthesis of the Tricyclic Core of Calyciphylline A-Type Alkaloids via Intramolecular [3+2] Cycloaddition 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 4, 页码: 1076-1079
作者:  Wang, Lu;  Xu, Chen;  Chen, Li;  Hao, Xiaojiang;  Wang, David Zhigang
Adobe PDF(389Kb)  |  收藏  |  浏览/下载:278/62  |  提交时间:2014/04/09
Beta-hydroxy Ketones  Nitrile Oxide Cycloaddition  Daphniphyllum Alkaloids  Tetracyclic Core  Daphnilactone-b  Ring-system  Construction  Reduction  Delta-2-isoxazolines  Route  
A diterpenoid derivate compound targets selenocysteine of thioredoxin reductases and induces Bax/Bak-independent apoptosis 期刊论文
FREE RADICAL BIOLOGY AND MEDICINE, 2013, 卷号: 63, 期号: SI, 页码: 485-494
作者:  Liu, Jinhua;  Mu, Chenglong;  Yue, Wen;  Li, Jie;  Ma, Biao;  Zhao, Lixia;  Liu, Lei;  Chen, Quan;  Yan, Chen;  Liu, Haiyang;  Hao, Xiaojiang;  Zhu, Yushan
浏览  |  Adobe PDF(2679Kb)  |  收藏  |  浏览/下载:309/60  |  提交时间:2013/10/16
Thioredoxin Reductase  Bim  Ros  Apoptosis  Cancer  
New steroids and sesquiterpene from Turraea pubescens 期刊论文
FITOTERAPIA, 2013, 卷号: 90, 页码: 119-125
作者:  Yuan, Chun-Mao;  Tang, Gui-Hua;  Wang, Xiao-Ying;  Zhang, Yu;  Cao, Ming-Ming;  Li, Xiao-Hui;  Li, Yan;  Li, Shun-Lin;  Di, Ying-Tong;  He, Hong-Ping;  Hao, Xiao-Jiang;  Hua, Hui-Ming
Adobe PDF(899Kb)  |  收藏  |  浏览/下载:494/262  |  提交时间:2014/01/13
Turraea Pubescens  Meliaceae  Steroids  Sesquiterpene  Anti-inflammatory  
Alkaloids from the leaves of Daphniphyllum longeracemosum 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2006, 卷号: 69, 期号: 7, 页码: 1074-1076
作者:  Di, Ying-Tong;  He, Hong-Ping;  Lu, Yang;  Yi, Ping;  Li, n Li;  Wu, Li;  Hao, Xiao-Jiang
Adobe PDF(116Kb)  |  收藏  |  浏览/下载:305/140  |  提交时间:2011/11/24
Calyciphylline-a  Glaucescens  Calycinum  Skeleton  Paxianum  Cascade