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Addition of aldehydes with allyltrichlorosilane catalyzed by chiral bis-N-O secondary amides 期刊论文
TETRAHEDRON, 2013, 卷号: 69, 期号: 48, 页码: 10431-10437
作者:  Deng, Yu;  Pan, Wei;  Pei, Yu-Ning;  Li, Jin-Liang;  Bai, Bing;  Zhu, Hua-Jie
Adobe PDF(869Kb)  |  收藏  |  浏览/下载:683/130  |  提交时间:2014/01/21
Bis-n-o Amides  Allylation  L-tryptophan  Axial Ligand  
Total synthesis of (+/-)-brazilin and formal synthesis of (+/-)-brazilein, (+/-)-brazilide A using m-CPBA 期刊论文
TETRAHEDRON LETTERS, 2013, 卷号: 54, 期号: 45, 页码: 6029-6031
作者:  Li, Liang-Qun;  Li, Ming-Ming;  Wang, Kou;  Qin, Hong-Bo
Adobe PDF(608Kb)  |  收藏  |  浏览/下载:617/132  |  提交时间:2013/11/12
Total Synthesis  Brazilin  Brazilein  Brazilide a  M-cpba  
Scopariusic Acid, a New Meroditerpenoid with a Unique Cyclobutane Ring Isolated from Isodon scoparius 期刊论文
ORGANIC LETTERS, 2013, 卷号: 15, 期号: 17, 页码: 4446-4449
作者:  Zhou, Min;  Zhang, Hai-Bo;  Wang, Wei-Guang;  Gong, Ning-Bo;  Zhan, Rui;  Li, Xiao-Nian;  Du, Xue;  Li, Li-Mei;  Li, Yan;  Lu, Yang;  Pu, Jian-Xin;  Sun, Han-Dong
Adobe PDF(792Kb)  |  收藏  |  浏览/下载:429/111  |  提交时间:2014/01/21
2+2 Cycloadditions  Biyouyanagin-a  Biological Evaluation  Incarvillea-sinensis  Revised Structure  Skeleton  Littoralisone  Alkaloids  Diterpene  
Three new compounds from the cultures of basidiomycete Boreostereum vibrans 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2013, 卷号: 15, 期号: 9, 页码: 950-955
作者:  Wang, Gang-Qiang;  Wei, Kun;  Li, Zheng-Hui;  Feng, Tao;  Ding, Jian-Hai;  Wang, Qiu-An;  Liu, Ji-Kai
Adobe PDF(118Kb)  |  收藏  |  浏览/下载:227/61  |  提交时间:2014/01/13
Boreostereum Vibrans  Basidiomycete  Vibralactone Derivatives  
Synthesis and antitumor activities of novel dibenzo[b,d]furan-imidazole hybrid compounds 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 66, 页码: 423-437
作者:  Liu, Lan-Xiang;  Wang, Xue-Quan;  Yan, Ju-Ming;  Li, Yan;  Sun, Cheng-Jun;  Chen, Wen;  Zhou, Bei;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Adobe PDF(3339Kb)  |  收藏  |  浏览/下载:335/141  |  提交时间:2013/10/16
Hybrid Compound  Imidazole  Dibenzo[b  Antitumor Activities  d]Furan  Structure-activity Relationships  
Synthesis and cytotoxic activities of novel hybrid 2-phenyl-3-alkylbenzofuran and imidazole/triazole compounds 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 卷号: 23, 期号: 15, 页码: 4297-4302
作者:  Chen, Wen;  Deng, Xiao-Yan;  Li, Yan;  Yang, Li-Juan;  Wan, Wei-Chao;  Wang, Xue-Quan;  Zhang, Hong-Bin;  Yang, Xiao-Dong
Adobe PDF(820Kb)  |  收藏  |  浏览/下载:245/45  |  提交时间:2013/10/16
Hybrid Compound  Benzofuran  Imidazole  Triazole  Structure-activity Relationships  
Synthesis, biological evaluation and molecular modeling of substituted 2-aminobenzimidazoles as novel inhibitors of acetylcholinesterase and butyrylcholinesterase 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 14, 页码: 4218-4224
作者:  Zhu, Jinmei;  Wu, Chun-Feng;  Li, Xiaobing;  Wu, Gui-Sheng;  Xie, Shan;  Hu, Qian-Nan;  Deng, Zixin;  Zhu, Michael X.;  Luo, Huai-Rong;  Hong, Xuechuan
Adobe PDF(1174Kb)  |  收藏  |  浏览/下载:531/89  |  提交时间:2013/10/16
Alzheimer's Disease  Acetylcholinesterase  Butyrylcholinesterase  Molecular Modeling  2-aminobenzimidazole  
Discovery and structure-activity relationships of ent-Kaurene diterpenoids as potent and selective 11 beta-HSD1 inhibitors: Potential impact in diabetes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 403-414
作者:  Deng, Xu;  Shen, Yu;  Yang, Jing;  He, Juan;  Zhao, Yu;  Peng, Li-Yan;  Leng, Ying;  Zhao, Qin-Shi
Adobe PDF(1215Kb)  |  收藏  |  浏览/下载:403/151  |  提交时间:2013/10/16
Ent-kaurene Diterpenoids  Structure-activity Relationship Studies  Selective 11 Beta-hsd1 Inhibitors  Urea Derivatives  Diabetes  
Dual-Functional abeo-Taxane Derivatives Destabilizing Microtubule Equilibrium and Inhibiting NF-kappa B Activation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4749-4757
作者:  Zhao, Yu;  Su, Jia;  Goto, Masuo;  Morris-Natschke, Susan L.;  Li, Yan;  Zhao, Qin-Shi;  Yao, Zhu-Jun;  Lee, Kuo-Hsiung
Adobe PDF(531Kb)  |  收藏  |  浏览/下载:308/64  |  提交时间:2013/10/16
Natural-products  Biological-activity  Cancer-therapy  Paclitaxel  Taxol  Resistance  Drugs  Chemotherapy  Parthenolide  Brevifoliol  
Peltate Glandular Trichomes of Colquhounia coccinea var. mollis Harbor a New Class of Defensive Sesterterpenoids 期刊论文
ORGANIC LETTERS, 2013, 卷号: 15, 期号: 7, 页码: 1694-1697
作者:  Li, Chun-Huan;  Jing, Shu-Xi;  Luo, Shi-Hong;  Shi, Wei;  Hua, Juan;  Liu, Yan;  Li, Xiao-Nian;  Schneider, Bernd;  Gershenzon, Jonathan;  Li, Sheng-Hong
Adobe PDF(1541Kb)  |  收藏  |  浏览/下载:901/112  |  提交时间:2013/07/24
Leucosceptrum-canum