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Oxytocin inhibits the activity of acid-sensing ion channels through the vasopressin-1a receptor in primary sensory neurons1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-34
作者:  Fang Qiu;  Chun-Yu Qiu;  Huilan Cai;  Ting-Ting Liu;  Zu-Wei Qu;  Zhifan Yang;  Jia-Da Li;  Qun-Yong Zhou;  Wang-Ping Hu
Adobe PDF(850Kb)  |  收藏  |  浏览/下载:264/1  |  提交时间:2017/07/24
Oxytocin  Acid-sensing Ion Channel  Proton-gated Current  Vasopressin-1a Receptor  Dorsal Root Ganglion Neuron  Electrophysiology  Pain  
Chemical and biological comparison of different parts of Paeonia suffruticosa (Mudan) based on LCMS-IT-TOF and multi-evaluation in vitro 期刊论文
INDUSTRIAL CROPS AND PRODUCTS, 2020, 卷号: 144, 页码: 9
作者:  Pan, Yang;  Gao, Zhen;  Huang, Xiao-Yan;  Chen, Ji-Jun;  Geng, Chang-An
收藏  |  浏览/下载:224/0  |  提交时间:2020/03/24
Paeonia suffruticosa  Chemical profiles  LCMS-IT-TOF analyses  Biological comparison  Neurotransmitter receptors  Enzyme inhibition  
Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:  Zhou, Yeheng;  Sun, Wei;  Peng, Jiale;  Yan, Hui;  Zhang, Li;  Liu, Xingyong;  Zuo, Zhili
浏览  |  Adobe PDF(4739Kb)  |  收藏  |  浏览/下载:204/31  |  提交时间:2020/03/18
Acetylcholinesterase  Drug design  N-acylhydrazone  Dementia  Copper-chelating  N-Benzylpiperidine  
Identification of novel monoamine oxidase selective inhibitors employing a hierarchical ligand-based virtual screening strategy 期刊论文
FUTURE MEDICINAL CHEMISTRY, 2019, 卷号: 11, 期号: 8, 页码: 801-816
作者:  Wang, Dong;  Li, Zhaoyang;  Liu, Yi;  Chen, Mo;  Chen, Nianhang;  Zuo, Zhili;  Kong, De-Xin
浏览  |  Adobe PDF(1462Kb)  |  收藏  |  浏览/下载:176/36  |  提交时间:2019/09/10
BRS-3D  monoamine oxidase selective inhibitors  virtual screening  
Antidepressant potential of Uncaria rhynchophylla and its active flavanol, catechin, targeting melatonin receptors 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2019, 卷号: 232, 页码: 39-46
作者:  Geng, Chang-An;  Yang, Tong-Hua;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(3731Kb)  |  收藏  |  浏览/下载:215/49  |  提交时间:2019/06/24
Uncaria rhynchophylla  Catechin  Melatonin receptors  Metabolites  Antidepressant activity  
Celastrol Protects From Cholestatic Liver Injury Through Modulation of SIRT1-FXR Signaling 期刊论文
MOLECULAR & CELLULAR PROTEOMICS, 2019, 卷号: 18, 期号: 3, 页码: 520-533
作者:  Zhao, Qi;  Liu, Fang;  Cheng, Yan;  Xiao, Xue-Rong;  Hu, Dan-Dan;  Tang, Ying-Mei;  Bao, Wei-Min;  Yang, Jin-Hui;  Jiang, Tao;  Hu, Jia-Peng;  Gonzalez, Frank J.;  Li, Fei
浏览  |  Adobe PDF(4782Kb)  |  收藏  |  浏览/下载:183/60  |  提交时间:2019/07/29
Discovery of novel indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors by virtual screening 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2019, 卷号: 78, 页码: 306-316
作者:  Zhou, Yeheng;  Peng, Jiale;  Li, Penghua;  Du, Haibo;  Li, Yaping;  Li, Yingying;  Zhang, Li;  Sun, Wei;  Liu, Xingyong;  Zuo, Zhili
浏览  |  Adobe PDF(2732Kb)  |  收藏  |  浏览/下载:262/42  |  提交时间:2019/03/25
IDO1  Molecular docking  HipHop pharmacophore  3D-QSAR  PAINS  
Thiodiketopiperazines Produced by Penicillium crustosum and Their Activities to Promote Gastrointestinal Motility 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 2, 页码: 8
作者:  He, Xin;  Yang, Jing;  Qiu, Ling;  Feng, Dan;  Ju, Feng;  Tan, Lu;  Li, Yu-Zhi;  Gu, Yu-Cheng;  Zhang, Zhen;  Guo, Da-Le;  Deng, Yun
浏览  |  Adobe PDF(2070Kb)  |  收藏  |  浏览/下载:155/32  |  提交时间:2019/03/18
Penicillium crustosum  Isaria cicadae  thiodiketopiperazines  Mosher analysis  ECD calculation  gastrointestinal motility  
Synthesis and biological evaluation of magnolol derivatives as melatonergic receptor agonists with potential use in depression 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 期号: 0, 页码: 381-393
作者:  Yang, Tong-Hua;  Ma, Yun-Bao;  Geng, Chang-An;  Yan, De-Xiu;  Huang, Xiao-Yan;  Li, Tian-Ze;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(2088Kb)  |  收藏  |  浏览/下载:232/75  |  提交时间:2018/10/04
Depression  Magnolol Derivatives  Mt1/2 Receptors  Metabolites  Monoamine Neurotransmitter  
Research Progress of Polycyclic Polyprenylated Acylphloroglucinols 期刊论文
CHEMICAL REVIEWS, 2018, 卷号: 118, 期号: 7, 页码: 3508-3558
作者:  Yang, Xing-Wei;  Grossman, Robert B.;  Xu, Gang
浏览  |  Adobe PDF(27097Kb)  |  收藏  |  浏览/下载:548/108  |  提交时间:2018/05/08