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Oxytocin inhibits the activity of acid-sensing ion channels through the vasopressin-1a receptor in primary sensory neurons1 期刊论文
出版物, 3111, 期号: 0, 页码: 1-34
作者:  Fang Qiu;  Chun-Yu Qiu;  Huilan Cai;  Ting-Ting Liu;  Zu-Wei Qu;  Zhifan Yang;  Jia-Da Li;  Qun-Yong Zhou;  Wang-Ping Hu
Adobe PDF(850Kb)  |  收藏  |  浏览/下载:251/1  |  提交时间:2017/07/24
Oxytocin  Acid-sensing Ion Channel  Proton-gated Current  Vasopressin-1a Receptor  Dorsal Root Ganglion Neuron  Electrophysiology  Pain  
The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1 期刊论文
出版物, 2111, 页码: 1-44
作者:  1M S Grace;  T Lieu;  B Darby;  F C Abogadie;  N Veldhuis N W Bunnett;  P McIntyre
Adobe PDF(1611Kb)  |  收藏  |  浏览/下载:109/1  |  提交时间:2017/07/24
Transient Receptor Potential Ion Channel  Trpv4  Protease Activated Receptor  Par2  Pain  Tyrosine Kinase  Bafetinib  
Discovery of novel modulators targeting human TRPC5: Docking-based virtual screening, molecular dynamics simulation and binding af fi nity predication 期刊论文
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2021, 卷号: 102, 页码: 107795
作者:  Liu,Bin;  Zhang,Wei;  Guo,Sheng;  Zuo,Zhili
Adobe PDF(4277Kb)  |  收藏  |  浏览/下载:80/10  |  提交时间:2022/04/02
hTRPC5  Homology modeling  Molecular docking  Molecular dynamics simulation  Virtual screening  INHIBITOR  CHANNELS  GROMACS  POTENT  AMBER  IDENTIFICATION  CONSTRAINTS  INTEGRATION  AMYGDALA  
吴茱萸次碱抗急性白血病活性评价 学位论文
硕士, 2018
作者:  龚亮
Adobe PDF(4427Kb)  |  收藏  |  浏览/下载:35/0  |  提交时间:2021/01/05
紫金龙等五种药用植物异喹啉和吲哚结构及生物活性研究 学位论文
: 中国科学院大学, 2017
作者:  王蓓
Adobe PDF(5603Kb)  |  收藏  |  浏览/下载:264/14  |  提交时间:2019/06/14
Pyrazolopyrimidines as Potent Stimulators for Transient Receptor Potential Canonical 3/6/7 Channels 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 11, 页码: 4680-4692
作者:  Qu, Chunrong;  Ding, Mingmin;  Zhu, Yingmin;  Lu, Yungang;  Du, Juan;  Miller, Melissa;  Tian, Jinbin;  Zhu, Jinmei;  Xui, Jian;  Wen, Meng;  Er-Bu, Aga;  Wan, Jule;  Xiao, Yuling;  Wu, Meng;  McManus, Owen B.;  Li, Min;  Wu, Jilin;  Luo, Huai-Rong;  Cao, Zhengyu;  Shen, Bing;  Wang, Hongbo;  Zhu, Michael X.;  Hong, Xuechuan
浏览  |  Adobe PDF(1969Kb)  |  收藏  |  浏览/下载:207/77  |  提交时间:2017/08/29
Cognitive-enhancing effects of beta-sitosterol in vanadium-induced neurotoxicity in mice 期刊论文
JOURNAL OF NEUROCHEMISTRY, 2017, 卷号: 142, 页码: 238-238
作者:  Adebiyi,O.;  Olayemi,F.;  Olopade,J.;  Ning-Hua,T.
浏览  |  Adobe PDF(878Kb)  |  收藏  |  浏览/下载:149/65  |  提交时间:2017/10/23
顺式-5'-(2-氧代丙基)-烟碱的化学结构和生物活性 期刊论文
中国中药杂志, 2016, 期号: 4, 页码: 689-693
作者:  杨彩艳;  黄晓燕;  马云保;  耿长安;  张雪梅;  陈纪军
浏览  |  Adobe PDF(568Kb)  |  收藏  |  浏览/下载:260/46  |  提交时间:2016/12/19
顺式-5'-羰丙基烟碱  化学成分  生物活性  普通烟草  
The role of targeting kinase activity by natural products in cancer chemoprevention and chemotherapy (Review) 期刊论文
ONCOLOGY REPORTS, 2015, 卷号: 34, 期号: 2, 页码: 547-554
作者:  Luo, Xiangjian;  Yu, Xinfang;  Liu, Sufang;  Deng, Qipan;  Liu, Xiaolan;  Peng, Songling;  Li, Hongde;  Liu, Jikai;  Cao, Ya
Adobe PDF(755Kb)  |  收藏  |  浏览/下载:339/168  |  提交时间:2015/12/17
Natural Products  Grifolin  Neoalbaconol  Epigallocatechin-3-gallate  Cancer Prevention  
Identification and optimization of 2-aminobenzimidazole derivatives as novel inhibitors of TRPC4 and TRPC5 channels 期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2015, 卷号: 172, 期号: 14, 页码: 3495-3509
作者:  Zhu, Yingmin;  Lu, Yungang;  Qu, Chunrong;  Miller, Melissa;  Tian, Jinbin;  Thakur, Dhananjay P.;  Zhu, Jinmei;  Deng, Zixin;  Hu, Xianming;  Wu, Meng;  McManus, Owen B.;  Li, Min;  Hong, Xuechuan;  Zhu, Michael X.;  Luo, Huai-Rong
Adobe PDF(2298Kb)  |  收藏  |  浏览/下载:191/47  |  提交时间:2015/12/15