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Discovery and structure-activity relationships of ent-Kaurene diterpenoids as potent and selective 11 beta-HSD1 inhibitors: Potential impact in diabetes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 403-414
作者:  Deng, Xu;  Shen, Yu;  Yang, Jing;  He, Juan;  Zhao, Yu;  Peng, Li-Yan;  Leng, Ying;  Zhao, Qin-Shi
浏览  |  Adobe PDF(1215Kb)  |  收藏  |  浏览/下载:409/153  |  提交时间:2013/10/16
Ent-kaurene Diterpenoids  Structure-activity Relationship Studies  Selective 11 Beta-hsd1 Inhibitors  Urea Derivatives  Diabetes  
Discovery of natural estrogen receptor modulators with structure-based virtual screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 卷号: 23, 期号: 11, 页码: 3329-3333
作者:  Cao, Xianwen;  Jiang, Jing;  Zhang, Shoude;  Zhu, Lili;  Zou, Juan;  Diao, Yanyan;  Xiao, Weilie;  Shan, Lei;  Sun, Handong;  Zhang, Weidong;  Huang, Jin;  Li, Honglin
浏览  |  Adobe PDF(911Kb)  |  收藏  |  浏览/下载:337/98  |  提交时间:2013/07/24
Molecular Docking  Natural Product  Estrogen Receptor  Virtual Screening