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Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:  Shao, Li-Dong;  Bao, Ying;  Shen, Yu;  Su, Jia;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1336Kb)  |  收藏  |  浏览/下载:301/68  |  提交时间:2017/07/31
11 Beta-hsd1 Inhibitor  Hupehenols  Dammarane  Sar  
呋喃卡山烷二萜衍生物及其药物组合物和其在制药中的应用 专利
申请日期: 2017-01-13, 公开日期: 2017-06-09
发明人:  赵勤实;  冷颖;  吴兴德;  黄素玲;  苏佳;  邵立东;  彭丽艳
收藏  |  浏览/下载:145/0  |  提交时间:2018/05/10
Synthesis of hupehenols A, B, and E from protopanaxadiol 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 42, 页码: 35792-35803
作者:  Shao, Li-Dong;  Xu, Jun;  Li, Xiao-Nian;  Zhang, Zhi-Jun;  Shi, Xin;  Ren, Jian;  He, Juan;  Zhao, Yu;  Leng, Ying;  Xia, Chengfeng;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1402Kb)  |  收藏  |  浏览/下载:214/59  |  提交时间:2016/08/22
Hupehenols A-E, Selective 11 beta-Hydroxysteroid Dehydrogenase Type 1 (11 beta-HSD1) Inhibitors from Viburnum hupehense 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2015, 卷号: 78, 期号: 2, 页码: 330-334
作者:  Chen, Xuan-Qin;  Shao, Li-Dong;  Pal, Mahesh;  Shen, Yu;  Cheng, Xiao;  Xu, Gang;  Peng, Li-Yan;  Wang, Kou;  Pan, Zheng-Hong;  Li, Ming-Ming;  Leng, Ying;  He, Juan;  Zhao, Qin-Shi;  He,J (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650204,Yunnan,Peoples R China.;  hejuan@mail.kib.ac.cn;  qinshizhao@mail.kib.ac.cn
浏览  |  Adobe PDF(811Kb)  |  收藏  |  浏览/下载:300/88  |  提交时间:2015/06/29
Discovery and structure-activity relationships of ent-Kaurene diterpenoids as potent and selective 11 beta-HSD1 inhibitors: Potential impact in diabetes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 403-414
作者:  Deng, Xu;  Shen, Yu;  Yang, Jing;  He, Juan;  Zhao, Yu;  Peng, Li-Yan;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1215Kb)  |  收藏  |  浏览/下载:400/150  |  提交时间:2013/10/16
Ent-kaurene Diterpenoids  Structure-activity Relationship Studies  Selective 11 Beta-hsd1 Inhibitors  Urea Derivatives  Diabetes  
达玛烷三萜衍生物及其药物组合物和其在制药中的应用 专利
专利类型: 发明, 专利号: CN201210379644.7, 申请日期: 2012-10-09, 公开日期: 2014-04-09
发明人:  赵勤实;  夏成峰;  冷颖;  邵立东
Adobe PDF(1355Kb)  |  收藏  |  浏览/下载:161/4  |  提交时间:2016/12/19
丹参酮衍生物,其药物组合物及其在制药中的应用 专利
申请日期: 2011-07-02, 公开日期: 2012-01-04
发明人:  赵勤实;  冷颖;  赵昱;  邓旭;  沈瑜;  张丽娜
收藏  |  浏览/下载:97/0  |  提交时间:2018/05/10