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A small trypsin inhibitor from the frog of Odorrana grahami 期刊论文
BIOCHIMIE, 2008, 卷号: 90, 期号: 9, 页码: 1356-1361
作者:  Li, Jianxu;  Wu, Jing;  Wang, Yipeng;  Xu, Xueqing;  Liu, Tongguang;  Lai, Ren;  Zhu, Huajie
Adobe PDF(329Kb)  |  收藏  |  浏览/下载:290/150  |  提交时间:2011/11/24
Serine Protease Inhibitor  Amphibian  Odorrana Grahami  
Amide N-glycosylation by Asm25, an N-glycosyltransferase of ansamitocins 期刊论文
CHEMISTRY & BIOLOGY, 2008, 卷号: 15, 期号: 8, 页码: 863-874
作者:  Zhao, Peiji;  Bai, Linquan;  Ma, Juan;  Zeng, Ying;  Li, Lei;  Zhang, Yirong;  Lu, Chunhua;  Dai, Huanqin;  Wu, Zhaoxian;  Li, Yaoyao;  Wu, Xuan;  Chen, Gang;  Hao, Xiaojiang;  Shen, Yuemao;  Deng, Zixin;  Floss, Heinz G.
Adobe PDF(1375Kb)  |  收藏  |  浏览/下载:354/128  |  提交时间:2011/11/24
Biosynthetic Gene-cluster  Lechevalieria-aerocolonigenes Atcc-39243  Escherichia-coli  3-amino-5-hydroxybenzoic Acid  Actinosynnema-pretiosum  Maytansinoid Antibiotics  Streptomyces Sp  Indolocarbazole  Expression  Substrate  
Anti-HBV agents. Part 1: Synthesis of alisol A derivatives: A new class of hepatitis B virus inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 卷号: 18, 期号: 16, 页码: 4647-4650
作者:  Zhang, Quan;  Jiang, Zhi-Yong;  Luo, Jie;  Cheng, Pi;  Ma, Yun-Bao;  Zhang, Xue-Mei;  Zhang, Feng-Xue;  Zhou, Jun;  Chen, Ji-Jun
Adobe PDF(173Kb)  |  收藏  |  浏览/下载:255/79  |  提交时间:2011/11/24
Anti-hbv Activity  Alisol a  Derivatives  Synthesis  
Plant-derived small molecule albaconol suppresses LPS-triggered proinflammatory cytokine production and antigen presentation of dendritic cells by impairing NF-kappa B activation 期刊论文
INTERNATIONAL IMMUNOPHARMACOLOGY, 2008, 卷号: 8, 期号: 8, 页码: 1103-1111
作者:  Liu, Qiuyan;  Shu, Xiaoli;  Sun, Anna;  Sun, Qiaoling;  Zhang, Chaoxiong;  An, Huazhang;  Liu, Jikai;  Cao, Xuetao
Adobe PDF(929Kb)  |  收藏  |  浏览/下载:296/79  |  提交时间:2011/12/19
Dendritic Cell  Immunosuppression  Inflammation  Cytokines  Nf-kappa b  
Albaconol, a plant-derived small molecule, inhibits macrophage function by suppressing NF-kappa B activation and enhancing SOCS1 expression 期刊论文
CELLULAR & MOLECULAR IMMUNOLOGY, 2008, 卷号: 5, 期号: 4, 页码: 271-278
作者:  Liu, Qiuyan;  Shu, Xiaoli;  Wang, Li;  Sun, Anna;  Liu, Jikai;  Cao, Xuetao
Adobe PDF(393Kb)  |  收藏  |  浏览/下载:345/72  |  提交时间:2011/11/24
Immunosuppressant  Macrophage  Proinflammatory Cytokine  Nf-kappa b  Socs1  
Two new oleanane-type triterpenoids from Buddleja asiatica 期刊论文
ZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES, 2008, 卷号: 63, 期号: 7, 页码: 915-919
作者:  Liu, Ya-Ping;  Cai, Xiang-Hai;  Du, Zhi-Zhi;  Li, Wei-Qi;  Luo, Xiao-Dong
Adobe PDF(93Kb)  |  收藏  |  浏览/下载:369/109  |  提交时间:2012/07/25
Buddleja Asiatica  Oleanane Triterpenoids  13  28-epoxy-23-hydroxy-11-oleanene-3-one  13  28-epoxy-21 Beta  13  23-dihydroxy-11-oleanene-3-one  28-epoxy-3 Beta  23-o-isopropylidene-11-oleanene  
High-throughput screening of novel antagonists on melanin-concentrating hormone receptor-1 期刊论文
ACTA PHARMACOLOGICA SINICA, 2008, 卷号: 29, 期号: 6, 页码: 752-758
作者:  Yan, Jian-hua;  Li, Qun-yi;  Boutin, Jean A.;  Renard, M. Pierre;  Ding, Yi-xiang;  Hao, Xiao-jiang;  Zhao, Wei-min;  Wang, Ming-wei
Adobe PDF(435Kb)  |  收藏  |  浏览/下载:358/105  |  提交时间:2011/12/19
Melanin-concentrating Hormone  Melanin-concentrating Hormone Receptor-1  Antagonist  
Sulfonated guaianolides from Saussurea lappa 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2008, 卷号: 56, 期号: 6, 页码: 864-865
作者:  Wang, Fei;  Xie, Zheng-Hong;  Gao, Yuan;  Xu, Yao;  Cheng, Xue-Lian;  Liu, Ji-Kai
Adobe PDF(70Kb)  |  收藏  |  浏览/下载:276/77  |  提交时间:2012/10/12
Saussurea Lappa  Sesquiterpene Lactone  Sulfonated Guaianolide  Sulfocostunolide a  Sulfocostunolide b  
Characterization of tailoring genes involved in the modification of geldanamycin polyketide in Streptomyces hygroscopicus JCM4427 期刊论文
JOURNAL OF MICROBIOLOGY AND BIOTECHNOLOGY, 2008, 卷号: 18, 期号: 6, 页码: 1101-1108
作者:  Shin, Jin Chul;  Na, Zhu;  Lee, Dongho;  Kim, Woncheol;  Lee, Kyeong;  Shen, Yue-Mao;  Paik, Sang-Gi;  Hong, Young-Soo;  Lee, Jung Joon
Adobe PDF(1704Kb)  |  收藏  |  浏览/下载:321/111  |  提交时间:2011/11/24
Geldanamycin  Biosynthesis  Streptomyces  Polyketide  
Blockade of cholecystokinin-2 receptor and cyclooxygenase-2 synergistically induces cell apoptosis, and inhibits the proliferation of human gastric cancer cells in vitro 期刊论文
CANCER LETTERS, 2008, 卷号: 263, 期号: 2, 页码: 302-311
作者:  Sun, Wei-Hao;  Zhu, Feng;  Chen, Guo-Sheng;  Su, Han;  Luo, Cheng;  Zhao, Qin-Shi;  Zhang, Yuan;  Shao, Yun;  Sun, Jian;  Zhou, Su-Ming;  Ding, Guo-Xian;  Cheng, Yun-Lin
Adobe PDF(809Kb)  |  收藏  |  浏览/下载:347/103  |  提交时间:2011/11/24
Cholecystokinin-2 Receptor  Cyclooxygenase-2  Mkn-45 Cell  Proliferation  Apoptosis