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Oxytocin inhibits the activity of acid-sensing ion channels through the vasopressin-1a receptor in primary sensory neurons1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-34
作者:  Fang Qiu;  Chun-Yu Qiu;  Huilan Cai;  Ting-Ting Liu;  Zu-Wei Qu;  Zhifan Yang;  Jia-Da Li;  Qun-Yong Zhou;  Wang-Ping Hu
Adobe PDF(850Kb)  |  收藏  |  浏览/下载:487/1  |  提交时间:2017/07/24
Oxytocin  Acid-sensing Ion Channel  Proton-gated Current  Vasopressin-1a Receptor  Dorsal Root Ganglion Neuron  Electrophysiology  Pain  
Pharmacology and anti-addiction effects of the novel kappa opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin A 期刊论文
出版物, 3111, 期号: 0, 页码: 1-53
作者:  B Simonson;  A S Morani;  A W M Ewald;  L Walker;  N Kumar;  D Simpson;  J H Miller;  T E Prisinzano;  B M Kivell
Adobe PDF(1394Kb)  |  收藏  |  浏览/下载:491/1  |  提交时间:2017/07/24
Pharmacological characterizationof tachykinin tetrabranched derivatives 期刊论文
出版物, 3111, 期号: 0, 页码: 1-36
作者:  Chiara Ruzza;  Anna Rizzi;  Davide Malfacini;  Maria Camilla Cerlesi;  Federica Ferrari;  Erika Marzola;  Caterina Ambrosio;  Cristina Gro;  Salvadori Severo;  Tommaso Costa;  Girolamo Calo;  Remo Guerrini
Adobe PDF(1277Kb)  |  收藏  |  浏览/下载:302/1  |  提交时间:2017/07/24
Tachykinins  Substance p  Pwt2-sp  Nk1 Receptor  Calcium Mobilization  Bioluminescence Resonance Energy Transfer  Guinea Pig Ileum  Rat Urinary Bladder  Nociceptive Behaviour Induced By Spinal Substance p  Mice  
Discovery of potentially biased agonists of mu-opioid receptor (MOR) through molecular docking, pharmacophore modeling, and MD simulation 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2021, 卷号: 90, 页码: 107405
作者:  Jiang,Xuan;  Li,Shuxiang;  Zhang,Hongbin;  Wang,Liang-Liang
浏览  |  Adobe PDF(6441Kb)  |  收藏  |  浏览/下载:426/50  |  提交时间:2022/04/02
mu-Opioid receptors (MOR)  Biased ligands  Molecular docking  Hip-hop pharmacophore  MD simulation  
Label-free cell phenotypic study of opioid receptors and discovery of novel mu opioid ligands from natural products 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2021, 卷号: 270, 页码: 113872
作者:  Hou,Tao;  Xu,Fangfang;  Peng,Xingrong;  Zhou,Han;  Zhang,Xiuli;  Qiu,Minghua;  Wang,Jixia;  Liu,Yanfang;  Liang,Xinmiao
收藏  |  浏览/下载:237/0  |  提交时间:2022/04/02
Opioid receptors  Dynamic mass redistribution  Natural products  Antagonist  Selectivity  IDENTIFICATION  ANTAGONISTS  SUBSTANCES  NALOXEGOL  AGONISTS  SAFETY  MACA  
Identification of novel phytocannabinoids from Ganoderma by label-free dynamic mass redistribution assay 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2020
作者:  Zhou, Han;  Peng, Xingrong;  Hou, Tao;  Zhao, Nan;  Qiu, Minghua;  Zhang, Xiuli;  Liang, Xinmiao
浏览  |  Adobe PDF(3740Kb)  |  收藏  |  浏览/下载:303/78  |  提交时间:2021/01/05
Homology modeling and 3D-QSAR study of benzhydrylpiperazine delta opioid receptor agonists 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2019, 卷号: 83, 页码: 9
作者:  Pan, Chenling;  Meng, Hao;  Zhang, Shuqun;  Zuo, Zhili;  Shen, Yuehai;  Wang, Liangliang;  Chang, Kwen-Jen
浏览  |  Adobe PDF(1542Kb)  |  收藏  |  浏览/下载:598/113  |  提交时间:2020/03/18
delta opioid receptor agonists  3D-QSAR  Homology modeling  Molecular dynamics simulation  Molecular docking  
The opioid receptor triple agonist DPI-125 produces analgesia with less respiratory depression and reduced abuse liability 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 7, 页码: 977-989
作者:  Yi, Shou-pu;  Kong, Qing-hong;  Li, Yu-lei;  Pan, Chen-ling;  Yu, Jie;  Cui, Ben-qiang;  Wang, Ying-fei;  Wang, Guan-lin;  Zhou, Pei-lan;  Wang, Li-li;  Gong, Ze-hui;  Su, Rui-bin;  Shen, Yue-hai;  Yu, Gang;  Chang, Kwen-jen
浏览  |  Adobe PDF(854Kb)  |  收藏  |  浏览/下载:568/132  |  提交时间:2017/08/29
Opioid Receptor  Mixed Agonist  Dpi-125  Analgesia  Respiratory Depression  Addiction  
Cognitive-enhancing effects of beta-sitosterol in vanadium-induced neurotoxicity in mice 期刊论文
JOURNAL OF NEUROCHEMISTRY, 2017, 卷号: 142, 页码: 238-238
作者:  Adebiyi,O.;  Olayemi,F.;  Olopade,J.;  Ning-Hua,T.
浏览  |  Adobe PDF(878Kb)  |  收藏  |  浏览/下载:391/143  |  提交时间:2017/10/23
阿片受体三重激动剂KUST201的大鼠镇痛、耐受与戒断反应研究 期刊论文
中国药理学通报, 2016, 期号: 5, 页码: 652-658
作者:  李玖玲;  孔庆宏;  郁洁;  伊首璞;  李亚民;  王冠林;  沈悦海;  张宽仁
浏览  |  Adobe PDF(445Kb)  |  收藏  |  浏览/下载:359/109  |  提交时间:2016/12/19
Kust201  Dpi-125  镇痛  耐受  戒断  阿片受体三重激动剂