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The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1 期刊论文
出版物, 2111, 页码: 1-44
作者:  1M S Grace;  T Lieu;  B Darby;  F C Abogadie;  N Veldhuis N W Bunnett;  P McIntyre
Adobe PDF(1611Kb)  |  收藏  |  浏览/下载:109/1  |  提交时间:2017/07/24
Transient Receptor Potential Ion Channel  Trpv4  Protease Activated Receptor  Par2  Pain  Tyrosine Kinase  Bafetinib  
New Phenolic Dimers from Plant Paeonia suffruticosa and Their Cytotoxicity and NO Production Inhibition 期刊论文
Molecules, 2023
作者:  Qianqian Meng;  Shunyao Tong;  Yuqing Zhao;  Xingrong Peng;  Zhenghui Li;  Tao Feng;  Jikai Liu
浏览  |  Adobe PDF(1414Kb)  |  收藏  |  浏览/下载:429/60  |  提交时间:2023/10/07
New Monoterpenoid Indole Alkaloids from Tabernaemontana crassa Inhibit beta-Amyloid42 Production and Phospho-Tau (Thr217) 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 2, 页码: 1487
作者:  Li,Sheng;  Han,Ling-Ling;  Huang,Ke-Pu;  Ma,Ye-Han;  Guo,Ling-Li;  Guo,Yarong;  Ran,Xiaoqian;  Yao,Yong-Gang;  Hao,Xiao-Jiang;  Luo,Rongcan;  Zhang,Yu
浏览  |  Adobe PDF(5266Kb)  |  收藏  |  浏览/下载:7/4  |  提交时间:2024/05/09
Tabernaemontana crassa  monoterpenoid indole alkaloids  A beta 42  phospho-tau (Thr217)  Alzheimer's disease  ALZHEIMERS-DISEASE  BISINDOLE ALKALOIDS  CDK5  GEMFIBROZIL  PREVENTION  ALGORITHM  AUTOPHAGY  MODELS  PLANTS  MOUSE  
蕊木和奶子藤中生物碱类化学成分及其生物活性评价 学位论文
: 中国科学院大学, 2022
作者:  陈谌
Adobe PDF(17478Kb)  |  收藏  |  浏览/下载:37/0  |  提交时间:2024/05/14
夹竹桃科  Apocynaceae  蕊木  Kopsia arborea  奶子藤  Bousigonia mekongensis  单萜吲哚生物碱  Monoterterpene indole alkaloids  生物活性  Biological activity  
生物碱alstocholarine和daphenylline的不对称合成研究 学位论文
: 中国科学院大学, 2022
作者:  姚建能
Adobe PDF(7993Kb)  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/05/14
不对称合成, 虎皮楠生物碱, 单萜吲哚生物碱,天然产物  asymmetric synthesis, daphniphyllum alkaloids, monoterpenoid indole alkaloid, natural product  
Tabernaesine J, a Novel Vincamine-Type Indole Alkaloid with 6/5/6/6/6/5/5 Heptacyclic-Ring System Scaffold from Tabernaemontana pachysiphon 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2022, 卷号: 40, 期号: 4, 页码: 475-479
作者:  Yi,Wen-Fang;  Adelakun,Tiwalade A.;  Bai,Xue;  Zhang,Yu;  Hao,Xiao-Jiang
浏览  |  Adobe PDF(1252Kb)  |  收藏  |  浏览/下载:135/47  |  提交时间:2022/04/02
Natural products  Alkaloids  Structure elucidation  Tabernaemontana pachysiphon  Tabernaesine J  BISINDOLE ALKALOIDS  A-I  ALGORITHM  
云南百部和闷奶果的化学成分及生物活性研究 学位论文
, 2021
作者:  石宝宝
Adobe PDF(11462Kb)  |  收藏  |  浏览/下载:41/0  |  提交时间:2024/03/20
HRESIMS-guided isolation of aspidosperma-scandine type bisindole alkaloids from Melodinus cochinchinensis and their anti-inflammatory and cytotoxic activities 期刊论文
PHYTOCHEMISTRY, 2021, 卷号: 184, 页码: 112673
作者:  Li,Fang-Ru;  Liu,Lu;  Liu,Ya-Ping;  Wang,Jin-Tang;  Yang,Mei-Lian;  Khan,Afsar;  Qin,Xu-Jie;  Wang,Yu-Dan;  Cheng,Gui-Guang
收藏  |  浏览/下载:66/0  |  提交时间:2022/04/02
Melodinus cochinchinensis (Lour.) Merr. (Apocynaceae)  melokhanines  Bisindole alkaloids  Anti-inflammatory  Cytotoxicity  MONOTERPENOID INDOLE ALKALOIDS  CHEMISTRY  FRUITS  
Chemical constituents from Melodinus cochinchinensis (Lour.) Merr. and their chemotaxonomic significance 期刊论文
BIOCHEMICAL SYSTEMATICS AND ECOLOGY, 2021, 卷号: 95, 页码: 104245
作者:  Yang,Lin;  He,Jun-Jie;  Cui,Xiao-Yan;  Liu,Ya-Ping;  Wang,Bei
收藏  |  浏览/下载:55/0  |  提交时间:2022/04/02
Lignans  Indole alkaloids  Melodinus cochinchinensis (Lour.) Merr.  Chemotaxonomy  MONOTERPENOID INDOLE ALKALOIDS  LIGNANS  NEOLIGNANS  ANTIBACTERIAL  
The safety and tolerability of alkaloids from Alstonia scholaris leaves in healthy Chinese volunteers: a single-centre, randomized, double-blind, placebo-controlled phase I clinical trial 期刊论文
PHARMACEUTICAL BIOLOGY, 2021, 卷号: 59, 期号: 1, 页码: 484-493
作者:  Gou,Zhong-Ping;  Zhao,Yun-Li;  Zou,Lin-Ling;  Wang,Ying;  Shu,Shi-Qing;  Zhu,Xiao-Hong;  Zheng,Li;  Shen,Qi;  Luo,Zhu;  Miao,Jia;  Wang,Yong-Sheng;  Luo,Xiao-Dong;  Feng,Ping
收藏  |  浏览/下载:65/0  |  提交时间:2022/04/02
Clinical safety  healthy subject  dose-escalation study  MONOTERPENOID INDOLE ALKALOIDS  FLIGHT MASS-SPECTROMETRY  EXTRACT  IDENTIFICATION  CONSTITUENTS