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虚拟筛选与蛋白降解在TRPC5调节剂发现设计中的实践 学位论文
, 2021
作者:  刘斌
Microsoft Word(8818Kb)  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/03/20
Discovery of novel modulators targeting human TRPC5: Docking-based virtual screening, molecular dynamics simulation and binding af fi nity predication 期刊论文
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2021, 卷号: 102, 页码: 107795
作者:  Liu,Bin;  Zhang,Wei;  Guo,Sheng;  Zuo,Zhili
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hTRPC5  Homology modeling  Molecular docking  Molecular dynamics simulation  Virtual screening  INHIBITOR  CHANNELS  GROMACS  POTENT  AMBER  IDENTIFICATION  CONSTRAINTS  INTEGRATION  AMYGDALA  
Identification of Novel TRPC5 Inhibitors by Pharmacophore-Based and Structure-Based Approaches 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2020
作者:  Li, Shuxiang;  Zhang, Shuqun;  Chen, Dingyuan;  Jiang, Xuan;  Liu, Bin;  Zhang, Hongbin;  Rachakunta, Munikishore;  Zuo, Zhili
浏览  |  Adobe PDF(4261Kb)  |  收藏  |  浏览/下载:171/46  |  提交时间:2021/01/05
M084抗衰老机制及WWP-1调控脂代谢与衰老机制的研究 学位论文
: 中国科学院大学, 2017
作者:  丁爱军
Adobe PDF(4584Kb)  |  收藏  |  浏览/下载:121/1  |  提交时间:2019/06/14
Benzimidazole derivative M084 extends the lifespan of Caenorhabditis elegans in a DAF-16/FOXO-dependent way 期刊论文
MOLECULAR AND CELLULAR BIOCHEMISTRY, 2017, 卷号: 426, 期号: 1-2, 页码: 101-109
作者:  Ding, Ai-Jun;  Wu, Gui-Sheng;  Tang, Bin;  Hong, Xuechuan;  Zhu, Michael X.;  Luo, Huai-Rong
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Aging  Benzimidazole Derivative M084  Caenorhabditis Elegans  Lifespan  
Current Perspective in the Discovery of Anti-aging Agents from Natural Products. 期刊论文
Natural products and bioprospecting, 2017, 卷号: 7, 期号: 5, 页码: 335-404
作者:  Ding, Ai-Jun;  Zheng, Shan-Qing;  Huang, Xiao-Bing;  Xing, Ti-Kun;  Wu, Gui-Sheng;  Sun, Hua-Ying;  Qi, Shu-Hua;  Luo, Huai-Rong
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2017年中科院昆明植物研究所年报 其他
2017-01-01
作者:  昆明植物所
Adobe PDF(19558Kb)  |  收藏  |  浏览/下载:261/13  |  提交时间:2018/08/01
小鼠海马下托腹侧向全脑的顺向投射研究 学位论文
: 中国科学院大学, 2016
作者:  唐贺
Adobe PDF(3991Kb)  |  收藏  |  浏览/下载:90/1  |  提交时间:2019/06/14
Acute Treatment with a Novel TRPC4/C5 Channel Inhibitor Produces Antidepressant and Anxiolytic-Like Effects in Mice 期刊论文
PLOS ONE, 2015, 卷号: 10, 期号: 8
作者:  Yang, Li-Ping;  Jiang, Fang-Jie;  Wu, Gui-Sheng;  Deng, Ke;  Wen, Meng;  Zhou, Xiaoju;  Hong, Xuechuan;  Zhu, Michael X.;  Luo, Huai-Rong
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Identification and optimization of 2-aminobenzimidazole derivatives as novel inhibitors of TRPC4 and TRPC5 channels 期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2015, 卷号: 172, 期号: 14, 页码: 3495-3509
作者:  Zhu, Yingmin;  Lu, Yungang;  Qu, Chunrong;  Miller, Melissa;  Tian, Jinbin;  Thakur, Dhananjay P.;  Zhu, Jinmei;  Deng, Zixin;  Hu, Xianming;  Wu, Meng;  McManus, Owen B.;  Li, Min;  Hong, Xuechuan;  Zhu, Michael X.;  Luo, Huai-Rong
浏览  |  Adobe PDF(2298Kb)  |  收藏  |  浏览/下载:230/54  |  提交时间:2015/12/15