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Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
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Potential role of CYP1B1 in the development and treatment of metabolic diseases 期刊论文
PHARMACOLOGY & THERAPEUTICS, 2017, 卷号: 178, 页码: 18-30
作者:  Li, Fei;  Zhu, Weifeng;  Gonzalez, Frank J.
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Cyp1b1  Metabolic Diseases  Metabolic Pathways  Metabolomics  
Anti-HIV Activities and Mechanism of 12-O-Tricosanoylphorbol-20-acetate, a Novel Phorbol Ester from Ostodes katharinae 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 9, 页码: 1498
作者:  Chen, Huan;  Zhang, Rong;  Luo, Rong-Hua;  Yang, Liu-Meng;  Wang, Rui-Rui;  Hao, Xiao-Jiang;  Zheng, Yong-Tang
浏览  |  Adobe PDF(1939Kb)  |  收藏  |  浏览/下载:192/38  |  提交时间:2017/10/23
Antiviral Agent  12-o-tricosanoylphorbol-20-acetate  Hiv  Vif  Apobec3g  Phorbol Ester  
Diterpenoids from Isodon species: an update 期刊论文
NATURAL PRODUCT REPORTS, 2017, 卷号: 34, 期号: 9, 页码: 1090-1140
作者:  Liu, Miao;  Wang, Wei-Guang;  Sun, Han-Dong;  Pu, Jian-Xin
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Ent-kaurane Diterpenoids  Japonica Var. Glaucocalyx  Nf-kappa-b  Hepatocellular-carcinoma Cells  C-h Functionalization  Dna-binding Activity  Serra Maxim. Hara  Maoecrystal-v  Abietane Diterpenoids  Chemical-constituents  
(+/-)-Rubioncolin D, a pair of enantiomeric naphthohydroquinone dimers from Rubia oncotricha 期刊论文
TETRAHEDRON LETTERS, 2017, 卷号: 58, 期号: 31, 页码: 3041-3043
作者:  Zhao, Si-Meng;  Wang, Zhe;  Chen, Xiao-Qiang;  Huang, Mao-Bo;  Tan, Ning-Hua
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Rubio Oncotricha  Naphthohydroquinone Dimers  Rubioncolin d  
ZC4H2 stabilizes Smads to enhance BMP signalling, which is involved in neural development in Xenopus 期刊论文
OPEN BIOLOGY, 2017, 卷号: 7, 期号: 8, 页码: 170122
作者:  Ma, Pengcheng;  Ren, Biyu;  Yang, Xiangcai;  Sun, Bin;  Liu, Xiaoliang;  Kong, Qinghua;  Li, Chaocui;  Mao, Bingyu
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Zc4h2  Smad  Smurf  Bone Morphogenesis Protein Signalling  Neural Development  
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
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11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
Foragers of sympatric Asian honey bee species intercept competitor signals by avoiding benzyl acetate from Apis cerana alarm pheromone 期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7, 页码: 6721
作者:  Wen, Ping;  Cheng, Yanan;  Qu, Yufeng;  Zhang, Hongxia;  Li, Jianjun;  Bell, Heather;  Tan, Ken;  Nieh, James
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Sting Apparatus  Evolution  Information  Dorsata  Communication  Cooperation  Components  Altruism  Tadpoles  Behavior  
Click Glycosylation for the Synthesis of 1,2,3-Triazole-Linked Picropodophyllotoxin Glycoconjugates and Their Anticancer Activity 期刊论文
CHEMISTRYSELECT, 2017, 卷号: 2, 期号: 18, 页码: 5038-5044
作者:  Zi, Cheng-Ting;  Yang, Liu;  Gao, Wei;  Li, Yan;  Zhou, Jun;  Ding, Zhong-Tao;  Hu, Jiang-Miao;  Jiang, Zi-Hua
浏览  |  Adobe PDF(3775Kb)  |  收藏  |  浏览/下载:226/45  |  提交时间:2017/10/23
Anticancer Activity  Cu(i)-catalyzed Click Reaction  Glycoconjugates  Picropodophyllotoxin  Podophyllotoxin  
The opioid receptor triple agonist DPI-125 produces analgesia with less respiratory depression and reduced abuse liability 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 7, 页码: 977-989
作者:  Yi, Shou-pu;  Kong, Qing-hong;  Li, Yu-lei;  Pan, Chen-ling;  Yu, Jie;  Cui, Ben-qiang;  Wang, Ying-fei;  Wang, Guan-lin;  Zhou, Pei-lan;  Wang, Li-li;  Gong, Ze-hui;  Su, Rui-bin;  Shen, Yue-hai;  Yu, Gang;  Chang, Kwen-jen
浏览  |  Adobe PDF(854Kb)  |  收藏  |  浏览/下载:341/66  |  提交时间:2017/08/29
Opioid Receptor  Mixed Agonist  Dpi-125  Analgesia  Respiratory Depression  Addiction