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An efficient and concise synthesis of a selective small molecule non-peptide inhibitor of cathepsin L: KGP94 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 105317
作者:  Munikishore,Rachakunta;  Wang,Liang-Liang;  Zhang,Shuqun;  Zhao,Qin-Shi;  Zuo,Zhili
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Cathepsin L  small-molecule inhibitor  gram-scale synthesis  KGP94  cancer  FUNCTIONALIZED BENZOPHENONE  BIOLOGICAL EVALUATION  TUMOR PROGRESSION  CELL INVASION  EXPRESSION  ANALOGS  SUPPRESSION  DERIVATIVES  ACID  
(-)-Isoscopariusin A, a Naturally Occurring Immunosuppressive Meroditerpenoid: Structure Elucidation and Scalable Chemical Synthesis 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 卷号: 60, 期号: 23, 页码: 12859-12867
作者:  Yan,Bing-Chao;  Zhou,Min;  Li,Jian;  Li,Xiao-Nian;  He,Shi-Jun;  Zuo,Jian-Ping;  Sun,Han-Dong;  Li,Ang;  Puno,Pema-Tenzin
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bioactivity  cyclobutane  natural products  scalable synthesis  structure elucidation  
Academician Qi-Yi Xing (Chi-Yi Hsing): pioneer organic chemist of synthetic insulin 期刊论文
PROTEIN & CELL, 2021
作者:  Qiu,Ming-Hua
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Ir-Catalyzed Asymmetric Total Syntheses of Bisdehydrotuberostemonine D, Putative Bisdehydrotuberostemonine E and Structural Revision of the Latter 期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2021, 卷号: 143, 期号: 49, 页码: 20622-20627
作者:  Deng,Yi;  Liang,Xiao;  Wei,Kun;  Yang,Yu-Rong
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ENANTIOSELECTIVE TOTAL-SYNTHESIS  ALDEHYDE OXIDATION LEVEL  UNIFIED TOTAL-SYNTHESIS  STEMONA ALKALOIDS  CARBONYL ALLYLATION  ALPHA-ALLYLATION  IRIDIUM  ALCOHOL  TUBEROSTEMONINE  HYDROGENATION  
Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:  Zhou, Yeheng;  Sun, Wei;  Peng, Jiale;  Yan, Hui;  Zhang, Li;  Liu, Xingyong;  Zuo, Zhili
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Acetylcholinesterase  Drug design  N-acylhydrazone  Dementia  Copper-chelating  N-Benzylpiperidine  
Total Synthesis of (+/-)-Cochlearol A 期刊论文
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 17, 页码: 6761-6764
作者:  Zhang, Da-Wei;  Xu, Wen-Dan;  Fan, Hui-Lan;  Liu, Hao-Miao;  Chen, Dong;  Liu, Dan-Dan;  Qin, Hong-Bo
浏览  |  Adobe PDF(999Kb)  |  收藏  |  浏览/下载:331/54  |  提交时间:2019/10/28
中性烯烃与α、β-不饱和亚胺构建含氮杂环体系 学位论文
硕士: 中国科学院昆明植物研究所, 2019
作者:  孙柔婧
Adobe PDF(8220Kb)  |  收藏  |  浏览/下载:176/0  |  提交时间:2022/08/29
α  β-不饱和亚胺  中性烯烃  环加成反应  Lewis酸催化  含氮杂环  
Synthesis of 2,6-dimethoxy-9-phenyl-1H-phenalen-1-one and structural revision of the benzoindenone from Eichhornia crassipes 期刊论文
, 2019
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浏览  |  Adobe PDF(228Kb)  |  收藏  |  浏览/下载:179/65  |  提交时间:2020/04/02
吡啶盐的脱氢偶联反应研究 学位论文
博士, 2018
作者:  尚文斌
Microsoft Word(37803Kb)  |  收藏  |  浏览/下载:71/0  |  提交时间:2021/01/05
Transition-metal-free dehydrogenation coupling of pyridinium through a self-promoted hydride transfer process 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2017, 卷号: 4, 期号: 9, 页码: 1789-1793
作者:  Shang, Wenbin;  Li, Shanyong;  Ding, Yuzhen;  Pan, Zhiqiang;  Tong, Xiaogang;  Xia, Chengfeng
浏览  |  Adobe PDF(634Kb)  |  收藏  |  浏览/下载:369/79  |  提交时间:2017/10/23
C-h Functionalization  Hydrogen Evolution Reaction  Nickel/lewis Acid Catalysis  Visible-light Catalysis  Quinoline N-oxides  Direct Arylation  Bond Activation  Selective Alkenylation  Grignard-reagents  Dft Calculations