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NaMLP, a new identified Kunitz trypsin inhibitor regulated synergistically by JA and ethylene, confers Spodoptera litura resistance in Nicotiana attenuata 期刊论文
PLANT CELL REPORTS, 2023
作者:  Yang,Mao;  Cheng,Junbin;  Yin,Min;  Wu,Jinsong
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Ethylene  Jasmonate  Miraculin-like protein  Nicotiana  Spodoptera  Trypsin protease inhibitor  BIOINSECTICIDAL ACTIVITY  PHYTOALEXIN SCOPOLETIN  PROTEINASE-INHIBITORS  ALTERNARIA-ALTERNATA  DEFENSE RESPONSES  JASMONATE  MIRACULIN  EXPRESSION  PATHWAYS  PERCEPTION  
Structurally Diverse Cytotoxic Polyphenols from Garcinia gracilis 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2023, 卷号: 86, 期号: 9, 页码: 2206-2215
作者:  Ye,Yan-Song;  Duan,Yao-Tao;  Zhou,Zhuo;  Thepkaysone,Khamphanh;  Douangdeuane,Bounleuane;  Xu,Gang
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CAGED XANTHONES  CONSTITUENTS  INHIBITORS  BENZOPHENONES  DERIVATIVES  BIPHENYL  TWIGS  
Discovery and Biomimetic Semisynthesis of Spirophyllines A-D from Uncaria rhynchophylla 期刊论文
ORGANIC LETTERS, 2023, 卷号: 25, 期号: 24, 页码: 4434-4438
作者:  Zhou,Hao-Feng;  Li,Wen-Yan;  Wu,Qi;  Ren,Jian;  Peng,Li-Yan;  Li,Xiao-Nian;  Zhao,Qin-Shi
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ATRIAL  INHIBITORS  CHANNELS  
Discovery of potential novel TRPC5 inhibitors by virtual screening and bioassay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 94, 页码: 117477
作者:  Shen,Meiling;  Li,Lingfeng;  Li,Yue;  Gu,Xi;  Bai,Longhui;  Xia,Chengfeng;  Xiong,Wenyong;  Zuo,Zhili
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TRPC5  Inhibitors  Virtual screening  Ca 2+channel  CHANNELS  IDENTIFICATION  PERMEABILITY  CALCIUM  
Abietane derived diterpenoids as Cav3.1 antagonists from Salvia digitaloides 期刊论文
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 4, 页码: 107737
作者:  Zhao,Jianjun;  Du,Shuzong;  Hu,Kun;  Hu,Yali;  Xia,Fan;  Ye,Yansong;  Yang,Jian;  Nian,Yin;  Xu,Gang
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10-Methylated 6  7  6 carbon ring system  Icetexane  Diterpenoid  Salvia digitaloides  Ca v 3  1 low voltage -gated Ca 2+channel  (LVGCC)  ROOTS  TANSHINLACTONE  CONSTITUENTS  ELUCIDATION  INHIBITORS  CHANNELS  SKELETON  SYSTEM  
Tissue-specific regulation of volatile emissions moves predators from flowers to attacked leaves 期刊论文
CURRENT BIOLOGY, 2023, 卷号: 33, 期号: 11, 页码: 2321-+
作者:  Munawar,Asim;  Xu,Yi;  Abou El-Ela,Amr S.;  Zhang,Yadong;  Zhong,Jian;  Mao,Zhiyao;  Chen,Xuan;  Guo,Han;  Zhang,Chao;  Sun,Yiqiao;  Zhu,Zengrong;  Baldwin,Ian T.;  Zhou,Wenwu
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BIOLOGICAL-CONTROL  INDIRECT DEFENSE  PLANT  EVOLUTION  HERBIVORY  BIOSYNTHESIS  POLLINATION  INHIBITORS  MUTUALISM  JASMONATE  
Bioassay-guided isolation of α-Glucosidase inhibitory constituents from Hypericum sampsonii 期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 6, 页码: 443-453
作者:  Tao,Linlan;  Xu,Shuangyu;  Zhang,Zizhen;  Li,Yanan;  Yang,Jue;  Gu,Wei;  Yi,Ping;  Hao,Xiaojiang;  Yuan,Chunmao
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Hypericum sampsonii  Chemical constituents  Structure elucidation  alpha-Glucosidase  Molecular docking  POLYCYCLIC POLYPRENYLATED ACYLPHLOROGLUCINOLS  POTENT INHIBITORS  SPECTROSCOPY  DERIVATIVES  CHEMISTRY  AMYLASE  ROOTS  
Oligomeric phloroglucinols with hAChE inhibitory and antibacterial activities from tropic Rhodomyrtus tomentosa 期刊论文
BIOORGANIC CHEMISTRY, 2023, 卷号: 141, 页码: 106836
作者:  Luo,E-E;  Liu,Si-Na;  Wang,Zhao-Jie;  Chen,Ling-Yun;  Liang,Cheng-Qin;  Yu,Mu-Yuan;  Qin,Xu-Jie
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Rhodomyrtus tomentosa  Oligomeric phloroglucinols  h AChE inhibitors  Molecular docking  Antibacterial effects  MYRTUCOMMULONE  DERIVATIVES  ACYLPHLOROGLUCINOLS  MYRTUCOMMUACETALONE  LEAVES  
Artemiprinolides A-M, thirteen undescribed sesquiterpenoid dimers from Artemisia princeps and their antihepatoma activity 期刊论文
PHYTOCHEMISTRY, 2023, 卷号: 211, 页码: 113714
作者:  Su,Li-Hua;  Ma,Wen-Jing;  Ma,Yun-Bao;  Li,Tian-Ze;  Geng,Chang-An;  Dong,Wei;  He,Xiao-Feng;  Chen,Ji-Jun
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Artemisia princeps Pamp  Sesquiterpenoid dimers  Artemiprinolides A-M  Antihepatoma activity  Apoptosis  FARNESYL-PROTEIN TRANSFERASE  ETHANOL EXTRACT  PAMPANINI  INHIBITORS  JACEOSIDIN  
先导化合物设计与开发 学位论文
: 中国科学院大学, 2022
作者:  Munikishore Rachakunta
Microsoft Word(14465Kb)  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/05/14
Buxus alkaloids  Buxus alkaloids  Cyclovirobuxine-D  Cyclovirobuxine-D  Synthesis, Calcium channel inhibitors  Synthesis, Calcium channel inhibitors  SAR studies  SAR studies  Anti-cardiovascular agents.  Anti-cardiovascular agents.