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Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:  Chen, Duo-zhi;  Yang, Bi-juan;  He, Xiao-li;  Fan, Shi-rui;  Cai, Jie-yun;  Jing, Chen-xu;  Zhang, Heng;  Zhang, Yu;  Li, Lin;  Hao, Xiao-jiang
浏览  |  Adobe PDF(3047Kb)  |  收藏  |  浏览/下载:312/37  |  提交时间:2019/03/18
Wnt/beta-catenin signalling pathway agonist  Phenanthridine derivatives  Structural optimization  Structure-activity relationships (SARs)  
C. elegans-based screen identifies lysosome-damaging alkaloids that induce STAT3-dependent lysosomal cell death 期刊论文
PROTEIN & CELL, 2018, 卷号: 9, 期号: 12, 页码: 1013-1026
作者:  Li, Yang;  Zhang, Yu;  Gan, Qiwen;  Xu, Meng;  Ding, Xiao;  Tang, Guihua;  Liang, Jingjing;  Liu, Kai;  Liu, Xuezhao;  Wang, Xin;  Guo, Lingli;  Gao, Zhiyang;  Hao, Xiaojiang;  Yang, Chonglin
收藏  |  浏览/下载:102/0  |  提交时间:2019/03/29
Autocatalytic synthesis of 3-ethyl-3-hydroxy-indole-2-ones and their neuroprotection and antitumor activities' evaluation 期刊论文
COMPTES RENDUS CHIMIE, 2018, 卷号: 21, 期号: 5, 页码: 471-474
作者:  Chen, Gang;  Lin, Jiao;  Zhang, Jie;  Wu, Ya;  Gu, Xuefan;  Hao, Xiaojiang;  Zhang, Yu
收藏  |  浏览/下载:122/0  |  提交时间:2019/03/29
Isatin  3-Ethyl-3-hydroxy-indole-2-one  Antitumor  Neuroprotection  
Two novel diterpenoid heterodimers, Bisebracteolasins A and B, from Euphorbia ebracteolata Hayata, and the cancer chemotherapeutic potential of Bisebracteolasin A 期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 页码: 1
作者:  Yuan, Wen-Juan;  Ding, Xiao;  Wang, Zhe;  Yang, Bi-Juan;  Li, Xiao-Nian;  Zhang, Yu;  Chen, Duo-Zhi;  Li, Shun-Lin;  Chen, Quan;  Di, Ying-Tong;  Aisa, Haji Akber;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(3375Kb)  |  收藏  |  浏览/下载:285/53  |  提交时间:2017/12/18
Synthesis, Neuro-protection and Anti-cancer Activities of Simple Isatin Mannich and Schiff Bases 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2016, 卷号: 13, 期号: 5, 页码: 395-400
作者:  Chen, Gang;  Ning, Yang;  Zhao, Wei;  Zhang, Yanqiu;  Zhang, Yu;  Hao, Xiaojiang;  Wang, Ye;  Mu, Shuzhen
浏览  |  Adobe PDF(1361Kb)  |  收藏  |  浏览/下载:229/70  |  提交时间:2016/08/22
Isatin  Mannich Base  Schiff Base  Synthesis  Neuro-protection  Anti-tumor  
New vobasinyl-ibogan type bisindole alkaloids from Tabernaemontana corymbosa 期刊论文
FITOTERAPIA, 2015, 卷号: 100, 页码: 150-155
作者:  Zhang, Yu;  Guo, Lingli;  Yang, Guangmei;  Guo, Feng;  Di, Yingtong;  Li, Shunlin;  Chen, Duozhi;  Hao, Xiaojiang
浏览  |  Adobe PDF(553Kb)  |  收藏  |  浏览/下载:330/95  |  提交时间:2015/06/17
Tabernaemontana Corymbosa  Bisindole Alkaloids  Tabercorines A-c  Cytotoxicity  
Synthesis, Cytoprotective and Anti-tumor Activities of Isatin Schiff Bases 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2015, 卷号: 12, 期号: 10, 页码: 802-805
作者:  Chen, Gang;  Meng, Mei;  Zhang, Yu;  Hao, Xiaojiang;  Wang, Ye;  Mu, Shuzhen
浏览  |  Adobe PDF(1108Kb)  |  收藏  |  浏览/下载:138/38  |  提交时间:2016/01/19
Isatin  Synthesis  Schiff Base  Structure  Cytoprotective  Anti-tumor  
Spiramine derivatives induce apoptosis of Bax(-/-)/Bak(-/-) cell and cancer cells 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 8, 页码: 1884-1888
作者:  Yan, Chen;  Huang, Li;  Liu, Hong-Chun;  Chen, Duo-Zhi;  Liu, Hai-Yang;  Li, Xiao-Hui;  Zhang, Yu;  Geng, Mei-Yu;  Chen, Quan;  Hao, Xiao-Jiang
Adobe PDF(1562Kb)  |  收藏  |  浏览/下载:297/45  |  提交时间:2014/06/23
Spiramine Derivative  Bax(-/-)/bak(-/-) Cells  Alpha  Apoptosis  Beta-unsaturated Ketone  Cytotoxicity  
A new Amaryllidaceae alkaloid from the bulbs of Lycoris radiata 期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2013, 卷号: 11, 期号: 4, 页码: 406-410
作者:  Huang Sheng-Dian;  Zhang Yu;  He Hong-Ping;  Li Shi-Fei;  Tang Gui-Hua;  Chen Duo-Zhi;  Cao Ming-Ming;  Di Ying-Tong;  Hao Xiao-Jiang
浏览  |  Adobe PDF(606Kb)  |  收藏  |  浏览/下载:297/55  |  提交时间:2013/10/16
Lycoris Radiata  Amaryllidaceae Alkaloids  Homolycorine-type  2 Alpha-methoxy-6-o-methyloduline  2 Alpha-methoxy-6-beta-ethyloduline  
Three novel beta-carboline alkaloids from Gelsemium elegans 期刊论文
FITOTERAPIA, 2012, 卷号: 83, 期号: 4, 页码: 704-708
作者:  Zhang, Zhen;  Zhang, Yu;  Wang, Yue-Hu;  Zhang, Qiang;  Yan, Xiao-Hui;  Di, Ying-Tong;  He, Hong-Ping;  Hao, Xiao-Jiang
Adobe PDF(341Kb)  |  收藏  |  浏览/下载:283/78  |  提交时间:2014/04/02
Loganiaceae  Gelsemium Elegans  Beta-carboline Alkaloids  Gelebolines A-c  Biogenetic Relationship