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Stereoselective Synthesis of Diazabicyclic beta-Lactams through Intramolecular Amination of Unactivated C(sp(3))-H Bonds of Carboxamides by Palladium Catalysis 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 81, 期号: 3, 页码: 956-968
作者:  Zhang, Shi-Jin;  Sun, Wen-Wu;  Cao, Pei;  Dong, Xiao-Ping;  Liu, Ji-Kai;  Wu, Bin
Adobe PDF(866Kb)  |  收藏  |  浏览/下载:317/54  |  提交时间:2016/06/27
Construction of Tetracyclic 3-Spirooxindole through Cross-Dehydrogenation of Pyridinium: Applications in Facile Synthesis of (+/-)-Corynoxine and (+/-)-Corynoxine B 期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2014, 卷号: 136, 期号: 52, 页码: 17962-17965
作者:  Xu, Jun;  Shao, Li-Dong;  Li, Dashan;  Deng, Xu;  Liu, Yu-Chen;  Zhao, Qin-Shi;  Xia, Chengfeng
Adobe PDF(696Kb)  |  收藏  |  浏览/下载:510/83  |  提交时间:2015/06/17
Synthesis and cytotoxic activity of novel 1-((indol-3-yl)methyl)-1H-imidazolium salts 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 21, 页码: 4926-4930
作者:  Xu, Xiao-Liang;  Wang, Jia;  Yu, Chun-Lei;  Chen, Wen;  Li, Ying-Chao;  Li, Yan;  Zhang, Hong-Bin;  Yang, Xiao-Dong;  Li,Y (reprint author),Chinese Acad Sci,Kunming Inst Bot,State Key Lab Phytochem & Plant Resources West Ch,Kunming 650204,Peoples R China.;  liyanb@mail.kib.ac.cn;  zhanghbyd@gmail.com;  xdyang@ynu.edu.cn
Adobe PDF(670Kb)  |  收藏  |  浏览/下载:378/90  |  提交时间:2014/11/25
Indole  Imidazolium Salts  Structure-activity Relationships  Cell Apoptosis  
Aspergillines A-E, Highly Oxygenated Hexacyclic Indole-Tetrahydrofuran-Tetramic Acid Derivatives from Aspergillus versicolor 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 19, 页码: 5016-5019
作者:  Zhou, Min;  Miao, Ming-Ming;  Du, Gang;  Li, Xiao-Nian;  Shang, Shan-Zhai;  Zhao, Wei;  Liu, Zhi-Hua;  Yang, Guang-Yu;  Che, Chun-Tao;  Hu, Qiu-Fen;  Gao, Xue-Mei;  Hu,QF (reprint author),China Tobacco Yunnan Ind Co Ltd,Key Lab Tobacco Chem Yunnan Prov,Kunming 650231,Peoples R China.;  huqiufena@aliyun.com;  gao_xuemei@hotmail.com
Adobe PDF(277Kb)  |  收藏  |  浏览/下载:314/91  |  提交时间:2014/11/25
Cyclopiazonic Acid  Biological-activity  Biosynthesis  Flavus  
Synthesis, structure-activity relationships and biological evaluation of dehydroandrographolide and andrographolide derivatives as novel anti-hepatitis B virus agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 10, 页码: 2353-2359
作者:  Chen, Hao;  Ma, Yun-Bao;  Huang, Xiao-Yan;  Geng, Chang-An;  Zhao, Yong;  Wang, Li-Jun;  Guo, Rui-Hua;  Liang, Wen-Juan;  Zhang, Xue-Mei;  Chen, Ji-Jun
Adobe PDF(3861Kb)  |  收藏  |  浏览/下载:305/73  |  提交时间:2014/06/23
Anti-hbv Activity  DehydroAndrographolide And  Andrographolide Derivatives  Structure-activity Relationships  Octanol-water Partition Coefficients  
Palladium-Catalyzed Unactivated C(sp(3))-H Bond Activation and intramolecular Amination of Carboxamides: A New Approach to beta-Lactams 期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 2, 页码: 480-483
作者:  Sun, Wen-Wu;  Cao, Pei;  Mei, Ren-Qiang;  Li, Yue;  Ma, Yuan-Liang;  Wu, Bin
Adobe PDF(326Kb)  |  收藏  |  浏览/下载:622/62  |  提交时间:2014/04/09
C-h Activation  Carbon-hydrogen Bonds  Side-chain Sar  Acid Derivatives  Directing Group  Arylation  Functionalization  Inhibitors  Gamma  Construction  
Casuarines A and B, Lycopodium alkaloids from Lycopodium casuarinoides 期刊论文
TETRAHEDRON LETTERS, 2013, 卷号: 54, 期号: 34, 页码: 4555-4557
作者:  Liu, Fei;  Wu, Xing-De;  He, Juan;  Deng, Xu;  Peng, Li-Yan;  Luo, Huai-Rong;  Zhao, Qin-Shi
Adobe PDF(519Kb)  |  收藏  |  浏览/下载:267/48  |  提交时间:2013/10/16
Lycopodium Alkaloid  Lycopodium Casuarinoides  Casuarines a And b  Anti-ache Activity  
Swerpunilactones A and B, the first example of xanthone and secoiridoid heterodimers from Swertia punicea, S. hispidicalyx, and S. yunnanensis 期刊论文
TETRAHEDRON LETTERS, 2013, 卷号: 54, 期号: 21, 页码: 2710-2712
作者:  Wang, Hong-Ling;  Cao, Tuan-Wu;  Jiang, Fu-Qiang;  Geng, Chang-An;  Zhang, Xue-Mei;  Huang, Xiao-Yan;  Wang, Li-Jun;  Kang-He, Sing Wd;  Hao-Chen;  Liang, Wen-Juan;  Rong, Guang-Qing;  Chen, Ji-Jun
Adobe PDF(393Kb)  |  收藏  |  浏览/下载:498/140  |  提交时间:2013/06/08
Swerpunilactones A-b  Anti-hbv Activity  Swertia Punicea  Swertia Hispidicalyx  Swertia Yunnanensis  
Lycospidine A, a New Type of Lycopodium Alkaloid from Lycopodium complanatum 期刊论文
ORGANIC LETTERS, 2013, 卷号: 15, 期号: 10, 页码: 2438-2441
作者:  Cheng, Jin-Tang;  Liu, Fei;  Li, Xiao-Nian;  Wu, Xing-De;  Dong, Liao-Bin;  Peng, Li-Yan;  Huang, Sheng-Xiong;  He, Juan;  Zhao, Qin-Shi
Adobe PDF(448Kb)  |  收藏  |  浏览/下载:759/128  |  提交时间:2013/07/24
Inhibiting Acetylcholinesterase  A-c  Palhinhaea-cernua  Lycoposerramine-z  Huperzia-serrata  Biosynthesis  Casuarinoides  Intermediate  Pelletierine  Japonicum  
Griseusins F and G, Spiro-Naphthoquinones from a Tin Mine Tailings-Derived Alkalophilic Nocardiopsis Species 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2012, 卷号: 75, 期号: 11, 页码: 1994-1998
作者:  Ding, Zhang-Gui;  Zhao, Jiang-Yuan;  Li, Ming-Gang;  Huang, Rong;  Li, Qing-Ming;  Cui, Xiao-Long;  Zhu, Hua-Jie;  Wen, Meng-Liang
Adobe PDF(290Kb)  |  收藏  |  浏览/下载:573/112  |  提交时间:2013/01/22
Streptomyces-griseus  Biological-activity  Antibiotics  Pyranonaphthoquinones  Dihydrofusarubin  Configuration