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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:376/42  |  提交时间:2017/12/18
Bioactive sesquiterpenoids from the flowers of Inula japonica 期刊论文
PHYTOCHEMISTRY, 2016, 卷号: 129, 页码: 68-76
作者:  Wu, Xing-De;  Ding, Lin-Fen;  Tu, Wen-Chao;  Yang, Hui;  Su, Jia;  Peng, Li-Yan;  Li, Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1070Kb)  |  收藏  |  浏览/下载:257/62  |  提交时间:2016/11/04
Inula Japonica  Asteraceae  Sesquiterpenoids  Inujaponins A-i  Cytotoxicity  Nitric Oxide (No)  
Three new monoterpenoid indole alkaloids from Vinca major 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2016, 卷号: 18, 期号: 4, 页码: 328-333
作者:  Zhang, Zhi-Jun;  Du, Ru-Nan;  He, Juan;  Wu, Xing-De;  Li, Yan;  Li, Rong-Tao;  Zhao, Qin-Shi
浏览  |  Adobe PDF(822Kb)  |  收藏  |  浏览/下载:244/71  |  提交时间:2016/08/22
Apocynaceae  Vinca Major  Monoterpenoid Indole Alkaloid  Cytotoxicity  
Identification and validation of p50 as the cellular target of eriocalyxin B 期刊论文
ONCOTARGET, 2014, 卷号: 5, 期号: 22, 页码: 11354-11364
作者:  Kong, Ling-Mei;  Deng, Xu;  Zuo, Zhi-Li;  Sun, Han-Dong;  Zhao, Qin-Shi;  Li, Yan
浏览  |  Adobe PDF(3014Kb)  |  收藏  |  浏览/下载:280/71  |  提交时间:2015/06/17
Erib  Activity-based Probes  P50  Nf-kappa b Signaling  Apoptosis  
Vincamajorines A and B, monoterpenoid indole alkaloids with new carbon skeletons from Vinca major 期刊论文
TETRAHEDRON LETTERS, 2014, 卷号: 55, 期号: 47, 页码: 6490-6494
作者:  Zhang, Zhi-Jun;  Yang, Jing;  He, Juan;  Wu, Xing-De;  Shao, Li-Dong;  Li, Yan;  Huang, Sheng-Xiong;  Li, Rong-Tao;  Zhao, Qin-Shi;  Li,RT (reprint author),Kunming Univ Sci & Technol,Fac Life Sci & Technol,Chenggong Campus,Kunming 650050,Yunnan,Peoples R China.;  rongtaolikm@163.com;  qinshizhao@mail.kib.ac.cn
浏览  |  Adobe PDF(763Kb)  |  收藏  |  浏览/下载:301/72  |  提交时间:2015/01/20
Vinca Major  Monoterpenoid Indole Alkaloids  Quantum Chemical Calculations  
New alkaloids sinomacutines A-E, and cephalonine-2-O-beta-D-glucopyranoside from rhizomes of Sinomenium acutum 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 46, 页码: 8893-8899
作者:  Li, Yan-Hong;  Li, Hong-Mei;  Li, Yan;  He, Juan;  Deng, Xu;  Peng, Li-Yan;  Gao, Ling-Huan;  Zhao, Qin-Shi;  Li, Rong-Tao;  Wu, Xing-De;  Li,RT (reprint author),Kunming Univ Sci & Technol,Fac Life Sci & Technol,Kunming 650500,Yunnan,Peoples R China.;  rongtaolikm@gmail.com;  wuxingde@mail.kib.ac.cn
浏览  |  Adobe PDF(673Kb)  |  收藏  |  浏览/下载:262/71  |  提交时间:2015/01/20
Sinomenium Acutum  Bistetrahydroisoquinoline Alkaloid  Acid Hydrolysis  Cytotoxicity  Anti-inflammatory Activity  
Identification of two novel inhibitors of mTOR signaling pathway based on high content screening 期刊论文
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2013, 卷号: 72, 期号: 4, 页码: 799-808
作者:  Yan, Juming;  Zhou, Hongyu;  Kong, Lingmei;  Zhang, Jing;  Zhao, Qinshi;  Li, Yan
Adobe PDF(1971Kb)  |  收藏  |  浏览/下载:676/103  |  提交时间:2013/11/12
Mtor Signaling  Inhibitor  High Content Screening  Cancer  Apoptosis  
Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-kappa B Activation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4749-4757
作者:  Zhao, Yu;  Su, Jia;  Goto, Masuo;  Morris-Natschke, Susan L.;  Li, Yan;  Zhao, Qin-Shi;  Yao, Zhu-Jun;  Lee, Kuo-Hsiung
浏览  |  Adobe PDF(531Kb)  |  收藏  |  浏览/下载:311/65  |  提交时间:2013/10/16
Natural-products  Biological-activity  Cancer-therapy  Paclitaxel  Taxol  Resistance  Drugs  Chemotherapy  Parthenolide  Brevifoliol  
Norditerpenoids from Salvia castanea Diels f. pubescens 期刊论文
FITOTERAPIA, 2012, 卷号: 83, 期号: 6, 页码: 1072-1075
作者:  Pan, Zheng-Hong;  Li, Yan;  Wu, Xing-De;  He, Juan;  Chen, Xuan-Qin;  Xu, Gang;  Peng, Li-Yan;  Zhao, Qin-Shi
Adobe PDF(278Kb)  |  收藏  |  浏览/下载:580/175  |  提交时间:2012/11/30
Salvia Castanea Diels F. Pubescens  Norditerpenoid  Castanol A-c  Cytotoxic Activity  
Three New Sucrose Fatty Acid Esters from Equisetum hiemale L. 期刊论文
HELVETICA CHIMICA ACTA, 2012, 卷号: 95, 期号: 7, 页码: 1158-1163
作者:  Cheng, Jin-Tang;  He, Juan;  Li, Xing-Yao;  Wu, Xing-De;  Shao, Li-Dong;  Dong, Liao-Bin;  Deng, Xu;  Gao, Xiu;  Peng, Li-Yan;  Cheng, Xiao;  Li, Yan;  Zhao, Qin-Shi
Adobe PDF(187Kb)  |  收藏  |  浏览/下载:323/97  |  提交时间:2012/09/03
Equisetum Hiemale  Fatty Acid Esters  Sucrose  Glycosides