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Design and synthesis of new 2-arylnaphthyridin-4-ones as potent antitumor agents targeting tumorigenic cell lines 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 90, 页码: 775-787
作者:  Liu, Chin-Yu;  Cheng, Yung-Yi;  Chang, Ling-Chu;  Huang, Li-Jiau;  Chou, Li-Chen;  Huang, Chi-Hung;  Tsai, Meng-Tung;  Liao, Chih-Chang;  Hsu, Mei-Hua;  Lin, Hui-Yi;  Wu, Tian-Shung;  Wen, Yen-Fang;  Zhao, Yu;  Kuo, Sheng-Chu;  Lee, Kuo-Hsiung;  Kuo,SC (reprint author),China Med Univ,Grad Inst Pharmaceut Chem,91 Hsueh Shih Rd,Taichung 40402,Taiwan.;  sckuo@mail.cmu.edu.tw;  khlee@unc.edu
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2-arylnaphthyridin-4-ones  Antitumor Agents  Phosphate Prodrug  
Indole alkaloids from cultivated Vinca major 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 45, 页码: 8723-8729
作者:  Cheng, Gui-Guang;  Zhao, Yun-Li;  Zhang, Yu;  Lunga, Paul-Keilah;  Hu, Dong-Bao;  Li, Yan;  Gu, Ji;  Song, Chang-Wei;  Sun, Wei-Bang;  Liu, Ya-Ping;  Luo, Xiao-Dong;  Liu,YP (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  liuyaping@mail.kib.ac.cn;  xdluo@mail.kib.ac.cn
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Indole Alkaloids  Cytotoxicity  Absolute Configuration  Vinca Major  
Rubischumanins A-C, new cytotoxic cyclopeptides from Rubia schumanniana 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 42, 页码: 7627-7631
作者:  Huang, Mao-Bo;  Zhao, Si-Meng;  Zeng, Guang-Zhi;  Kuang, Bin;  Chen, Xiao-Qiang;  Tan, Ning-Hua;  Zeng,GZ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  gzh_zeng@mail.kib.ac.cn;  nhtan@mail.kib.ac.cn
Adobe PDF(498Kb)  |  收藏  |  浏览/下载:401/63  |  提交时间:2014/11/25
Rubia Schumanniana  Rubischumanins A-c  Cyclopeptides  Cytotoxicity  
Characterization and biological evaluation of six new dimeric lignans with an unusual alpha,beta-unsaturated ketone motif from Zanthoxylum simulans 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 19, 页码: 4667-4671
作者:  Wang, Jun-Feng;  Deng, Yi-Hui;  Yang, Sheng-Hui;  Liu, Yan-Qun;  Wang, Yue-Hu;  Pan, Wei-Wei;  Zhou, Xiao-Jiang;  Zhou,XJ (reprint author),Hunan Univ Chinese Med,Coll Pharm,Changsha 410208,Hunan,Peoples R China.;  gale9888@163.com
Adobe PDF(1369Kb)  |  收藏  |  浏览/下载:223/41  |  提交时间:2014/11/25
Zanthoxylum Simulans  Dimeric Lignans  Synovial Cells  Splenocytes  
Anti-Hepatitis B Virus Norbisabolane Sesquiterpenoids from Phyllanthus acidus and the Establishment of Their Absolute Configurations Using Theoretical Calculations 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2014, 卷号: 79, 期号: 12, 页码: 5432-5447
作者:  Lv, Jun-Jiang;  Yu, Shan;  Wang, Ya-Feng;  Wang, Dong;  Zhu, Hong-Tao;  Cheng, Rong-Rong;  Yang, Chong-Ren;  Xu, Min;  Zhang, Ying-Jun;  Xu,M (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  minxu@mail.kib.ac.cn;  zhangyj@mail.kib.ac.cn
Adobe PDF(655Kb)  |  收藏  |  浏览/下载:322/93  |  提交时间:2014/07/28
Antineoplastic Agents  Acuminatus Vahl  Glycosides  Emblica  Roots  Secretion  Norsesquiterpenoids  Pyrimidine  Inhibitors  
Isolation and Complete Structural Assignment of Lycopodium Alkaloid Cernupalhine A: Theoretical Prediction and Total Synthesis Validation 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 10, 页码: 2700-2703
作者:  Dong, Liao-Bin;  Wu, Ya-Nan;  Jiang, Shi-Zhi;  Wu, Xing-De;  He, Juan;  Yang, Yu-Rong;  Zhao, Qin-Shi
Adobe PDF(319Kb)  |  收藏  |  浏览/下载:346/55  |  提交时间:2014/06/23
Fawcettimine-related Alkaloids  Alpha  Unified Total Syntheses  Beta-unsaturated Carbonyl-compounds  Palhinhaea-cernua  Unprecedented Skeleton  Helquist Annulation  A-c  Japonicum  (-)-8-deoxyserratinine  (+)-lycoflexine  
Spiramine derivatives induce apoptosis of Bax(-/-)/Bak(-/-) cell and cancer cells 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 8, 页码: 1884-1888
作者:  Yan, Chen;  Huang, Li;  Liu, Hong-Chun;  Chen, Duo-Zhi;  Liu, Hai-Yang;  Li, Xiao-Hui;  Zhang, Yu;  Geng, Mei-Yu;  Chen, Quan;  Hao, Xiao-Jiang
Adobe PDF(1562Kb)  |  收藏  |  浏览/下载:299/45  |  提交时间:2014/06/23
Spiramine Derivative  Bax(-/-)/bak(-/-) Cells  Alpha  Apoptosis  Beta-unsaturated Ketone  Cytotoxicity  
Structural Characterization and Antioxidative Activity of Lancifonins: Unique Nortriterpenoids from Schisandra lancifolia 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 5, 页码: 1370-1373
作者:  Shi, Yi-Ming;  Yang, Jie;  Xu, Li;  Li, Xiao-Nian;  Shang, Shan-Zhai;  Cao, Peng;  Xiao, Wei-Lie;  Sun, Han-Dong
Adobe PDF(340Kb)  |  收藏  |  浏览/下载:277/81  |  提交时间:2014/05/16
Lancifodilactone g  Micrandilactone  Cyclization  Chinensis  
Anti-hepatitis B virus activities and absolute configurations of sesquiterpenoid glycosides from Phyllanthus emblica 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2014, 卷号: 12, 期号: 43, 页码: 8764-8774
作者:  Lv, Jun-Jiang;  Wang, Ya-Feng;  Zhang, Jing-Min;  Yu, Shan;  Wang, Dong;  Zhu, Hong-Tao;  Cheng, Rong-Rong;  Yang, Chong-Ren;  Xu, Min;  Zhang, Ying-Jun;  Xu,M (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  minxu@mail.kib.ac.cn;  zhangyj@mail.kib.ac.cn
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Constituents  Model  Aspongopus Chinensis  Insects  Norepinephrine Derivatives  Sesquiterpenoids  Lactam  Biological Evaluation  
Sesquiterpenoids with New Carbon Skeletons from the Resin of Toxicodendron vernicifluum as New Types of Extracellular Matrix Inhibitors 期刊论文
ORGANIC LETTERS, 2013, 卷号: 15, 期号: 14, 页码: 3602-3605
作者:  He, Jiang-Bo;  Luo, Jie;  Zhang, Li;  Yan, Yong-Min;  Cheng, Yong-Xian
浏览  |  Adobe PDF(274Kb)  |  收藏  |  浏览/下载:410/83  |  提交时间:2013/10/16
Diabetic-nephropathy  Metabolism