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The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP)1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-42
作者:  C Pergola;  J Gerstmeier;  B Monch;  B Çaliskan;  S Luderer;  C Weinige;  D Barz;  J Maczewsky;  S Pace;  A Rossi;  L Sautebin;  E Banoglu;  O Werz
Adobe PDF(1387Kb)  |  收藏  |  浏览/下载:495/1  |  提交时间:2017/07/24
Discovery and bioinspired total syntheses of unprecedented sesquiterpenoid dimers unveiled bifurcating [4+2] cycloaddition and target differentiation of enantiomers 期刊论文
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 4
作者:  He, Tao-Bin;  Yan, Bing-Chao;  Zhou, Yuan-Fei;  Sang, Yue-Qian;  Li, Xiao-Nian;  Sun, Han-Dong;  Wang, Chu;  Xue, Xiao-Song;  Puno, Pema-Tenzin
浏览  |  Adobe PDF(3322Kb)  |  收藏  |  浏览/下载:256/85  |  提交时间:2024/05/09
DIELS-ALDER REACTION  BIOMIMETIC SYNTHESES  EFFICIENT ACCESS  DEHYDROGENATION  CYCLOHEXANONES  BIOSYNTHESIS  CONVERSION  OXIDATION  DYNAMICS  PHENOLS  
Sesquiterpenoids from Alpinia oxyphylla with GLP-1 Stimulative Effects through Ca2+/CaMKII and PKA Pathways and Multiple-Enzyme Inhibition 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 71, 期号: 43, 页码: 16148-16159
作者:  Cui,Can;  Wu,Sheng-Li;  Chen,Ji-Jun;  Gongpan,Pianchou;  Guan,Min;  Geng,Chang-An
浏览  |  Adobe PDF(2550Kb)  |  收藏  |  浏览/下载:191/43  |  提交时间:2024/07/10
Alpinia oxyphylla  sesquiterpenoids  GLP-1 stimulation  Ca2+/CaMKII and PKA pathways  alpha-glucosidase and PTP1B inhibitory activity  
Dirigent gene editing of gossypol enantiomers for toxicity-depleted cotton seeds 期刊论文
NATURE PLANTS, 2023, 卷号: 9, 期号: 4, 页码: 605-+
作者:  Lin,Jia-Ling;  Fang,Xin;  Li,Jian-Xu;  Chen,Zhi-Wen;  Wu,Wen-Kai;  Guo,Xiao-Xiang;  Liu,Ning-Jing;  Huang,Jia-Fa;  Chen,Fang-Yan;  Wang,Ling-Jian;  Xu,Baofu;  Martin,Cathie;  Chen,Xiao-Ya;  Huang,Jin-Quan
浏览  |  Adobe PDF(9213Kb)  |  收藏  |  浏览/下载:195/66  |  提交时间:2024/07/22
DOMAIN-CONTAINING PROTEIN  BIOSYNTHESIS  (-)-GOSSYPOL  SYNTHASE  (+)-GOSSYPOL  METABOLISM  EXPRESSION  REDUCTION  
Meroterpenoids from Ganoderma petchii inhibiting migration of triple negative breast cancer cells 期刊论文
FITOTERAPIA, 2023, 卷号: 167, 页码: 105505
作者:  Zhang,Jiao-Jiao;  Guo,Ping-Xia;  Yang,Zhong-Hui;  Cai,Dan;  Dai,Wei-Feng;  Lu,Qing;  Cheng,Yong-Xian
浏览  |  Adobe PDF(3320Kb)  |  收藏  |  浏览/下载:149/37  |  提交时间:2024/07/25
Ganoderma petchii  Meroterpenoids  Triple negative breast cancer  Cell migration  
海菜花的化学成分及其生物活性研究 学位论文
: 中国科学院大学, 2022
作者:  刘洪星
Adobe PDF(6132Kb)  |  收藏  |  浏览/下载:142/0  |  提交时间:2024/05/14
海菜花,Ottelione,二芳基庚烷,糖尿病,抗肿瘤  Ottelia acuminata, Ottelione, Diarylheptanoids, DM, Antitumor  
玛咖活性成分及其不同加工方式下化学成分变化的研究 学位论文
: 中国科学院大学, 2022
作者:  张然然
Adobe PDF(5266Kb)  |  收藏  |  浏览/下载:66/0  |  提交时间:2024/05/14
十字花科,玛咖,硫代乙内酰脲,生物活性, UPLC-MS/MS-MRM,成分分析  Cruciferous, Lepidium meyenii, Thiohydantoin, Bioactivity, UPLCMS/MS-MRM, Analysis of chemical constituents  
中药砂仁降血糖活性成分研究 学位论文
: 中国科学院大学, 2022
作者:  丁敏
Adobe PDF(6349Kb)  |  收藏  |  浏览/下载:220/0  |  提交时间:2024/05/14
砂仁,姜科,降木脂素,降血糖活性,促GLP-1分泌,GPa抑制活性  Amomum villosum  Zingiberaceae  norlignans  antidiabetic effects  GLP-1 stimulation  GPa inhibition  
瘤枝五味子的化学成分及其生物活性研究 学位论文
: 中国科学院大学, 2022
作者:  张水妹
Adobe PDF(5213Kb)  |  收藏  |  浏览/下载:194/0  |  提交时间:2024/05/14
瘤枝五味子,木脂素,倍半萜,量子化学计算,神经保护活性  Schisandra bicolor var. tuberculata, Lignans, Sesquiterpenoids, Quantum chemical calculation, Neuroprotective activities  
Phaeosphspirone (1/1 '), a pair of unique polyketide enantiomers with an unusual 6/5/5/6 tetracyclic ring from the desert plant endophytic fungus Phaeosphaeriaceae sp. 期刊论文
PHYTOCHEMISTRY, 2022, 卷号: 194, 页码: 112969
作者:  Xu,Zhen-Lu;  Yan,Dao-Jiang;  Tan,Xiang-Mei;  Niu,Shu-Bin;  Yu,Meng;  Sun,Bing-Da;  Ding,Cai-Feng;  Zhang,Yong-Gang;  Ding,Gang
收藏  |  浏览/下载:440/0  |  提交时间:2022/04/02
Phaeosphspirone  Phaeosphaeriaceae  Absolute configurations  Biosynthetic pathway  Cytotoxicity  ASSISTED STRUCTURE ELUCIDATION  BIOSYNTHESIS  REVISION