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Salvifarinin A, a neo-clerodane diterpenoid with a 6/5/7 tricyclic skeleton from Salvia farinacea 期刊论文
TETRAHEDRON LETTERS, 2018, 卷号: 59, 期号: 32, 页码: 3065-3068
作者:  Fan, Min;  Chen, Xue-Jiao;  Wu, Xing-De;  Shao, Li-Dong;  Ji, Xu;  Zhao, Qin-Shi
收藏  |  浏览/下载:362/0  |  提交时间:2018/09/17
Neo-clerodane Diterpenoids  Salvia Farinacea  Lipid-lowering Activity  
A practical total synthesis of (+/-)-cermizine D and a formal synthesis of (+/-)-cermizine C 期刊论文
JOURNAL OF CHEMICAL RESEARCH, 2018, 期号: 5, 页码: 274-279
作者:  Shi, Xin;  Bao, Ying;  Deng, Zhen-Tao;  Zhu, Yu;  Shao, Li-Dong;  Zhang, Hong-Bin;  Zhao, Qin-Shi
收藏  |  浏览/下载:240/0  |  提交时间:2018/07/30
Cermizine c  Cermizine d  Total Synthesis  Michael Addition  Reductive Amination  
Vibsane-Type Diterpenoids from Viburnum odoratissimum and Their Cytotoxic and HSP90 Inhibitory Activities 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 5, 页码: 1800049
作者:  Zhu, Qin-Feng;  Qi, Yan-Yan;  Zhang, Zhi-Jun;  Fan, Min;  Bi, Ran;  Su, Jia;  Wu, Xing-De;  Shao, Li-Dong;  Zhao, Qin-Shi
收藏  |  浏览/下载:346/0  |  提交时间:2018/07/16
Vibsane-type Diterpenoids  Viburnum Odoratissimum  Cytotoxicity  Hsp90 Inhibitor  
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:385/42  |  提交时间:2017/12/18
Total Synthesis of (+/-)-Cermizine B 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 82, 期号: 20, 页码: 11110-11116
作者:  Shi, Xin;  Deng, Zhen-Tao;  Zhu, Yu;  Bao, Ying;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:193/47  |  提交时间:2017/12/18
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:316/73  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
A biomimetic semisynthesis enables structural elucidation of selaginellin U: a tautomeric cyclic alkynylphenol from Selaginella tamariscina 期刊论文
ROYAL SOCIETY OPEN SCIENCE, 2017, 卷号: 4, 期号: 7, 页码: 170352
作者:  Zhu, Qin-Feng;  Bao, Ying;  Zhang, Zhi-Jun;  Su, Jia;  Shao, Li-Dong;  Zhao, Qin-Shi
浏览  |  Adobe PDF(698Kb)  |  收藏  |  浏览/下载:169/23  |  提交时间:2017/10/23
Biomimetic Semisynthesis  Structural Elucidation  Selaginellins  Alkynylphenol  Selaginella Tamariscina  
Tilifodiolide及其衍生物在制备治疗或预防II型糖尿病药物中的应用 专利
申请日期: 2017-03-16, 公开日期: 2017-07-18
发明人:  赵勤实;  樊献俄;  张人伟;  杨春雷;  苏佳;  彭丽艳;  邵立东;  吴兴德
收藏  |  浏览/下载:160/0  |  提交时间:2018/05/10
黄藤内酯及其衍生物在制备治疗或预防II型糖尿病药物中的应用 专利
申请日期: 2017-03-16, 公开日期: 2017-11-24
发明人:  赵勤实;  樊献俄;  张人伟;  杨春雷;  苏佳;  彭丽艳;  吴兴德;  邵立东
收藏  |  浏览/下载:157/0  |  提交时间:2018/05/10
呋喃卡山烷二萜衍生物及其药物组合物和其在制药中的应用 专利
申请日期: 2017-01-13, 公开日期: 2017-06-09
发明人:  赵勤实;  冷颖;  吴兴德;  黄素玲;  苏佳;  邵立东;  彭丽艳
收藏  |  浏览/下载:155/0  |  提交时间:2018/05/10