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Stereoselective Synthesis of Diazabicyclic beta-Lactams through Intramolecular Amination of Unactivated C(sp(3))-H Bonds of Carboxamides by Palladium Catalysis 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 81, 期号: 3, 页码: 956-968
作者:  Zhang, Shi-Jin;  Sun, Wen-Wu;  Cao, Pei;  Dong, Xiao-Ping;  Liu, Ji-Kai;  Wu, Bin
浏览  |  Adobe PDF(866Kb)  |  收藏  |  浏览/下载:311/52  |  提交时间:2016/06/27
Design, Synthesis, and Structural Optimization of Lycorine-Derived Phenanthridine Derivatives as Wnt/beta-Catenin Signaling Pathway Agonists 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2016, 卷号: 79, 期号: 1, 页码: 180-188
作者:  Chen, Duo-Zhi;  Jing, Chen-Xu;  Cai, Jie-Yun;  Wu, Ji-Bo;  Wang, Sheng;  Yin, Jun -Lin;  Li, Xiao-Nian;  Li, Lin;  Hao, Xiao-Jiang
浏览  |  Adobe PDF(3043Kb)  |  收藏  |  浏览/下载:304/73  |  提交时间:2016/06/27
Design and synthesis of new 2-arylnaphthyridin-4-ones as potent antitumor agents targeting tumorigenic cell lines 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 90, 页码: 775-787
作者:  Liu, Chin-Yu;  Cheng, Yung-Yi;  Chang, Ling-Chu;  Huang, Li-Jiau;  Chou, Li-Chen;  Huang, Chi-Hung;  Tsai, Meng-Tung;  Liao, Chih-Chang;  Hsu, Mei-Hua;  Lin, Hui-Yi;  Wu, Tian-Shung;  Wen, Yen-Fang;  Zhao, Yu;  Kuo, Sheng-Chu;  Lee, Kuo-Hsiung;  Kuo,SC (reprint author),China Med Univ,Grad Inst Pharmaceut Chem,91 Hsueh Shih Rd,Taichung 40402,Taiwan.;  sckuo@mail.cmu.edu.tw;  khlee@unc.edu
浏览  |  Adobe PDF(1696Kb)  |  收藏  |  浏览/下载:328/74  |  提交时间:2015/06/29
2-arylnaphthyridin-4-ones  Antitumor Agents  Phosphate Prodrug  
Dopamine derivatives from the insect Polyrhachis dives as inhibitors of ROCK1/2 and stimulators of neural stem cell proliferation 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 46, 页码: 8852-8857
作者:  Tang, Jian-Jun ab;  Zhang, Li;  Jiang, Li-Ping;  Di, Lei;  Yan, Yong-Ming;  Tu, Zheng-Chao;  Yang, Cui-Ping;  Zuo, Zhi-Li;  Hou, Bo;  Xia, Hou-Lin;  Chen, Yong-Bin;  Cheng, Yong-Xian;  Tu,ZC (reprint author),Chinese Acad Sci,Guangzhou Inst Biomed & Hlth,Key Lab Regenerat Biol,Guangzhou 510530,Guangdong,Peoples R China.;  tu_zhengchao@gibh.ac.cn;  ybchen@mail.kiz.ac.cn;  yxcheng@mail.kib.ac.cn
浏览  |  Adobe PDF(678Kb)  |  收藏  |  浏览/下载:445/95  |  提交时间:2015/01/20
Polyrhachis Dives  Dopamine Derivative  Rock1/2 Inhibitors  Nscs  
Four New Polycyclic Meroterpenoids from Ganoderma cochlear 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 20, 页码: 5262-5265
作者:  Peng, Xing-Rong;  Liu, Jie-Qing;  Wan, Luo-Sheng;  Li, Xiao-Nian;  Yan, Yu-Xin;  Qiu, Ming-Hua;  Qiu,MH (reprint author),Chinese Acad Sci,Kunming Inst Bot,Key Lab Phytochem & Plant Resources West China,Kunming 650201,Peoples R China.;  mhchiu@mail.kib.ac.cn
Adobe PDF(290Kb)  |  收藏  |  浏览/下载:333/101  |  提交时间:2014/11/25
Triterpenoids  Fornicatum  Lucidum  Sinense  
Multidrug resistance-selective antiproliferative activity of Piper amide alkaloids and synthetic analogues 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 20, 页码: 4818-4821
作者:  Wang, Yue-Hu;  Goto, Masuo;  Wang, Li-Ting;  Hsieh, Kan-Yen;  Morris-Natschke, Susan L.;  Tang, Gui-Hua;  Long, Chun-Lin;  Lee, Kuo-Hsiung;  Wang,YH (reprint author),Univ N Carolina,Eshelman Sch Pharm,Nat Prod Res Labs,Chapel Hill,NC 27599 USA.;  wangyuehu@mail.kib.ac.cn;  khlee@unc.edu
Adobe PDF(492Kb)  |  收藏  |  浏览/下载:289/67  |  提交时间:2014/11/25
Piper  Piperaceae  Amide Alkaloids  Cytotoxicity  Multidrug Resistance  
Aspergillines A-E, Highly Oxygenated Hexacyclic Indole-Tetrahydrofuran-Tetramic Acid Derivatives from Aspergillus versicolor 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 19, 页码: 5016-5019
作者:  Zhou, Min;  Miao, Ming-Ming;  Du, Gang;  Li, Xiao-Nian;  Shang, Shan-Zhai;  Zhao, Wei;  Liu, Zhi-Hua;  Yang, Guang-Yu;  Che, Chun-Tao;  Hu, Qiu-Fen;  Gao, Xue-Mei;  Hu,QF (reprint author),China Tobacco Yunnan Ind Co Ltd,Key Lab Tobacco Chem Yunnan Prov,Kunming 650231,Peoples R China.;  huqiufena@aliyun.com;  gao_xuemei@hotmail.com
Adobe PDF(277Kb)  |  收藏  |  浏览/下载:309/88  |  提交时间:2014/11/25
Cyclopiazonic Acid  Biological-activity  Biosynthesis  Flavus  
Synthesis and conformation studies of rubiyunnanin B analogs 期刊论文
TETRAHEDRON, 2014, 卷号: 70, 期号: 37, 页码: 6630-6640
作者:  Liu, Na-Na;  Zhao, Si-Meng;  Zhao, Jing-Feng;  Zeng, Guang-Zhi;  Tan, Ning-Hua;  Liu, Jian-Ping;  Tan, NH (reprint author), Chinese Acad Sci, Kunming Inst Bot, State Key Lab Phytochem & Plant Resources West Ch, Kunming 650201, Peoples R China.;  nhtan@mail.kib.ac.cn;  jpliu@ynu.edu.cn
Adobe PDF(619Kb)  |  收藏  |  浏览/下载:211/48  |  提交时间:2014/10/11
Rubiyunnanin b Analogs  Synthesis  Conformation Studies  Bioactivities  
Cyclohexane-Fused Octahydroquinolizine Alkaloids from Myrioneuron faberi with Activity against Hepatitis C Virus 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2014, 卷号: 79, 期号: 17, 页码: 7945-7950
作者:  Cao, Ming-Ming;  Zhang, Yu;  Li, Xiao-Hui;  Peng, Zong-Gen;  Jiang, Jian-Dong;  Gu, Yu-Cheng;  Di, Ying-Tong;  Li, Xiao-Nian;  Chen, Duo-Zhi;  Xia, Cheng-Feng;  He, Hong-Ping;  Li, Shun-Lin;  Hao, Xiao-Jiang;  haoxj@mail.kib.ac.cn
Adobe PDF(364Kb)  |  收藏  |  浏览/下载:287/75  |  提交时间:2014/11/25
Biomimetic Synthesis  Nutans  Nitraramine  Skeleton  Therapy  
Anti-Hepatitis B Virus Norbisabolane Sesquiterpenoids from Phyllanthus acidus and the Establishment of Their Absolute Configurations Using Theoretical Calculations 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2014, 卷号: 79, 期号: 12, 页码: 5432-5447
作者:  Lv, Jun-Jiang;  Yu, Shan;  Wang, Ya-Feng;  Wang, Dong;  Zhu, Hong-Tao;  Cheng, Rong-Rong;  Yang, Chong-Ren;  Xu, Min;  Zhang, Ying-Jun;  Xu,M (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  minxu@mail.kib.ac.cn;  zhangyj@mail.kib.ac.cn
Adobe PDF(655Kb)  |  收藏  |  浏览/下载:310/90  |  提交时间:2014/07/28
Antineoplastic Agents  Acuminatus Vahl  Glycosides  Emblica  Roots  Secretion  Norsesquiterpenoids  Pyrimidine  Inhibitors