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Structural and mechanistic basis of penicillin-bindingprotein inhibition by lactivicins 期刊论文
NATURE CHEMICAL BIOLOGY, 3111, 期号: 0, 页码: 1—5
作者:  Pauline Macheboeuf;  Delphine S Fischer;  Tom Brown Jr;  Astrid Zervosen;  Andre´Luxen;  Bernard Joris;  Andrea Dessen;  Christopher J Schofield
Adobe PDF(425Kb)  |  收藏  |  浏览/下载:95/1  |  提交时间:2017/07/21
An efficient and concise synthesis of a selective small molecule non-peptide inhibitor of cathepsin L: KGP94 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 105317
作者:  Munikishore,Rachakunta;  Wang,Liang-Liang;  Zhang,Shuqun;  Zhao,Qin-Shi;  Zuo,Zhili
浏览  |  Adobe PDF(523Kb)  |  收藏  |  浏览/下载:73/19  |  提交时间:2022/04/02
Cathepsin L  small-molecule inhibitor  gram-scale synthesis  KGP94  cancer  FUNCTIONALIZED BENZOPHENONE  BIOLOGICAL EVALUATION  TUMOR PROGRESSION  CELL INVASION  EXPRESSION  ANALOGS  SUPPRESSION  DERIVATIVES  ACID  
Lepithiohydimerins A-D: Four Pairs of Neuroprotective Thiohydantoin Dimers Bearing a Disulfide Bond from Maca (Lepidium meyenii Walp.) 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 10, 页码: 2738-2744
作者:  Peng,Xing-Rong;  Zhang,Ran-Ran;  Liu,Jun-Hong;  Li,Zhong-Rong;  Zhou,Lin;  Qiu,Ming-Hua
浏览  |  Adobe PDF(1698Kb)  |  收藏  |  浏览/下载:101/47  |  提交时间:2022/04/02
Lepidium meyenii Walp  Thiohydantoin dimers  Natural products  Structure elucidation  Biological activity  STRUCTURAL ELUCIDATION  DERIVATIVES  ANTIOXIDANT  HYDANTOIN  
Bioinspired Network Analysis Enabled Divergent Syntheses and Structure Revision of Pentacyclic Cytochalasans 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 卷号: 60, 期号: 29, 页码: 15963-15971
作者:  Wu,Hai;  Ding,Yiming;  Hu,Kun;  Long,Xianwen;  Qu,Chunlei;  Puno,Pema-Tenzin;  Deng,Jun
浏览  |  Adobe PDF(2675Kb)  |  收藏  |  浏览/下载:76/19  |  提交时间:2022/04/02
bioinspired network analysis  biomimetic synthesis  natural products  pentacyclic cytochalasans  structure elucidation  DIELS-ALDER REACTION  ISOINDOLONE NUCLEUS  RING-SYSTEM  MEROCYTOCHALASANS  REASSIGNMENT  DESATURATION  GENERATION  ALKALOIDS  CARBONATE  SKELETONS  
3-Hydroxy-4-methyldecanoic Acid-Containing Cyclotetradepsipeptides from an Endolichenic Beauveria sp. 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 4, 页码: 1244-1253
作者:  Zhou,Yuan-Fei;  Hu,Kun;  Wang,Fang;  Tang,Jian-Wei;  Zhang,Liang;  Sun,Han-Dong;  Cai,Xiang-Hai;  Puno,Pema-Tenzin
浏览  |  Adobe PDF(2249Kb)  |  收藏  |  浏览/下载:92/25  |  提交时间:2022/04/02
DOUBLE-BLIND  CYCLODEPSIPEPTIDES  CONFIGURATION  METABOLITES  SUROTOMYCIN  VANCOMYCIN  ADULTS  FUNGI  H-1  
(-)-Isoscopariusin A, a Naturally Occurring Immunosuppressive Meroditerpenoid: Structure Elucidation and Scalable Chemical Synthesis 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 卷号: 60, 期号: 23, 页码: 12859-12867
作者:  Yan,Bing-Chao;  Zhou,Min;  Li,Jian;  Li,Xiao-Nian;  He,Shi-Jun;  Zuo,Jian-Ping;  Sun,Han-Dong;  Li,Ang;  Puno,Pema-Tenzin
浏览  |  Adobe PDF(1930Kb)  |  收藏  |  浏览/下载:81/18  |  提交时间:2022/04/02
bioactivity  cyclobutane  natural products  scalable synthesis  structure elucidation  
Phyllanthacidoid U: a new N-glycosyl norbisabolane sesquiterpene from Phyllanthus acidus (L.) skeels 期刊论文
NATURAL PRODUCT RESEARCH, 2021, 卷号: 35, 期号: 21, 页码: 3540-3547
作者:  Xin,Ying;  Xu,Min;  Wang,Ya-Feng;  Zheng,Xiao-Hong;  Zhu,Hong-Tao;  Wang,Dong;  Yang,Chong-Ren;  Zhang,Ying-Jun
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Phyllanthus acidus  phyllanthacidoid U  norbisabolane sesquiterpenoid  amide  TUSSILAGO-FARFARA  FLOWER BUDS  EXTRACTS  PLANTS  
An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:82/18  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
广西莪术、团花、角茴香的化学成分及抗炎镇痛活性研究 学位论文
, 2020
作者:  袁海恋
Adobe PDF(5757Kb)  |  收藏  |  浏览/下载:40/1  |  提交时间:2023/11/02
暗绿蒿、玫黄黄肉牛肝菌和绿盖粉孢牛肝菌抗肝癌活性成分 学位论文
, 2020
作者:  苏丽花
Adobe PDF(11827Kb)  |  收藏  |  浏览/下载:38/0  |  提交时间:2023/11/02