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An Approach for the Synthesis of Pyrazolo[1,5-a]pyrimidines via Cu(II)-Catalyzed [3+3] Annulation of Saturated Ketones with Aminopyrazoles 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 18, 页码: 12762-12771
作者:  Ren,Jian;  Ding,Shihua;  Li,Xiaonian;  Bi,Ran;  Zhao,Qinshi
浏览  |  Adobe PDF(1469Kb)  |  收藏  |  浏览/下载:70/15  |  提交时间:2022/04/02
BIOLOGICAL EVALUATION  REGIOSELECTIVE SYNTHESIS  CASCADE REACTIONS  FUNCTIONALIZATION  DEHYDROGENATION  DISCOVERY  POTENT  BOND  SAR  
Huperserratines A and B, Two Macrocyclic Lycopodium Alkaloids with an Unusual Skeleton from Huperzia serrata 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020
作者:  Wu, Xing-De;  Li, Xiao-Nian;  Peng, Li-Yan;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1810Kb)  |  收藏  |  浏览/下载:133/66  |  提交时间:2021/01/05
Activation of SIK1 by phanginin A inhibits hepatic gluconeogenesis by increasing PDE4 activity and suppressing the cAMP signaling pathway 期刊论文
MOLECULAR METABOLISM, 2020
作者:  Liu, Siwen;  Huang, Suling;  Wu, Xingde;  Feng, Ying;  Shen, Yu;  Zhao, Qin-shi;  Leng, Ying
Adobe PDF(3899Kb)  |  收藏  |  浏览/下载:101/28  |  提交时间:2021/01/05
Magnograndins J-M, elemane sesquiterpenoids from the leaves of Magnolia grandiflora and their inhibitory effects on nitric oxide production 期刊论文
PHYTOCHEMISTRY LETTERS, 2019, 卷号: 31, 页码: 121-124
作者:  Ding, Lin-Fen;  Liu, Jiang-Xin;  Xie, Zhang-Qiao;  Wang, De-Shen;  Nie, Wei;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
浏览  |  Adobe PDF(649Kb)  |  收藏  |  浏览/下载:152/27  |  提交时间:2019/07/29
Magnolia grandiflora  Elemane sesquiterpenoid  Nitric oxide (NO)  
Three new Lycopodium alkaloids from Lycopodium japonicum 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2019, 卷号: 21, 期号: 1, 页码: 17-24
作者:  Zhu, Yu;  Dong, Liao-Bin;  Zhang, Zhi-Jun;  Fan, Min;  Zhu, Qin-Feng;  Qi, Yan-Yan;  Liu, Yu-Chen;  Peng, Li-Yan;  Wu, Xing-De;  Zhao, Qin-Shi
Adobe PDF(1103Kb)  |  收藏  |  浏览/下载:221/54  |  提交时间:2019/05/24
Lycopodiaceae  Lycopodium japonicum  Lycopodium alkaloids  T-type calcium channel  
Vibsane-Type Diterpenoids from Viburnum odoratissimum and Their Cytotoxic and HSP90 Inhibitory Activities 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 5, 页码: 1800049
作者:  Zhu, Qin-Feng;  Qi, Yan-Yan;  Zhang, Zhi-Jun;  Fan, Min;  Bi, Ran;  Su, Jia;  Wu, Xing-De;  Shao, Li-Dong;  Zhao, Qin-Shi
收藏  |  浏览/下载:335/0  |  提交时间:2018/07/16
Vibsane-type Diterpenoids  Viburnum Odoratissimum  Cytotoxicity  Hsp90 Inhibitor  
Hypofolins A - L, ent-Labdane Diterpenoids from the Roots of Hypoestes phyllostachya "Pink Splash' 期刊论文
CHEMISTRY & BIODIVERSITY, 2018, 卷号: 15, 期号: 6, 页码: e1800124
作者:  Cheng, Bin;  Ding, Lin-Fen;  Yan, Tong;  Xie, Zhang-Qiao;  Zhang, Zhi-jun;  Song, Liu-Dong;  Wu, Xing-De;  Zhao, Qin-Shi
Adobe PDF(1276Kb)  |  收藏  |  浏览/下载:135/74  |  提交时间:2019/03/29
Design, Synthesis, and Biological Activities of Vibsanin B Derivatives: A New Class of HSP90 C-Terminal Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 9053-9066
作者:  Shao, Li-Dong;  Su, Jia;  Ye, Baixin;  Liu, Jiang-Xin;  Zuo, Zhi-Li;  Li, Yan;  Wang, Yue-Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
Adobe PDF(5724Kb)  |  收藏  |  浏览/下载:368/41  |  提交时间:2017/12/18
Lycoplanine A, a C16N Lycopodium Alkaloid with a 6/9/5 Tricyclic Skeleton from Lycopodium complanatum 期刊论文
ORGANIC LETTERS, 2017, 卷号: 19, 期号: 17, 页码: 4668-4671
作者:  Zhang, Zhi-Jun;  Nian, Yin;  Zhu, Qin-Feng;  Li, Xiao-Nian;  Su, Jia;  Wu, Xing-De;  Yang, Jian;  Zhao, Qin-Shi
Adobe PDF(600Kb)  |  收藏  |  浏览/下载:300/99  |  提交时间:2017/10/23
Inhibitors  Huperzine  Channels  
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:297/68  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar