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Synthesis and biological evaluation of chepraecoxin A derivatives as alpha-glucosidase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020
作者:  Yang, Xiao-Tong;  Geng, Chang-An;  Li, Tian-Ze;  Deng, Zhen-Tao;  Chen, Ji-Jun
Adobe PDF(675Kb)  |  收藏  |  浏览/下载:127/27  |  提交时间:2021/01/05
Amomutsaokols A-K, diarylheptanoids from Amomum tsao-ko and their alpha-glucosidase inhibitory activity 期刊论文
PHYTOCHEMISTRY, 2020
作者:  He, Xiao-Feng;  Wang, Hui-Mei;  Geng, Chang-An;  Hu, Jing;  Zhang, Xue-Mei;  Guo, Yuan-Qiang;  Chen, Ji-Jun
浏览  |  Adobe PDF(3949Kb)  |  收藏  |  浏览/下载:99/40  |  提交时间:2021/01/05
Tsaokopyranols A-M, 2,6-epoxydiarylheptanoids from Amomum tsao-ko and their alpha-glucosidase inhibitory activity 期刊论文
BIOORGANIC CHEMISTRY, 2020
作者:  He, Xiao-Feng;  Zhang, Xu-Ke;  Geng, Chang-An;  Hu, Jing;  Zhang, Xue-Mei;  Guo, Yuan-Qiang;  Chen, Ji-Jun
浏览  |  Adobe PDF(2442Kb)  |  收藏  |  浏览/下载:85/32  |  提交时间:2021/01/05
Polybenzyls from Gastrodia elata, their agonistic effects on melatonin receptors and structure-activity relationships 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3299-3306
作者:  Chen, Si-Yue;  Geng, Chang-An;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Yang, Xiao-Tong;  Su, Li-Hua;  He, Xiao-Feng;  Li, Tian-Ze;  Deng, Zhen-Tao;  Gao, Zhen;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(1837Kb)  |  收藏  |  浏览/下载:176/35  |  提交时间:2019/09/10
Gastrodia elata  Polybenzyls  Melatonin receptors  Structure-activity relationships  Docking study  
Synthesis and Cytotoxicity Evaluation of Tropinone Derivatives. 期刊论文
Natural products and bioprospecting, 2017, 卷号: 7, 期号: 2, 页码: 215-223
作者:  Yin, Xiu-Juan;  Geng, Chang-An;  Chen, Xing-Long;  Sun, Chang-Li;  Yang, Tong-Hua;  Li, Tian-Ze;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(758Kb)  |  收藏  |  浏览/下载:216/128  |  提交时间:2019/03/29
Bioactivity-guided synthesis of gramine derivatives as new MT1 and 5-HT1A receptors agonists 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2017, 卷号: 19, 期号: 6, 页码: 610-622
作者:  Yin, Xiu-Juan;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Geng, Chang-An;  Li, Tian-Ze;  Chen, Xing-Long;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
浏览  |  Adobe PDF(2718Kb)  |  收藏  |  浏览/下载:317/58  |  提交时间:2017/07/10
Gramine  Melatonin Receptor  5-hydroxy-tryptamine Receptor  Agonistic Activity  Structure-activity Relationships  
Bioactivity-guided synthesis of tropine derivatives as new agonists for melatonin receptors 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 51, 页码: 45059-45063
作者:  Yin, Xiu-Juan;  Geng, Chang-An;  Huang, Xiao-Yan;  Chen, Hao;  Ma, Yun-Bao;  Chen, Xing-Long;  Sun, Chang-Li;  Yang, Tong-Hua;  Zhou, Jun;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(1380Kb)  |  收藏  |  浏览/下载:235/62  |  提交时间:2016/08/22
Synthesis of erythrocentaurin derivatives as a new class of hepatitis B virus inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 7, 页码: 1568-1571
作者:  Geng, Chang-An;  Huang, Xiao-Yan;  Ma, Yun-Bao;  Zhang, Xue-Mei;  Chen, Ji-Jun;  Chen,JJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  chenjj@mail.kib.ac.cn
Adobe PDF(1409Kb)  |  收藏  |  浏览/下载:288/110  |  提交时间:2015/06/29
Erythrocentaurin  Anti-hbv Activity  Structure-activity Relationships  
Isolation, synthesis and anti-hepatitis B virus evaluation of p-hydroxyacetophenone derivatives from Artemisia capillaris 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 7, 页码: 1509-1514
作者:  Zhao, Yong;  Geng, Chang-An;  Chen, Hao;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Cao, Tuan-Wu;  He, Kang;  Wang, Hao;  Zhang, Xue-Mei;  Chen, Ji-Jun;  Chen,JJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.;  chenjj@mail.kib.ac.cn
Adobe PDF(2494Kb)  |  收藏  |  浏览/下载:298/96  |  提交时间:2015/06/29
Artemisia Capillaris  P-hydroxyacetophenone Derivatives  Anti-hbv Activity  Structure-activity Relationships  
Design, Synthesis and Biological Evaluation of Caudatin Analogs as Potent Hepatitis B Virus Inhibitors 期刊论文
MEDICINAL CHEMISTRY, 2015, 卷号: 11, 期号: 2, 页码: 165-179
作者:  Wang, Li-Jun;  Chen, Hao;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Geng, Chang-An;  Zhang, Xue-Mei;  Chen, Ji-Jun;  Chen,JJ (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650201,Peoples R China.
Adobe PDF(375Kb)  |  收藏  |  浏览/下载:192/66  |  提交时间:2015/06/29
Anti-hbv Activity  Caudatin Analogs  Hepatitis b e Antigen (Hbeag)  Hepatitis b Surface Antigen (Hbsag)  Hbv Dna Replication  Structure-activity Relationships(Sars)  Synthesis