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Anti-arthritis effects of (E)-2,4-bis(p-hydroxyphenyl)-2-butenal through inhibition of STAT3 pathway 期刊论文
出版物, 3111, 期号: 0, 页码: 1-50
作者:  Jung Ok Ban;  Dae Hwan Kim;  Hee Pom Lee;  Chul Ju Hwang;  Jung-Hyun Shim;  Dae Joong Kim;  Tae Myoung Kim;  Heon Sang Jeong;  Seong Su Nah;  Hanyong Chen;  Zigang Dong;  Young Wan Ham;  Youngsoo Kim;  Sang-Bae Han;  Jin Tae Hong
Adobe PDF(1327Kb)  |  收藏  |  浏览/下载:163/3  |  提交时间:2017/07/24
Pharmacology and anti-addiction effects of the novel kappa opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin A 期刊论文
出版物, 3111, 期号: 0, 页码: 1-53
作者:  B Simonson;  A S Morani;  A W M Ewald;  L Walker;  N Kumar;  D Simpson;  J H Miller;  T E Prisinzano;  B M Kivell
Adobe PDF(1394Kb)  |  收藏  |  浏览/下载:275/1  |  提交时间:2017/07/24
The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:266/1  |  提交时间:2017/07/24
YC-1 inhibits proliferation of breast cancer cells by downregulating EZH2 expression via activation of c-Cbl and ERK 期刊论文
出版物, 3111, 期号: 0, 页码: 1-46
作者:  Ling-Chu Chang;  Hui-Yi Lin;  Meng-Tung Tsai;  Ruey-Hwang Chou;  Fang-Yu Lee;  Che-Ming Teng;  Min-Tsang Hsieh;  Hsin-Yi Hung;  Li-Jiau Huang;  Yung-Luen Yu;  Sheng-Chu Kuo
Adobe PDF(1357Kb)  |  收藏  |  浏览/下载:287/1  |  提交时间:2017/07/24
Yc-1  Triple-negative Breast Cancer  Erk  Ezh2  C-cbl  
Effects of CO-RM2 on LPS-induced vascular cell adhesion molecule-1 expression and leukocyte adhesion in human rheumatoid synovial fibroblasts 期刊论文
出版物, 3111, 期号: 0, 页码: 1-44
作者:  Pei-Ling Chi;  Yu-Chen Chuang;  Yu-Wen Chen;  Chih-Chung Lin;  Li-Der Hsiao;  Chuen-Mao Yang
Adobe PDF(1319Kb)  |  收藏  |  浏览/下载:157/1  |  提交时间:2017/07/24
Carbon Monoxide  Lipopolysaccharide  Vcam-1  Leukocyte Adhesion  
Resveratrol Decrease Fructose-Induced Oxidative Stress Mediated by NADPH Oxidase via an AMPK-Dependent Mechanism1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-44
作者:  Pei-Wen Cheng, PhD;  Wen-Yu Ho, MD, PhD;  Yu-Ting Su, MS;  Pei-Jung Lu,PhD;  Bo-Zone Chen MS;  Wen-Han Cheng, MS;  Wen-Hsien Lu, MD, MS;  Gwo-Ching Sun, MD;  Tung-Chen Yeh, MD;  Michael Hsiao DVM, PhD;  Ching-Jiunn Tseng, MD, PhD
Adobe PDF(1555Kb)  |  收藏  |  浏览/下载:107/1  |  提交时间:2017/07/24
Ampk  Hypertension  Nucleus Tractus Solitarii  Nitrogen Oxides  Resveratrol  
Nociceptin/Orphanin FQ peptide receptor antagonist JTC-801 reverses pain and anxiety symptoms in a rat model of PTSD 期刊论文
出版物, 3111, 期号: 0, 页码: 1-33
作者:  Y Zhang;  C D Simpson-Durand;  K M Standifer
Adobe PDF(1098Kb)  |  收藏  |  浏览/下载:106/1  |  提交时间:2017/07/24
Mono-/Bis-Alkenoic Acid Derivatives From an Endophytic Fungus Scopulariopsis candelabrum and Their Antifungal Activity 期刊论文
FRONTIERS IN CHEMISTRY, 2022
作者:  Tang, Jun;  Huang, Xueshuang;  Cao, Ming-Hang;  Wang, Zhiyan;  Yu, Zhiyin;  Yan, Yijun;  Huang, Jian-Ping;  Wang, Li;  Huang, Sheng-Xiong
Adobe PDF(1321Kb)  |  收藏  |  浏览/下载:139/57  |  提交时间:2023/09/08
Triterpenoids from Uncaria rhynchophylla and Their PTP1B Inhibitory Activity 期刊论文
PHYTON-INTERNATIONAL JOURNAL OF EXPERIMENTAL BOTANY, 2022, 卷号: 91, 期号: 8, 页码: 1809-1816
作者:  Luo, Shuaibin;  Zhang, Xuemei;  He, Kang;  Zou, Juan;  Geng, Chang-An
Adobe PDF(486Kb)  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/04/30
Uncaria rhynchophylla  triterpenoids  antidiabetic effects  PTP1B inhibitors  ALKALOIDS  
Synthesis and biological evaluation of (20S,24R)-epoxy-dammarane-3 beta,12 beta,25-triol derivatives as alpha-glucosidase and PTP1B inhibitors 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2022, 卷号: 31, 期号: 2, 页码: 350-367
作者:  Yang, Xiao-Tong;  Li, Tian-Ze;  Geng, Chang-An;  Liu, Pei;  Chen, Ji-Jun
Adobe PDF(1348Kb)  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/04/30
(20S,24R)-epoxy-dammarane-3 beta,12 beta,25-triol  alpha-glucosidase inhibitors  PTP1B inhibitors  Enzyme kinetics  TYROSINE-PHOSPHATASE 1B  DIABETES-MELLITUS  EPIDEMIOLOGY