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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:65/15  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Caesalpanins A-C, Three Dimeric Cassane Diterpenoids from the Seeds of Caesalpinia sappan L. 期刊论文
CHEMISTRY & BIODIVERSITY, 2020
作者:  Wang, De-Sheng;  Nie, Wei;  Jiang, Ting-Ting;  Ding, Lin-Fen;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1960Kb)  |  收藏  |  浏览/下载:147/46  |  提交时间:2021/01/05
Two New Anti-Proliferative C-18-Norditerpenes from the Roots of Podocarpus macrophyllus 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 4, 页码: e1800043
作者:  Qi, Yan-Yan;  Su, Jia;  Zhang, Zhi-Jun;  Li, Lai-Wei;  Fan, Min;  Zhu, Yu;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1080Kb)  |  收藏  |  浏览/下载:474/107  |  提交时间:2018/07/02
Podocarpus Macrophyllus  Norditerpenoid  Anti-proliferative Activity  Activity-guided Fractionation  Structure Revision  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:366/41  |  提交时间:2017/12/18
Bioactive sesquiterpenoids from the flowers of Inula japonica 期刊论文
PHYTOCHEMISTRY, 2016, 卷号: 129, 页码: 68-76
作者:  Wu, Xing-De;  Ding, Lin-Fen;  Tu, Wen-Chao;  Yang, Hui;  Su, Jia;  Peng, Li-Yan;  Li, Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1070Kb)  |  收藏  |  浏览/下载:248/61  |  提交时间:2016/11/04
Inula Japonica  Asteraceae  Sesquiterpenoids  Inujaponins A-i  Cytotoxicity  Nitric Oxide (No)  
Six new cassane diterpenoids from the seeds of Caesalpinia sappan 期刊论文
PHYTOCHEMISTRY LETTERS, 2016, 卷号: 16, 页码: 207-212
作者:  Deng, Zhen-Tao;  Su, Jia;  Ding, Lin-Fen;  Tu, Wen-Chao;  Yang, Hui;  Peng, Li-Yan;  Zhao, Qin-Shi;  Song, Liu-Dong;  Wu, Xing-De
浏览  |  Adobe PDF(854Kb)  |  收藏  |  浏览/下载:196/73  |  提交时间:2016/08/22
Caesalpinia Sappan l  Leguminosae  Cassane Diterpenoids  Cytotoxicity  
Identification and validation of p50 as the cellular target of eriocalyxin B 期刊论文
ONCOTARGET, 2014, 卷号: 5, 期号: 22, 页码: 11354-11364
作者:  Kong, Ling-Mei;  Deng, Xu;  Zuo, Zhi-Li;  Sun, Han-Dong;  Zhao, Qin-Shi;  Li, Yan
浏览  |  Adobe PDF(3014Kb)  |  收藏  |  浏览/下载:266/68  |  提交时间:2015/06/17
Erib  Activity-based Probes  P50  Nf-kappa b Signaling  Apoptosis  
Compounds from Dryopteris Fragrans (L.) Schott with Cytotoxic Activity 期刊论文
MOLECULES, 2014, 卷号: 19, 期号: 3, 页码: 3345-3355
作者:  Zhao, Dan-Dan;  Zhao, Qin-Shi;  Liu, Li;  Chen, Zhong-Qin;  Zeng, Wei-Min;  Lei, Hong;  Zhang, Yan-Long
Adobe PDF(408Kb)  |  收藏  |  浏览/下载:259/54  |  提交时间:2014/06/23
Dryopteris Fragrans (L.) Schott  Compounds  Mtt  Cytotoxic Activity  
Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-kappa B Activation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4749-4757
作者:  Zhao, Yu;  Su, Jia;  Goto, Masuo;  Morris-Natschke, Susan L.;  Li, Yan;  Zhao, Qin-Shi;  Yao, Zhu-Jun;  Lee, Kuo-Hsiung
浏览  |  Adobe PDF(531Kb)  |  收藏  |  浏览/下载:298/62  |  提交时间:2013/10/16
Natural-products  Biological-activity  Cancer-therapy  Paclitaxel  Taxol  Resistance  Drugs  Chemotherapy  Parthenolide  Brevifoliol  
Melissoidesin G, a diterpenoid purified from Isodon melissoides, induces leukemic-cell apoptosis through induction of redox imbalance and exhibits synergy with other anticancer agents 期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2007, 卷号: 121, 期号: 9, 页码: 2084-2094
作者:  Yu, Zu-Yin;  Liang, Yu-Guang;  Xiao, He;  Shan, Ya-Jun;  Dong, Bo;  Huang, Rui;  Fu, Ya-Li;  Zhao, Zhen-Hu;  Liu, Ze-Yuan;  Zhao, Qin-Shi;  Wang, Sheng-Qi;  Chen, Jia-Pei;  Mao, Bing-Zhi;  Cong, Yu-Wen
Adobe PDF(894Kb)  |  收藏  |  浏览/下载:288/78  |  提交时间:2011/11/24
Melissoidesin g  Leukemia  Apoptosis  Redox  Arsenic Trioxide